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Matches 751 - 800 out of 4,296

Document Document Title
JP2014172839A
To provide a process for producing a tertiary alcohol derivative of high optical purity from a racemic tertiary alcohol derivative or a tertiary alcohol derivative of low optical purity.Provided is a method for producing an optically act...  
JP2014172856A
To produce a high-purity optically active tetrahydrofuran-2-carboxylic acid having optical activity efficiently with high productivity.There is provided a method for producing a high-purity (R)- or (S)-tetrahydrofuran-2-carboxylic acid, ...  
JP2014169252A
To provide a new method of producing optically active β-formyl-β-hydroxy-α-substituted aldehyde compounds.A method of producing an optically active β-formyl-β-hydroxy-α-substituted aldehyde compound (2) includes the step of making ...  
JP2014523896A
The present invention relates to the new nitryl compound shown in formulas I and II. (I) Formula I(The inside of a formula and X are *CH (s).)3Or it is *C≡N. (II) Formula II(The inside of a formula and X are *CH (s).)3Or as for R, Y is...  
JP2014169294A
To provide an optically active piperidine derivative which is excellent in antihistaminic activity and antiallergic activity, has little hygroscopicity and is excellent in physicochemical stability, and a manufacturing method thereof.Thi...  
JP2014523416A
The present invention relates to the medicine constituent which has the antiviral activity which contains 1, 3* dioxo indene derivative, its salt permitted pharmacologically or an optical isomer, its preparing method, and it as an active...  
JP5585822B2  
JP2014152156A
To provide a method for obtaining an optically active material, when erythro ADPE or MA is used as a reagent for optical resolution, having a sign opposite to the previously obtained one without forming a diastereomeric salt again.To pro...  
JP2014148531A
To provide, among other things, novel compounds useful for treating bacterial infections, pharmaceutical compositions containing such compounds, as well as combinations of these compounds with at least one additional therapeutically effe...  
JP2014520077A
Improved stabilityIt has. (4S, 4aS, 5aR, 12aS) -4-dimethylamino 3, The crystalline mono-chloride salt of 10, 12, and 12a-tetra-hydroxy 7- [(methoxy (methyl) amino) - methyl] -1 and 11-dioxo 1, 4, 4a, 5, 5a, 6, and 11 and 12a-octahydro NA...  
JP2014520140A
Deuteration 1* piperazino *3* phenyl * Indang where the present invention has activity in dopamine receptors D1 and D2 of a central nervous system, and 5HT2 receptor, and its salt, It is related with a therapeutic method including use of...  
JP2014520126A
The present invention is a new method for manufacture of ソリフェナシン or its acid addition salt permitted pharmacologically, and is the bottom of existence of acid, and (R) * quinuclidine *3* イル. Reaction of フェネチル ...  
JP5566103B2  
JP5563830B2  
JP2014133771A
To provide processes and intermediates for the preparation of 3-benzazepines and salts thereof which can be useful as serotonin (5-HT) receptor agonists for the treatment of, for example, central nervous system disorders such as obesity....  
JP5553911B2  
JP5557292B2  
JP2014516920A
The present invention relates to those use as *4* cyano *3 replaced (3R, 4R), 4* diphenyl butanoic acid compounds, those manufacturing methods, a weed killer, and a plant growth regulation agent. The compound of formula (I) in an optical...  
JP5552422B2  
JP5544298B2  
JP2014122211A
To provide an GPR40 activator containing a compound having a novel GPR40 agonist effect or a salt thereof or a solvate thereof and the like as an active ingredient, especially an insulin secretion promoter, a prevention and/or therapeuti...  
JP5534460B2  
JP5536869B2  
JP5531097B2  
JP5533654B2  
JP5531288B2  
JP2014514243A
2R*2* (N, N dimethylamino) * propionic acid ドデシル (R*DDAIP), The activity unexpectedly improved in passing a biomembrane and an organization and easy-izing transportation of an active compound pharmacologically as compared with S*...  
JP5520077B2  
JP5518337B2  
JP5513621B2  
JP5510040B2  
JP5514549B2  
JP5503546B2  
JP2014088389A
To provide a diagnostic agent for positron emission tomography, comprising a [F-18]-labeled compound.A diagnostic agent for positron emission tomography (PET) comprises a compound which is a L-glutamic acid or L-glutamic acid derivative ...  
JP5487440B2  
JP2014074033A
To provide methods for isolating from a reaction mixture a salt of a mono-propargylated aminoindane (rasagiline), which is a selective inhibitor of MAO-B and useful in treating Parkinson's disease etc.Disclosed are production methods for...  
JP5476859B2  
JP2014509592A
The present invention provides the compound of formula (I), this salt permitted as medicine, a prodrug, a biological activity metabolite, a stereoisomeric form, and an opposite-sex object, and the variable thing is defined in this specif...  
JP2014509304A
The present invention experiences the new method for manufacturing Sis *1* ammonium *4* alkoxy cyclohexane カルボ nitril salts, and the manufacturing method by the present invention, or relates to the new intermediate output or the st...  
JP5468003B2  
JP5456871B2  
JP5455394B2  
JP5452165B2  
JP5451870B2  
JP2014043463A
To provide alkanoylamino benzamide aniline HDAC inhibitor compounds.The present invention provides a compound of the general formula (I) having histone deacetylase (HDAC) inhibitory activity, a pharmaceutical composition comprising the c...  
JP5437525B1
[Subject] The present invention is melatonin MT.1In addition to a tyrosine derivative useful as a receptor antagonist, in a benzene ring of m* tyrosine, an iodine machine is introduced by good site selectivity and quantity 収率 at leas...  
JP5435656B2  
JP5436438B2  
JP5425806B2  
JP5424650B2  

Matches 751 - 800 out of 4,296