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Patent Searching and Data


Matches 851 - 900 out of 7,335

Document Document Title
WO/2003/079984A2
The present invention pertains, at least in part, to novel substituted tetracycline compounds. These tetracycline compounds can be used to treat numerous tetracycline compound-responsive states, such as bacterial infections and neoplasms...  
WO/2003/077828A2
The present invention relates to novel florfenicol compounds having the chemical structure (I) wherein the compounds are useful for the treatment and/or prevention of bacterial infections in a broad range of patients such as, without lim...  
WO/2003/078376A1
A NK1 antagonist having the formula (I), with the variables defined herein, which is useful for treating a number of disorders, including emesis, depression, anxiety and cough.  
WO/2003/078386A1
The present invention relates to novel naphthyl semicarbazone, naphthylhydrazone, naphthyl thiosemicarbazone, and naphthyl thiohydrazone compounds. The invention also relates to therapeutic uses of such compounds and&sol or their iron co...  
WO/2003/076374A1
A process for producing a compound (I) which comprises the step of reacting a compound (II) with a base in an aprotic solvent as shown by the scheme: (II) (I) wherein R1 and R2 each independently represents lower alkyl.  
WO/2003/074462A1
A process for the purification of 2-methoxy-5-trifluor-methoxy benzaldehyde oil in which the oil is converted to amine by reaction of a nitroaniline with the oil; the imine is isolated as a solid; and the solid imine is converted back to...  
WO/2003/074491A1
A compound of formula (I): F1 Het is a 5− or 6−membered heterocyclic ring containing one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, the ring being substituted by groups R4, R5 and R6&semi R1 ...  
WO/2003/074496A1
The invention relates to compounds of formula (I), where R1 = R5-O-&num , R5-O-CH2-&num , (a), (b), (c), (d) or (e), T= (f), (g), or (h), several methods for production and use thereof for the prevention of harmful organisms and novel in...  
WO2002031896A3
The present invention is generally directed to a polymeric metal complex comprising a polymeric material having a plurality of a first-type functional groups, wherein at least a portion of the functional groups are coordinated to at leas...  
WO/2003/072538A1
The invention relates to a method for producing 2-chloromethylphenyl acetic acid derivatives of formula (I), in which X represents C1-C4 alkoxy or methylamino, by cleaving the ether bonds in compounds of formula (II), in which R represen...  
WO2003006070A3
The present invention relates to improved chelator conjugates of formula (II) with biological targeting molecules, suitable for forming metal complexes with radiometals. The radiometal complexes, especially with the radiometal<99m>Tc, ar...  
WO/2003/066578A1
A pinene derivative represented by the general formula (I) or a salt thereof; and a process for producing the derivative or salt or a process for producing from the derivative or salt an optionally active 2-(t-butoxycarbonyl)amino-3-hydr...  
WO/2003/064359A1
The present invention relates to non-classical cannabinoids that are ligands of the peripheral cannabinoid receptor CB2, and to pharmaceutical compositions thereof comprising as an active ingredient novel (+) α-pinene derivatives, which...  
WO/2003/063758A2
The present invention relates to non−classical cannabinoids that are ligands of the peripheral cannabinoid receptor CB2, and to pharmaceutical compositions thereof comprising as an active ingredient novel (&plus ) &agr −pinene deriva...  
WO/2003/062253A1
This invention relates to metal complexes which are useful as catalyst components in olefin metathesis reactions, atom or group transfer radical polymerisation or addition reactions and vinylation reactions. It also relates, preferably w...  
WO2002094767A3
Compounds of formula (I), are novel P2X>3< and P2X>23< antagonists which are useful in treating pain, urinary incontinence and bladder overactivity.  
WO/2003/059064A1
Insecticides containing as the active ingredient hydrazone derivatives represented by the general formula (I); and novel hydrazone derivatives: (I) wherein A and Q are each aryl or a heterocyclic group; W is oxygen, aminylene, alkylene, ...  
WO/2003/059346A1
The invention relates to novel beta-secretase inhibitors.  
WO/2003/057169A2
The present invention pertains, at least in part, to novel substituted 4-dedimethylamino tetracycline compounds. These tetracycline compounds can be used to treat numerous tetracycline compound-responsive states, such as bacterial infect...  
WO/2003/057663A1
Alpha-diimines are prepared from anilines and alpha-ketals such as tetramethoxypropane in the presence of an acidic catalyst.  
WO/2003/049690A2
The present invention relates to the inhibition of HIV integrase, and to the treatment of AIDS or ARC by administering compounds of the following formula, or a tautomer of said compound, or a pharmaceutically acceptable salt, solvate or ...  
WO/2003/048110A1
The invention relates to a process for treating an aqueous medium containing cyclohexanone oxime and cyclohexanone, said process comprising stripping the aqueous medium with steam, wherein said stripping is carried out at a pressure high...  
WO2002017712A3
Compounds of formula (I): wherein A, B, D, and R are as defined herein and their agriculturally acceptable salts are disclosed as effective insecticides. In addition, compositions comprising an insecticidally effective amount of a compou...  
WO/2003/048037A1
The invention relates to a process for preparing nitric acid by treating an aqueous medium containing organic compounds and phosphate, said process comprising: feeding the aqueous medium to a nitric acid synthesis zone, forming nitric ac...  
WO/2003/045899A1
A process for producing 4-bromo-2-oxyimino butyric acid, predominantly as the (Z)-isomer of formula (I), wherein R is hydrogen; a linear or branched C¿1-4? alkyl group; a linear or branched C¿1-4? alkyl group substituted by a carboxyli...  
WO/2003/044025A1
Nitrogen containing analogs of Copper II β−diketonates which analogs are more stable source reagents for copper deposition when substantially free of solvents of excess ligands. The nitrogen containing analogs replace −O− with −...  
WO2002094765A3
The present invention provides a substituted anilide derivative of formula (I): (I) (II) (III) {wherein Z is a group of formula (II) or (III) (in these formulas, A is C1-C6 alkylene, C2-C6 alkenylene, etc., R<1> is H, halogen, -C(R<5>=NO...  
WO/2003/043624A1
Compounds that are dual aP2/k-FABP inhibitors are provided having the formula (I), wherein A, B, X, Y, R?1¿, R?2¿ and R?3¿ are as described herein. A method is also provided for treating diabetes and related diseases, especially Type ...  
WO2002044144A3
Radiolabeled fluorinated compounds useful for imaging in the diagnosis of Parkinson's Disease are disclosed. Methods and kits for their synthesis are also disclosed.  
WO2002059165A3
Certain complexes containing ligands having a phosphino group, amino group or an imino group, and a second functional group such as amide, ester or ketone, when complexed to transition metals, catalyze the (co)polymerization of olefinic ...  
WO/2003/042145A1
A process for preparation of cyclopropylethanol which comprises subjecting a 3−cyclopropyl−2,3−epoxypropionic ester to solvolysis, treating the obtained product with an acid to form cyclopropylacetaldehyde, and reducing this aldehy...  
WO/2003/040096A2
Disclosed are compounds of the formula (I), wherein the variables RN, RC, R1, R25, R2, and R3 are as defined herein. These compounds have activity as inhibitors of betasecretase and are therefore useful in treating a variety of discorder...  
WO/2003/035604A1
A process for the preparation of a compound of formula (I): wherein Ar represents an optionally substituted aromatic carbocycle or heterocycle, and R?1¿ and R?2¿ independently represent hydrogen, C¿1-10?alkyl, C(O)C¿1-10?alkyl or opt...  
WO2003016282A3
This invention provides compounds of Formula I, methods for their preparation and use for preparing compounds of Formula II wherein R¿1?, R¿2?, R¿3?, R¿5?, R¿6?, X and n are as defined in the disclosure. This invention also disclose...  
WO2002036641A3
Improved Group 3-11 transition metal based catalysts and processes for the polymerization of olefins are described. Some of the ligands are characterized by a preferred substitution pattern which allows for higher productivities of highl...  
WO/2003/029189A1
A process for producing a compound represented by the formula [IV] which comprises the steps (1) to (3): a step in which a compound represented by the formula [I] is reacted with either a compound represented by the formula [VI] or a mix...  
WO/2003/024983A1
A transition metal complex represented by the formula (I): (I) [wherein M represents a Group 4 transition metal&semi −Y− represents (a): −C(R1)(R20)−A− (b): −C(R1)(R20)−A1(R30)−, (c): −C(R1)=A1−, or (d): −C(R1)=A1...  
WO2002096861A3
The invention relates to a process for treating an aqueous medium containing (i) phosphate and (ii) cyclohexanone and/or cyclohexanone oxime, said process comprising: feeding the aqueous medium to a stripping zone; passing steam through ...  
WO/2003/020685A1
A fluorine compound represented by the general formula (1). It is effective in incorporating fluorine atoms into a compound having an active group such as an oxygenic functional group and is usable in applications such as surface treatme...  
WO/2003/020689A1
The invention pertains to a chelating agent of the formula: (I) wherein Z is cyclohexylene or (CR¿2?)¿n? wherein R is independently H or C1-4 alkyl, and n is an integer of 2-4; X is (CR'¿2?)¿m?COO?-¿M?+¿ wherein R' is independently...  
WO/2003/018070A1
This invention relates to a method of imaging amyloid deposits and to labeled compounds, and methods of making labeled compounds useful in imaging amyloid deposits. This invention also relates to compounds, and methods of making compound...  
WO/2003/016282A2
This invention provides compounds of Formula (I), methods for their preparation and use for preparing compounds of Formula (II) wherein R¿1&quest , R¿2&quest , R¿3&quest , R¿5&quest , R¿6&quest , X and n are as defined in the disclo...  
WO/2003/016265A1
A compound represented by the following formula, which has excellent PPAR agonistic activity: (I) wherein a, b, and c each is 0 to 4&semi R1 to R6 each represents hydrogen, hydroxy, cyano, halogeno, etc.&semi A1 and A2 each represents a ...  
WO/2003/016283A1
This invention relates to a compound of Formula I, a method for its preparation and its use in the preparation of a compound of Formula II wherein R¿1?, R¿2?, R¿3?, X and n are as defined in the disclosure.This invention also disclose...  
WO/2003/016267A1
The present invention relates to compounds of Formula (I) which may be useful in the treatment of diseases, such as, metabolic disorders, dyslipidemia and/or hypercholesteremia: (I).  
WO/2003/015518A1
This invention pertains to a method for controlling lepidopteran, homopteran, hemipteran, thysanopteran and coleopteran insect pests comprising contacting the insects or their environment with an arthropodicidally effective amount of a c...  
WO/2003/015519A1
This invention provides compounds of Formula (1), their N-oxides and agriculturally suitable salts wherein R¿1?, R¿2?, R¿3?, R¿4a?, R¿4b? and R¿5? are as defined in the disclosure.Also disclosed are methods for controlling inverteb...  
WO/2003/014065A1
The invention relates to a method for producing the (2E)-2-(hydroxyphenyl)-2-(alkoxyimino)-N-methylacetamides of formula (I), wherein R represents C¿1?-C¿6? alkyl which is mono- to trisubstituted by fluorine or not substituted, by reac...  
WO/2003/014066A2
The invention relates to a novel method for producing 2-(hydroxyphenyl)-2-(alkoxyimino)-N-methylacetamide derivatives.  
WO/2003/014296A2
Compounds containing a specific saturated or unsaturated branched chain terminal group; a polar leading group; and a long-chain aliphatic, non-cyclic, saturated or unsaturated, substituted or unsubstituted, hydrocarbon group linking them...  

Matches 851 - 900 out of 7,335