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Matches 1 - 50 out of 15,130

Document Document Title
WO/2018/010965A1
Embodiments of the invention are directed to new equatorially modified polymer linked multimers of guanosine-3', 5'-cyclic monophosphate (cGMP) analogues that inhibit the cGMP-signaling system. The invention is also directed to related m...  
WO/2018/008727A1
The present invention provides a heterocyclic compound that exhibits a superior control against harmful arthropods and that is represented by formula (I): (I) [in the formula, Q1 represents an oxygen atom or the like; Q2 represents an ox...  
WO/2018/003924A1
Provided is a novel pest control agent, especially a bactericide or a nematicide. An alkynylpyridine-substituted amide compound represented by formula (I) or a salt thereof; and a pest control agent which contains the compound or the sal...  
WO/2018/003976A1
In agricultural and horticultural crop production, etc., damage by pests and the like remains devastating even today, and due to factors such as the occurrence of pests resistant to existing chemicals, there is a demand for the developme...  
WO/2017/220517A1
The invention relates to a compound of formula (I) wherein R1 to R4 and n are defined as in the description and in the claims. The compound of formula (I) can be used as a medicament.  
WO/2017/221158A1
The present invention relates to a nanoparticle composition comprising one or more β-triketones selected from leptospermone, isoleptospermone, grandiflorone and flavesone, together with a carrier.  
WO/2017/222996A1
Provided herein are compounds, compositions and method of using thereof to treat or prevent malaria.  
WO/2017/214683A1
The present invention provides a method for the treatment or prophylaxis of an ectoparasitic infestation, the method comprising the step of: contacting an external surface of an animal in need thereof with an effective amount of a berber...  
WO/2017/211909A1
The invention concerns a lipid composition that is self-emulsifying in the presence of a hydrophilic phase, comprising between 0.001% and 20% by weight, relative to the total weight of the composition, of at least one active substance; b...  
WO/2017/212239A1
The present invention provides a sulphur-containing compound for use in the prophylaxis or treatment of an infection associated with at least one microbe or microbial strain displaying at least some degree of drug resistance. Also provid...  
WO/2017/214076A1
The present invention describes rhomboid protease inhibitors having high specificity and inhibition characteristics providing novel antibiotics, anti-malarial pharmaceutical agents, and provides a strategy for designing RiBns (rhomboid-i...  
WO/2017/210262A1
The present invention targets the Zika virus and other disease-causing microbes including viruses, bacteria, fungi, and parasites. It does this using agents and methods with little toxicity compared to existing therapies.  
WO/2017/205464A1
Disclosed are compounds of Formula (I), methods of using the compounds as immunomodulators, and pharmaceutical compositions comprising such compounds. The compounds are useful in treating, preventing or ameliorating diseases or disorders...  
WO/2017/198178A1
A thiazole derivative serving as a DHODH inhibitor, and applications thereof. The present invention specifically relates to a compound represented by formula I, a pharmaceutical composition containing the compound represented by formula ...  
WO/2017/195069A1
The present invention provides oxaborole ester compounds and compositions thereof which are useful to treat diseases associated with parasites, such as Chagas Disease and African Animal Trypanosomosis.  
WO/2017/195136A1
The invention relates to novel N-(α-peroxy)indole compounds of Formula I and methods for use. (I) The N-(α-peroxy)indole compounds described herein are useful for treating or preventing parasitic infections, bacterial infections, and c...  
WO/2017/195138A1
The invention relates to novel N-(α-peroxy)carbazole compounds of Formula I and methods for use. (I) The N-(α-peroxy)carbazole compounds described herein are useful for treating or preventing parasitic infections, bacterial infections,...  
WO/2017/193017A1
The present disclosure relates generally to the field of antimicrobial compounds and to methods of making and using them. These compounds are useful for treating, preventing, reducing the risk of, and delaying the onset of microbial infe...  
WO/2017/191138A1
Compositions and methods for treating and preventing crustacean ectoparasitesinfection of fish are disclosed herein.  
WO/2017/192385A1
The present invention provides compounds of the formula : (I) wherein: X is O or S; Q1 and Q2 are independently CR5 or N, provided at least one of Q1 and Q2 is N; Y is a direct bond or CH2; R1 is H, optionally substituted alkyl, alkenyl,...  
WO/2017/186182A1
Provided herein is a humanized anti-BASIGIN antibody or antigen binding fragment thereof, which comprises heavy chain variable region(V H) comprising an amino acid sequence of SEQ ID NO:1, optionally further comprises light chain variabl...  
WO/2017/184456A1
Disclosed herein are polynucleotides encoding multi-epitope polypeptides and assemblies thereof, and their use for treating or limiting Toxoplasma gondii infection.  
WO/2017/184537A1
Compositions suitable for topical use to treat ectoparasite infestations are described. The compositions are suitable for use on the hair of humans or animals, without the need for pharmaceuticals or medicaments. The compositions are ess...  
WO/2017/177292A3
The present invention relates to a method for the selective control of populations of hematophagic arthropods, replacing or supplementing the use of pyrethroid insecticides by the use of tyrosine metabolism enzyme inhibitors, more specif...  
WO/2017/178524A1
The present invention relates to a process for the preparation of pyrvinium pamoate, which comprises reacting pyrvinium methyl sulphate salt of formula (II) with disodium pamoate of formula (III), in the presence of a base; to processes ...  
WO/2017/177433A1
The present invention provides a pharmaceutical composition for killing ectoparasites of animals. The pharmaceutical composition contains an active ingredient and monoester; the active ingredient comprises at least one of albendazole, am...  
WO/2017/178416A1
The present invention covers Pyrazolopyrimidine compounds of general formula (I), in which n, o, X, Y, R, Q, R1, R2, R3 and R4 are as defined herein, methods of preparing said compounds, intermediate compounds useful for preparing said c...  
WO/2017/176762A1
The disclosure provides, among other things, compositions that bind to and inhibit the biological activity of soluble biomolecules, as well as pharmaceutical compositions thereof. The compositions may comprise a plurality of particles th...  
WO/2017/173956A1
A compound represented by formula (I) for preventing and treating human or animal parasitic infection, wherein the R group is either a -CH3 or -C2H5 group; the R group is -CH3 in tenvermectin A and is -C2H5 in tenvermectin B. Both of the...  
WO/2017/176948A1
This invention relates to processes for the preparation of antiparasitic isoxazoline compounds enriched in an enantiomer using quinine- based chiral phase transfer catalysts. The invention also relates to novel quinine-based phase transf...  
WO/2017/174620A1
The present invention relates to compounds of formula (I) and salts thereof, pharmaceutical compositions containing such compounds and to their use in therapy.  
WO/2017/168476A1
An object of the present invention is to provide a novel anti-Tritrichomonas agent. Provided is an anti-Tritrichomonas agent containing luliconazole.  
WO/2017/173049A1
The present invention relates to compounds, and pharmaceutically acceptable compositions thereof, useful as inhibitors of cyclophilins, and for the treatment of cyclophilin-related disorders.  
WO/2017/173048A1
The present invention relates to compounds, and pharmaceutically acceptable compositions thereof, useful as inhibitors of cyclophilins, and for the treatment of cyclophilin- related disorders.  
WO/2017/173052A1
The present invention relates to compounds, and pharmaceutically acceptable compositions thereof, useful as inhibitors of cyclophilins, and for the treatment of cyclophilin-related disorders.  
WO/2017/170712A1
The present invention addresses the problem of providing a chemosynthetic adjuvant for selectively inducing TSLP. The present invention provides a vaccine adjuvant including a RAR γ agonist, and a vaccine obtained by combining the vacci...  
WO/2017/170970A1
A composition for controlling microsporidia in fishes is prepared by using, as an active ingredient, at least one kind of compound selected from the group consisting of a compound represented by general formula (I) [wherein R2, R4, R5, R...  
WO/2017/163171A1
The present invention relates to a vaccine composition based on a recombinant polypeptide chimera composed of specific epitopes of human and mice CD4+ and CD8+ T lymphocytes derived from four Leishmania proteins (LiHypl, LiHyp6, LiHyV an...  
WO/2017/164108A1
The compound according to the present invention, represented by formula (1) [where A1 represents a nitrogen atom or CR4, R4 representing a hydrogen atom or the like, any one of A2, A3, and A4 represents a nitrogen atom and the remainder ...  
WO/2017/163181A1
The present invention relates to a vaccine composition composed of two immnogenic proteins defined by SEQ ID No. 1 and 2, and to the use thereof for treating and/or preventing canine and human cutaneous and visceral leishmaniasis.  
WO/2017/159618A1
The purpose of the present invention is to provide a compound having a high activity against pests. The present invention provides: a substituted pyridine compound represented by formula (I) [wherein R1 represents an alkyl group or the l...  
WO/2017/159759A1
[Problem] The present invention addresses the problem of providing an additive and feed for controlling fish parasitic diseases in the culture of fish, said additive and feed being characterized by characterized by containing β-1,4-mann...  
WO/2017/161387A1
Synthetic drug development is slow and costly, often running into the billions of dollars. While the benefits of various abundant and inexpensive natural products, including natural oils and extracts, have been postulated and speculated ...  
WO/2017/157899A1
The present invention relates to antisense oligonucleotides that are capable of reducing expression of PD-L1 in a target cell. The oligonucleotides hybridize to PD-L1 mRNA. The present invention further relates to conjugates of the oligo...  
WO/2017/155103A1
Provided is a novel pest control agent, particularly a pesticide or a miticide. A condensed heterocyclic compound represented by formula (1), a salt of the compound, or an N-oxide of the compound or the salt. [Q represents a structure re...  
WO/2017/155465A1
The present invention provides a compound belonging to furanocoumarin derivative having core structure (A) as given below, its pharmaceutically acceptable salt, isomer or a combination thereof for the treatment and/or prevention of a par...  
WO/2017/150174A1
Provided is a pharmaceutical composition for the treatment or prevention of Plasmodium diseases, the pharmaceutical composition being characterized by containing at least one quinazoline derivative represented by general formula (I) or a...  
WO/2017/146226A1
The present invention addresses the problem of developing and providing a novel agricultural/horticultural insecticide in view of the fact that, in crop production, such as agriculture and horticulture, damage by harmful insects, etc., i...  
WO/2017/146221A1
The present invention addresses the problem of developing and providing a novel agricultural/horticultural insecticide in light of factors in agricultural and horticultural crop production such as the damage caused by harmful insects, wh...  
WO/2017/144517A1
A series of 3-imino-5-methyl-1,2,4-thiadiazinane 1,1-dioxide derivatives of formula (I), substituted in the 5-position by a phenyl moiety which in turn is meta-substituted by an optionally substituted fused bicyclic heteroaromatic ring s...  

Matches 1 - 50 out of 15,130