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JP2002516305A |
This invention provides compounds of Formula I having the structurewherein:B, C, D, and R1 are as defined hereinbefore in the specification, or a pharmaceutically acceptable salt thereof, which are useful in treating metabolic disorders ...
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JP2002516601A |
(57) [Summary] The present invention relates to 4,4- (disubstituted) cyclohexane-1-one and related compounds that are effective in treating allergic and inflammatory diseases.
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JP2002155035A |
To provide a compound which is expected to be a synthetic intermediate for medicines and agrochemicals, a separating agent for chromatography, or an optically resolving agent for racemates.This 3-amino-1-indanol represented by formula (I...
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JP2002155036A |
To provide a new compound useful as a medicine, especially an antifungal agent.Q73453 substance represented by formula (I) or its pharmaceutically acceptable salt. A method for producing the Q73453 substance, characterized by culturing a...
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JP2002515916A |
An anthraquinone mixture comprising three 1,4-hydroxyalkylamino-anthraquinone derivatives, wherein two of the anthraquinone compounds in the mixture are symmetric and the other anthraquinone compound is asymmetric, and wherein each of th...
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JP2002145836A |
To provide a group IV metal precursor having excellent volatility and thermal properties and chemical stability to hydrolysis, and suitable for the chemical vapor deposition for a multicomponent metal oxide thin film containing a group I...
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JP3283892B2 |
Isoxazole derivs. of formula (I) and their acid-addn. salts and solvates are new: In (I) R = 1-4C alkyl, allyl or cyclopropylmethyl; R1 = H, 1-4C alkyl, allyl, cyclopropylmethyl or aryl(1-4C)alkyl; X = CH2 or O; y = 4-R2-5-R3-3-isoxazoly...
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JP3283069B2 |
PURPOSE: To obtain a new substituted alkenyl ketone derivative useful as an insecticide capable of killing and controlling various kinds of noxious insects, especially rice insect pests such as Nilaparvata lugens and Nephotettix cinctice...
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JP2002511106A |
The object of the present patent application are agents for the oxidative coloring of keratin fibers, particularly hair, based on a developer-coupler combination, characterized in that they contain as the developer at least one 2,5-diami...
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JP2002509906A |
This invention relates to a novel advantageous process for the stereoselective preparation of 2-hydroxy-4-phenylbutyrates (HPB esters) and of their precursors. This is done by starting from readily accessible alpha-unsaturated alpha-hydr...
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JP3271052B2 |
To obtain a new compound useful as a photo-polymerization initiator for ethylene unsaturated compound and a photo-reaction initiator for the photo- setting of a pigment system as a printing ink or a white lacquer. This compound is expres...
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JP2002088060A |
To provide a method for profitably producing an indolenine compound, by which the indolenine compound useful as the basic raw material for polymethine dyes used as sensitizing dyes, dyes for photorecording media, or photothermal conversi...
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JP2002084990A |
To use an α-ketoenamine derivative having cooling effects.A compound having the general formula (wherein, R1 is N- pyrrolidinyl; R2 is methyl; X is ethylidene; and Y is an oxy radical) is used alone or in combination as an ingredient of...
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JP2002508777A |
The invention relates to a novel method for aminating mononuclear aromatic compounds and polynuclear compounds containing at least one aromatic ring. The inventive method enables simple separation of the aminated mononuclear aromatic com...
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JP2002506836A |
This invention relates to a novel, inventive process for the preparation of biphenyls or aromatic olefins by coupling reactions of the Suzuki coupling and Heck coupling type, using allylpalladium catalysts of the mu-halo(triisopropylphos...
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JP3261101B2 |
To obtain a new aromatic diamine suitable for a raw material for polyamide which is satisfactory to flexibility and moldability and useful as an adhesive. This compound is shown by formula I {(m) and (n) are each 0 or 1;R is shown by for...
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JP3257688B2 |
A novel process for producing a-[(dialkylamino)substituted-methylene]b-oxo-(substituted) propanenitriles of the formula: where R, R1 and R2 are defined in the specification by reacting a substituted isoxazole with a diaklylamide dimethyl...
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JP3256502B2 |
To screening the subject compound by providing the compound to the first and second cell types, measuring the influence thereof on the receptor activities, and selecting the compound providing the influence only to the first cell type. T...
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JP2002047256A |
To provide a method for producing an optically active α-hydroxy-β- aminocarboxylic acid derivative.The compound (3), the compound (1) and the compound (2) represented by the following formulas (wherein R1 is an aralkyl or the like; X1,...
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JP2002504529A |
Disubstituted lavendustin A analogs that are PTK inhibitors having antiproliferative activity are described. Preferred compounds of the present invention, without limitation, satisfy either Formula 1 or Formula 2. Currently preferred com...
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JP2002502385A |
The invention relates to non-steroidal gestagens of general formula (I), wherein R<1> and R<2> are the same or different and stand for a hydrogen atom, a C1-C5 alkyl group or a halogen atom, or together with the C atom of the chain stand...
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JP3245162B2 |
Rigid-rod macromonomers, and methods for preparing such macromonomers, having a polyaromatic backbone, solubilizing side groups, and reactive side groups are provided. The macromonomers are chemically incorporated into polymer systems to...
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JP3245163B2 |
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JP3241760B2 |
The invention provides cyclohexanone derivatives of the general formula in which n represents an integer from 0 to 5; each R represents a halogen atom, nitro, cyano, hydroxyl, alkyl, haloalkyl, alkoxy, haloalkoxy, amino, alkylamino, dial...
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JP2001526668A |
The present invention relates to the compounds of formula: in which R1, R2, R3, E, A, X, Z, p and n are as defined herein. These compounds are aldose reductase inhibitors.
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JP2001524468A |
The present invention provides compounds, and pharmaceutical compositions containing those compounds, that act as antagonists at metabotropic glutamate receptors. The compounds are useful for treating neurological diseases and disorders....
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JP2001524469A |
Disclosed is a three step synthesis of 11-aryl-5,6-dihydro-11H-dibenz[b,e]azepines from a 2-aminobenzophenone represented by the following structural formula:and a starting material represented by the following structural formula:Phenyl ...
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JP3232337B2 |
PURPOSE: To obtain the subject new compd. which is a β3adrenoreceptor agonist and useful for obesity, hypertension, hyperlipemia, etc. CONSTITUTION: The compd. is (R)4-[2-(2hydroxy-2phenylethylamino) ethoxy]phenyl acetic acid expressed ...
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JP2001521019A |
[Chemical 1]
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JP2001519810A |
The present invention provides novel methods for the asymmetric synthesis of (S)-6-chloro-4-cyclopropylethynyl-4-trifluoromethyl-1,4-dihy
dro-2H-3,1-benzoxazin-2-one of formula (VI-i) which is useful as a human immunodeficiency virus (HI...
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JP2001517649A5 |
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JP3205063B2 |
PURPOSE: To provide a polymerizable monomer capable of producing an antimicrobial polymer exhibiting an excellent antimicrobial activity, excellent in safety and stability and capable of keeping its activity over a long period. CONSTITUT...
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JP3203579B2 |
This invention relates to analogs of peptidase substrates in which the nitrogen atom of the scissile amide group of the substrate peptide has been replaced by a substituted malonyl moiety. The contemplated peptidase inhibitors of the for...
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JP2001512095A |
This invention concerns the use of a hydroxylic solvent in the preparation of enaminones from the corresponding amine N-oxides or propargylic amines via the general process outlined above (A).
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JP2001220356A |
To provide the design, development, composition and use of a new calcimimetic molecule capable of acting on extracellular calcium ion on the cell by a method mimicking the calcium ion, a calcilytic inhibiting the activity of the intercel...
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JP3197836B2 |
To provide a fixed Lewis acid catalyst high in reaction rate and reaction yield, easy in recovery and reuse, having rare earth metal in an active center and produced by fixing on a polymer compound, and the producing method, a synthesis ...
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JP2001510450A |
Compounds containing two aromatic systems covalently linked through a linker containing one or more atoms, or "linker" defined as including a covalent bond per se so as to space the aromatic systems at a distance 1.5-15 ANGSTROM , are ef...
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JP2001206867A |
To provide a new acetylene compound useful as a synthetic intermediate. This acetylene compound represented by the general formula (I), wherein R1 to R6 and R8 are each H, an alkyl, an aryl, a halogen, an alkoxy, an aryloxy, a perfluoroa...
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JP2001199906A |
To provide a method for carrying out the optical resolution of an enaminone derivative without unstabilize the structure because the optical resolution of the enaminone derivative by an optically active acid has hardly been reported and ...
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JP3185946B2 |
PURPOSE: To obtain a new compound useful as a synthetic intermediate for β-lactam-based antibiotic substances. CONSTITUTION: The compound of formula I(R1 is lower alkyl or phenyl; X is optically active 8-arylmenthyl or bornansultam), e....
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JP3182720B2 |
To obtain a mew α-aminoacetophenone derivative bearing allyl or aralkyl group on the α-site, having especially high activity as a photoinitiator, and effectively usable in esp. printing inks. This new derivative is a compound (acid-add...
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JP3181812B2 |
PURPOSE: To economically and inexpensively obtain the subject compound in high purity in terms of an industrial use in high yield with causing a small amount of industrial waste by using an inorganic acid as a solvent, useful as a liquid...
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JP3179942B2 |
PURPOSE: To provide new cycloalkylalkylamines which are specific sigma- receptor ligands and usable as psychotropic drugs, also in gastrointestinal diseases. CONSTITUTION: The compds. are cycloalkylalkylamines which are the sigma- recept...
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JP3167210B2 |
PURPOSE: To obtain a new compound, excellent in flexibility and biodegradability and suitable as a soft base, etc., for hair treating agents, etc., without stickiness in drying. CONSTITUTION: This compound is expressed by formula I {R1 a...
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JP2001107037A |
To provide a material for a green-red luminescent element which is driven by low voltage, can emit light with high luminance and efficiency, is excellent in stability under repeated use, and can exhibit homogeneous plane luminescence; a ...
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JP3157180B2 |
PURPOSE: To provide the subject reagent which consists of specific magnesium benzyl fluoromalonate, allows the introduction of fluoromethyl group into the carbon of a carbonyl group and yields fluoromethyl ketone at a high yield by react...
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JP2001098070A |
To provide a solventless process for easily producing a tetracarboxylic acid diamine salt being a precursor necessary in producing a polyimide resin applicable to heat-resistant films, etc., through a route of a tetracarboxylic acid diam...
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JP2001089429A |
To provide a cyclobutene derivative having an excellent ileum type bile acid transporter-inhibiting action, its pharmacologically acceptable salt, its ester or other derivatives. The cyclobutene derivative of general formula (I) [R1 is a...
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JP2001089426A |
To provide a new acetylene compound useful as a synthetic intermediate for thermosetting resins, liquid crystal materials, non-linear optical materials, gas separation membrane materials, and so on. This acetylene compound of the general...
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JP3151687B2 |
PURPOSE: To obtain a 3-amino-6-arylazophenol derivative in high yield by synthesizing a 4-amino-o-quinone derivative from catechol and an amine compound in high yield in the presence of an acid and oxidizing agent followed by condensatio...
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