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JP2018501270A |
The present invention is (3RS) *3* [(2SR) * (2* cyclopentyl *2* hydroxy *2* phenylacetyl) Oxy ] *1 and 1* Dimethyl pyridinium . Star's picture, It is suitable for production on an industrial scale, is further obtained in quantity yield a...
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JP2018500326A |
(R) Anhydride of *2* hydroxy *2* methyl *4* (2, 4, 5* Trimethyl *3, 6* dioxo cyclohexa *1, 4* dienyl) butaneamide, The method of using the constituent for the disposal of the polymorphism form of a hydrate and solvent Japanese food , an ...
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JP6255343B2 |
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JP6234999B2 |
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JP6234030B2 |
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JP6231151B2 |
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JP6226318B2 |
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JP2017529323A |
The present invention relates to a method for chiral resolution of a chiral kind contained in a fluid arranged in a cell formed of an inner wall and an outer wall surrounding an inner wall over at least one copy of an inner wall, Each of...
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JP6176259B2 |
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JP2017132793A |
To provide a novel process for the synthesis of R-biphenylalaninol and its intermediates useful in the synthesis of pharmaceutically active compounds.The present invention provides a process for obtaining a compound of formula I by Boc-p...
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JP2017128528A |
To provide a method for producing an (S)-2-hydroxypropanoic acid derivative and ambrisentan having high optical purity in an industrially advantageous manner.There is provided a method for producing an (S)-2-hydroxypropanoic acid derivat...
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JP2016523241A5 |
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JP2016528180A5 |
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JPWO2015118793A1 |
A manufacturing method of out (R) *1 including following process (A), (B), and (C), 1, and 3* Trimethyl *4* amino in. (A) : Optical division of out 1, 1, and 3* Trimethyl *4* amino in is carried out, (R) Process (B) which obtains out 3 [...
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JPWO2015064453A1 |
the present invention has a thiol group in a side chain -- optics -- it made into a subject to provide a method of manufacturing active D* object and/or L* object amino acid with sufficient yield by a simple method. The present invention...
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JP6086512B2 |
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JP6087504B2 |
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JPWO2014157607A1 |
optics useful as a manufacturing raw material of medicine, agricultural chemicals, and an industrial commodity -- the optical purity improving method of active 2* hydroxycarboxylic acid is provided. Hydroxycarboxylic acid denoted by the ...
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JPWO2014148344A1 |
The present invention is a manufacturing method of optical activity transformer 1, optical activity transformer 1 which makes it Crystallization from solution of 2* Diamino cyclohexane, and obtains a crystal of optical activity transform...
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JPWO2014125667A1 |
The present invention provides an optical isomer separating medium and a manufacturing method for the same. That is, the present invention is following formula (I) : Each sign in [type is as given in a specification. A spiral poly (diphe...
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JPWO2014119731A1 |
By non- A conversion reaction of L* isoleucine, a method of manufacturing D* alloisoleucine by a short process and quantity yield is provided. To the specific system of reaction in the state where L* isoleucine and D* alloisoleucine Epim...
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JP2017502020A |
Formula (1) [Formula 1] It is Of compound and they are inside of a formula, and R.1A Is hydrogen , Halo , C1*C4 Alkyl machine, C1*C4 Alkyl halide machine, and C1*C4 alkoxy *C2*C4 Alkyl machine, C2*C4 alkenyl group, C2*C4 alkynyl group, o...
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JP2016539924A |
Formula (I) [Formula 1] (The inside of a formula, X, R)1*R7It has a meaning defined as a The book specification. HBV replication inhibitor which is of HBV replication inhibitor and contains the stereochemical opposite-sex form, salt, a h...
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JP6045531B2 |
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JP6023794B2 |
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JP2016164191A |
To provide a method for producing a high-quality optically active thiazolylalanine derivative and salt thereof, in which the method does not require the use of any unsafe reagent and is economically advantageous, and is suitable for the ...
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JP5986380B2 |
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JP2016155849A |
To provide methods for producing substituted heterocycle fused gamma-carbolines, intermediates useful in producing them, methods for producing such intermediates and such heterocycle fused gamma-carbolines.The invention provides compound...
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JP5981719B2 |
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JP5968439B2 |
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JP5951825B2 |
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JP2016065046A |
To provide an industrial method for producing (2S,12Z)-2-acetoxy-12-heptadecene which is a sexual pheromone of pistachio twig borer.The present invention can provide a production method and the like including at least the steps of: react...
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JP2016065024A |
To provide a method for optical resolution of carboxylic acid.Provided is a method for optical resolution of carboxylic acid in which (S)-3-cyclohexene-1-carboxylic acid represented by the chemical structure of the left side in formula (...
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JP5901292B2 |
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JP2015505827A5 |
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JP2016040282A |
To provide methods for production of cyclopropyl ring-fused pyrrolidine compounds of dipeptidyl peptidase IV inhibitors.The present invention provides a method for production of a free base compound represented by formula M'.SELECTED DRA...
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JP5888993B2 |
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JP2014525895A5 |
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JPWO2013154066A |
a subject of the present invention -- optics -- it is manufacturing an active bicyclic compound efficiently. enzyme -- optics -- an active bicyclic compound is manufactured efficiently.
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JP2014530809A5 |
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JP2015526384A |
[Subject] Offer of a new manufacturing method of a stereoselective epoxy ketone compound. [Means for Solution] A manufacturing method of an epoxy ketone compound denoted by a formula (1) denoted by the following scheme. Thereby, an epoxy...
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JP2015129121A |
To provide a method for obtaining a dihydro-1,3,5-triazine amine derivative useful as a pharmaceutical composition in a high yield and high excess enantiomorph ratio.There is provided a method for separating an enantiomer of a dihydro-1,...
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JP5744076B2 |
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JP5743595B2 |
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JP5738204B2 |
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JP5734533B2 |
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JP2015091886A |
To provide an alternative preparation method for amino acid derivatives.An improved method of producing lacosamide (LCM), or (R)-2-acetamido-N-benzyl-3-methoxypropion-amide, useful as an anticonvulsant agent is provided. In a specific em...
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JP5714213B2 |
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JPWO2013089188A |
carrying out optical division using optical activity amine -- optics -- an active bicyclic compound is manufactured efficiently.
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JP2015509496A |
It is provided for this specification, The unusually high level, the disease related as it is active, or state of TNF-alpha is treated or prevented. It is a new preparing method of the amino sulfone intermediate for composition of useful...
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