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WO/2008/145010A1 |
Preparation methods of 4-acetyl-2,3,4,5-tetrahydro-benzo[1,4]diazepine and their intermediates. Compounds represented by the formula I and II. The preparation methods of 4-acetyl-2,3,4,5-tetrahydro-benzo[1,4]diazepine in which compounds ...
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WO/2008/144981A1 |
The invention provides compounds of formula (I) and (II), and method for preparing 4-acetyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine through intermediates of formula (I) and (II).
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WO/2008/143141A1 |
Disclosed is a method for producing a halogenated aromatic compound, which is characterized in that an aromatic compound wherein one or more substituents and two or more hydrogen atoms are attached to a nucleus and an N-iodine bond type ...
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WO/2008/139056A1 |
The invention relates to a method for preparing 2-(n-butyl)-5-nitrobenzofuran from 1-halogeno-4-nitrobenzene, characterised in that it comprises reacting the 1-hexen-3-ol, then subjecting the product to a Claisen rearrangement, followed ...
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WO/2008/128711A1 |
The present invention provides novel aryl pyrrolidines having an excellent insecticidal action as insecticides. Aryl pyrrolidines represented by the formula (I) and use thereof as insecticide.
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WO/2008/124878A1 |
The present invention relates to non-steroidal compounds useful in the treatment of inflammatory conditions and pharmaceutical compositions comprising them. A representative example of these compounds is formula (III).
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WO/2008/125867A2 |
There is provided a compound of formula (III), and a process for preparing a compound of formula (V) comprising converting a compound of formula (III) to the compound (V), wherein (X) is fluoro, chloro, bromo or iodo. There is also provi...
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WO/2008/122555A1 |
A method is disclosed for producing 2-nitro-5-fluoro-3',4'-dichlorobiphenyl by decarboxylizing C-C linkage. The method relates to a decarboxylizing cross-coupling of 2-nitro-5-fluorobenzoic acid salts with 1-bromine-3,4-dichlorobenzol, w...
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WO/2008/119804A1 |
The invention related to a novel process, novel process steps and novel intermediates useful in the synthesis of pharmaceutically active compounds, especially renin inhibitors, such as Aliskiren. Inter alia, the invention relates to a pr...
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WO/2008/117704A1 |
3,3'-Diamino-5,5'-diphenyl-4,4'-biphenyldiol, which is useful as a monomer for high-performance polymers, especially ones satisfying a high degree of performance requirements in the field of semiconductors, such as polybenzoxazoles and p...
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WO/2008/110281A2 |
The jinvention relates to 3,4-disubstituted phenoxyphenylamidines of geenral formula (I), a method for production thereof, and use of said amidines for preventing undesired microorganisms and an agent for said purpose, comprising said ph...
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WO/2008/110280A2 |
The invention relates to 3-substituted phenoxyphenylamidines of general formula (I), a method for production thereof and use of said amidines for preventing undesired microorganisms and an agent for said purpose, comprising said phenoxya...
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WO/2008/110314A1 |
The invention relates to fluoroalkylphenylamidines of general formula (I), a method for production thereof and use of said amidines for preventing undesired microorganisms and an agent for said purpose, comprising said phenoxyamidines. T...
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WO/2008/111282A1 |
Disclosed is a hydrotalcite surface-immobilized metal particle catalyst, which is obtained by immobilizing at least one metal selected from Cu, Ag and Au, in the form of particles, on a hydrotalcite surface. Also disclosed is a method fo...
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WO/2008/110315A1 |
The invention relates to 4-cycloallkyl or 4-aryl substituted phenoxyphenylamidines of general formula (I), a method for production thereof and use of said amidines for preventing undesired microorganisms and an agent for said purpose, co...
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WO/2008/110279A1 |
The invention relates to dihalophenoxyphenylamidines of general formula (I), a method for production thereof, the use of said amidines to prevent undesired microorganisms, and an agent for said purpose comprising said phenoxyamidines. Th...
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WO/2008/107312A1 |
The aim of the invention is to provide a widely applicable method for the nitration of substituted benzenes.
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WO/2008/107502A1 |
The invention relates to a compound of general formula (I) or a salt thereof, for use as a pharmaceutical composition for treating infectious diseases, especially for treating diseases caused by Helicobacter. R1 is an H atom, an X atom o...
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WO/2008/102111A2 |
This invention relates to the field of novel explosives, compositions and munitions comprising the same, as well as methods of synthesis and their use. The invention particularly relates to the field of explosives which are switchable be...
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WO/2008/096145A1 |
The invention relates to a process for the preparation of anagrelide, and for the preparation of intermediates for use in preparing anagrelide. The invention also relates to the inteπnediates per se, in particular compounds of formula (...
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WO/2008/093668A1 |
Disclosed is a novel chiral iridium aqua complex which can be used for an asymmetric transfer hydrogenation reaction of a carbonyl compound. Specifically disclosed is a chiral iridium aqua complex represented by the following formula (1)...
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WO/2008/082486A2 |
Disclosed is a process for preparing 3-(amino)-3-cyclobutylmethyl-2-hydroxy-propionamide hydrochloride, an intermediate useful in the preparation of the HCV protease inhibitor (1R,5S)-N-[3-amino-1-(cyclobutylmethyl)-2,3-dioxopropyl]-3-[
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WO/2008/075427A1 |
A curing catalyst (clathrate compound) which is inhibited from catalyzing a curing reaction at low temperatures, is effective in improving one-pack stability, and can effectively cure a resin upon heating. The clathrate compound is chara...
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WO/2008/074755A2 |
This invention relates to novel cinnamic amide derivatives that are found to be potent modulators of ion channels and, as such, they are valuable candidates for the treatment of diseases or disorders as diverse as those which are respons...
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WO/2008/069313A1 |
It is intended to provide a method capable of producing a compound having an excellent HSD1 inhibitory action and a compound useful as a synthetic intermediate efficiently and at low cost, which is excellent in degree of achievement of a...
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WO/2008/066820A1 |
Hydroxy aromatic acids are produced in high yields and high purity (>95%) from halogenated aromatic acids in a reaction mixture containing a copper source and a ligand that coordinates to copper.
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WO/2008/061308A1 |
The present invention relates to protein tyrosine phosphatase (PTP) modulators, in particular PTP inhibitors and their use in the treatment or prophylaxis of disorders modulated by PTP such as cellular proliferation disorders; autoimmune...
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WO/2008/056808A1 |
Disclosed is a polyimide which is obtained by reacting a tetracarboxylic acid component with a diamine component containing a diamine compound represented by the following general formula (1). (In the formula, A represents a biphenylene ...
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WO/2008/041140A2 |
This invention is directed to substituted aryl compounds, which are linked to a substituted indole moiety by various linkers, and the kynurenine/kynuramine-like metabolites of these agents, their preparation and pharmaceutical compositio...
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WO/2008/023780A1 |
It is intended to provide a method of rapid methylation of an aromatic compound or an alkenyl compound, which is capable of obtaining an aromatic compound or an alkenyl compound labeled with a methyl group or a fluoromethyl group under a...
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WO/2008/018520A1 |
Disclosed is a method for producing an optically active hydroxycarboxylic acid derivative which is an intermediate important to production of pharmaceutical products, agricultural chemicals, chemical products and the like. This productio...
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WO/2008/010764A2 |
The present invention relates to a novel process for the preparation of compounds of formula (V) wherein X, Q, R1, Rla and R2 are as defined in the specification, the compounds being useful in the preparation of therapeutic agents.
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WO/2008/006576A1 |
The present invention relates to a method for producing alkenyl nitrobenzols and alkyl anilines that are significant as intermediate products for fungicidally effective alkyl anilides.
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WO/2008/007145A2 |
The present invention relates to a novel process for the preparation of -amino 5 acid s, such as (±)-3-(aminomethyl)-5-methyl-hexanoic acid 1, which is a key intermediate in the preparation of the potent anticonvulsant pregabalin, (S)-(...
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WO/2008/006574A2 |
The invention relates to nitrobenzol derivatives of formula (IV) with R1 hydrogen, halogen, -CR'(CF3)2, wherein R' is selected from ausgewählt ist H, F or -O-C1-4-alkyl; and R3 -CH=CH-i-prop, -CH2CH2-t-but, -CH2CH2-i-prop and (a); or R1...
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WO/2008/005451A2 |
An optical apparatus (fig. 1) for producing light of a predetermined intensity from light sources of less than the predetermined intensity includes a first light source; a second light source; a double dove anti-Gaussian generator in opt...
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WO/2008/005344A2 |
This application discloses provides a process for the introduction of nitro-group functionality into a compound which contains also a site of unsaturation and/or oxygen functionality by direct (one step) oxidation of an oxime functional ...
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WO/2007/147775A1 |
The present invention refers to a process for preparing a compound of the formula (I) wherein R denotes an organic radical which, together with the two carbon atoms to which it is bonded, forms a carbocyclic or heterocyclic ring; R1, R2,...
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WO/2007/138089A1 |
A process for preparing substituted biphenyls of the formula (I), in which the substituents are defined as follows: X is fluorine or chlorine; R1 is nitro, amino or NHR3; R2 is cyano, nitro, halogen, C1-C6-alkyl, C1-C6-alkenyl, C1-C6-alk...
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WO/2007/131638A1 |
The present invention relates to a method for the coupled production of chlorine and isocyanates, with the sulfuric acid which was used for both methods combined after its use, concentrated together, and flowing back into one or both met...
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WO/2007/129960A2 |
The present invention relates to a novel process for the preparation of compounds of Formula (I) wherein X, Q, R1 and R2 are as defined in the specification, the compounds being useful in the preparation of therapeutic agents. The invent...
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WO/2007/126142A1 |
Disclosed is a potassium fluoride dispersion solution composed substantially of potassium fluoride and an aprotic organic solvent having a boiling point higher than that of methanol, which is prepared by mixing a mixture of potassium flu...
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WO/2007/118329A1 |
The present invention relates to the treatment of tuberculosis (mycobacterial infections) by the use of KshAB complex inhibitors, or a KstD molecule, or a HsaAB complex, or a HsaC molecule, or a HsaD molecule. The application also includ...
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WO/2007/111026A1 |
This invention provides an optical film comprising one layer provided on a light transparent substrate and can satisfy a good balance among an anti-dazzling function, an enhanced contrast, color reproduction, and anti-glare prevention. T...
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WO/2007/108006A1 |
The present invention relates to a process for the preparation of 6-(4-chlorophenyl)-2,2-dimethyl-7-phenyl-2, 3-dihydro-1H-pyrrolizin-5-yl acetic acid, in which the key intermediate, 5-Benzyl-3,3-dimethyl-3,4-dihydro-2H-pyrrole is obtain...
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WO/2007/104361A1 |
The present invention relates to organic nanofibers that can be produced from organic compounds having a core according to formula (I), wherein X and/or Y are C or N and n is 2 to 4 by self-organized growth on a solid substrate upon depo...
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WO/2007/102334A1 |
A polysilane-supported transition metal catalyst or (polysilane/inorganic compound)-supported transition metal catalyst which comprises as a polymeric support either a polysilane compound or a combination of a polysilane compound and an ...
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WO/2007/102352A2 |
A dibenzothiazepine compound is suitably prepared by subjecting a 2-amino-2'-carboxy-diphenylsulfide compound to dehydration-condensation reaction in the presence of an acidic catalyst; the 2-amino-2'-carboxy-diphenylsulfide compound is ...
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WO/2007/102594A1 |
A polymer complex which has two or more kinds of pores capable of selectively taking up and/or releasing and/or transporting specific compounds ranging from gaseous low molecules to high molecules such as proteins and other living-body-d...
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WO/2007/101844A1 |
A process for the removal by distillation of dinitrotoluene from process wastewater from the preparation of dinitrotoluene by nitration of toluene by means of nitrating acid, which is characterized in that the process wastewater is broug...
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