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WO/2001/014320A1 |
The present invention relates to compounds of Formula (I) or a pharmaceutically acceptable salt, solvate, hydrate or formulation thereof. These compounds can be used for the inhibition of tryptase and for the treatment and/or prevention ...
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WO/2001/012585A1 |
A fungicidal compound of formula (I) having a fluorovinye- or fluoropropenyl-oxyphenyloxime moiety and stereoisomers thereof are useful for protecting crops from fungal diseases: wherein, X is CH or N; Y is O or NH; R?1¿ is hydrogen, CÂ...
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WO/2001/012589A1 |
Copper is preferentially extracted from iron in an aqueous feedstock solution containing dissolved copper and iron values by contacting the feedstock solution with a water-immiscible organic solution comprised of a hydrocarbon solvent an...
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WO/2001/012590A1 |
The invention relates to compounds having usefulness in the control of Take-All disease in plants, particularly cereals, a method for the control of Take-All disease, and fungicidal compositions for carrying out the method. Compounds of ...
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WO/2001/009084A1 |
Disclosed is a process for the preparation of cyclopropylglycine by a 5-step process wherein cyclopropanecarboxaldehyde is reacted with an $g(a)-aminoalkylaromatic compound to obtain an imine which is reacted with a cyanide to produce an...
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WO/2001/009087A1 |
The invention relates to novel, substituted arylhydrazone carboxylic acid derivatives of general formula (I), wherein R?1¿, R?2¿, R?3¿, R?4¿, R?5¿, R?6¿, R?7¿ and R?8¿ have the meaning defined in the description. The invention fu...
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WO/2001/007400A1 |
Substances inhibiting cell adhesion mediated by adhesion molecules (in particular, VLA-4) which enable the prevention and treatment of inflammatory diseases caused by leukocyte (for example, monocyte, lymphocyte or eosinocyte) infiltrati...
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WO/2001/007401A1 |
Compounds represented by general formula (I), prodrugs or salts thereof, or solvates of them; and drug compositions containing the compounds, prodrugs, salts or solvates, wherein A, B and C are each an aromatic carbo- or hetero-cycle or ...
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WO/2001/007032A1 |
Th2 differentiation inhibitors which contain compounds represented by general formula (I), prodrugs thereof, pharmaceutically acceptable salts thereof or solvates of the same, wherein the rings A, B and C are each an aromatic carbon ring...
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WO/2001/005925A1 |
Novel metal complexes of tripodal ligands are useful as catalysts to enhance the action of peroxygen compounds in washing, cleaning and disinfecting processes.
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WO/2001/004247A1 |
There is provided a process for producing particles of amine reaction product by means of a carrier having a melting point of less than 30 °C, optionally followed by a coating step. Processed amine reaction products and finished composi...
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WO/2001/004084A1 |
There is provided a process for producing amines, in particular suitable for industrial process, whereby high yields of the imine is obtained. This is achieved by having a selected temperature range upon the contacting of the amine conta...
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WO/2001/003826A1 |
A method for producing a photochemical reaction using a photochemical reaction apparatus having a plurality of discharge lamps arranged with a certain spacing which are lighted up by alternating current and the light emitting parts of wh...
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WO/2001/002334A1 |
The objective bicyclic amino alcohol (IV) is produced by reacting nopinone (I) (starting material) with XCH¿2?COOR?1¿ (wherein X is halogeno; and R?1¿ is alkyl) in the presence of an additive and a base to form a compound (II), conver...
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WO/2001/001779A1 |
The present invention relates to novel acrylate-type N-methyl E-2-((2-methylphenyl)oxymethyl)-6-methylphenylglyoxylamide O-methyl oxime represented by formula (1), its preparation method and its use as fungicides. The compound of the pre...
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WO/2001/000581A1 |
The present invention includes array of new chiral ligands that are optically active or racemic. These ligands are bidentate, tridentate, tetradentate or pentadentate ligands which include P-P, P-N, N-N, mixed P-N, Schiff base or carbene...
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WO/2000/073280A1 |
The present invention provides novel cathecol hydrazone derivatives of formula (I) or pharmaceutically acceptable salts thereof, wherein R?1¿ is C¿1-7? alkyl or C¿3-7? cycloalkyl; R?2¿ is hydrogen, hydroxy, C¿1-5? alkyl or -CH¿2?CH...
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WO/2000/071500A1 |
The invention relates to novel halogen compounds, to a method for producing them and to their use for treating plants for protecting them against attack from phytopathogenic microorganisms and insects. The invention also relates to novel...
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WO/2000/071504A1 |
The invention relates to novel methods of producing methoxyimino acetic amides.
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WO/2000/066638A1 |
Polyethylene is formed by contacting ethylene with a novel iron or cobalt complex of a selected 1,4,7-triaza-3-oxa-1,4,6-heptatriene or 2,5,8-triaza-1,8-nonadiene, optionally in the presence of a cocatalyst such as an alkylaluminum compo...
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WO/2000/066522A1 |
The present invention provides non-steroidal compounds of formula (I) which are selective modulators (i.e., agonists and antagonists) of a steroid receptor, specifically, the glucocorticoid receptor. The present invention also provides p...
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WO/2000/066587A2 |
Novel conformationally restricted polyamine analogs are provided, as well as compositions comprising these novel polyamine analogs. Methods of using the novel polyamine analogs in treatment of diseases such as cancer are also provided. A...
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WO/2000/066600A1 |
The invention relates to a method for producing 1,2-diimine compounds of general formula (I) in which the symbols have the following meanings: R?1¿ and R?2¿, independent of one another, represent alkyl radicals, aryl radicals or metall...
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WO/2000/066597A1 |
The invention relates to novel ionic liquids and to the production and use thereof. The novel ionic liquids are salts of sulphonated or carboxylated triesters of phosphorous acid as the anionic component and ammonium ions, which can be s...
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WO2000046235B1 |
The invention relates to novel betulinic acid derivatives of structural formula having modifications at C2, C3, C17, C20 and/or C29 positions, said derivatives being useful as inhibitors of tumor/cancer cells; process for preparation of ...
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WO/2000/064860A1 |
The present invention relates to new polyaldimines that are stable either per se or in a mixture with aromatic polyisocyanates. However, when exposed to moisture the polyaldimines readily generate polyamines upon hydrolysis. Moisture cur...
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WO/2000/063159A1 |
A description is given here of novel solid and stable derivatives of (-)-verbenone having formula (I) wherein, when X = O Z = H, =CHAr, =C(OH)COOEt, =NOR; Y = H, NH¿2?, NH¿3??+¿ X¿1??-¿, NHCOAr, NHCOR, NHCONHR, NHCONHAr; X¿1??-¿ =...
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WO/2000/063162A1 |
The invention relates to a process for the preparation of compounds of formula (I) wherein: R¿1? is optionally substituted alkyl, R¿2? is C¿1?-C¿6?alkyl, C¿3?-C¿6?cycloalkyl, C¿3?-C¿6?cycloalkyl-C¿1?-C¿2?alkyl, aryl, aryl-C¿1?...
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WO/2000/059954A1 |
The invention relates to a method for radical aqueous emulsion polymerization for producing an aqueous polymerization dispersion. According to the inventive method, ethylenically unsaturated monomers are polymerized by way of a radical p...
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WO/2000/059868A1 |
The invention relates to substituted aniline compounds of formula (1), wherein R?21¿, R?22¿ and R?23¿ have the meanings cited in the description. The inventive compounds are intermediate products used producing herbicidally active pyr...
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WO/2000/059866A1 |
The invention relates to novel compounds of formula (I) wherein R¿1? represents a polymer, aryl or alkyl group, R¿2? represents a hydrogen atom, a halogen atom, a radical CN, CF¿3?, OH, OCF¿3?, COOH, R?7¿, OR?7¿ or OCOR?7¿, R?3¿ ...
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WO/2000/059864A1 |
The invention concerns compounds inhibiting LTA¿4? hydrolase of formula (I). The invention also concerns their therapeutic, in particular anti-inflammatory, applications.
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WO/2000/058262A1 |
The present invention provides stereospecific processes for the preparation of tomoxetine using a nucleophilic aromatic displacement, processes to intermediates thereof, and intermediates thereof.
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WO/2000/058288A1 |
The invention relates to pyridine-2,3-dicarboxylic acid diamides of formula (I), wherein the variables have the meanings indicated in the description. The compounds are useful as herbicidal agents or for desiccating or defoliating plants.
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WO/2000/056702A1 |
The present invention relates to the use of certain resorcinol derivatives as skin lightening agents.
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WO/2000/055113A1 |
A process of reacting an N-protected $g(a)-amino acid ester with a dihalomethyllithium to thereby obtain an $g(a)-amino dihalomethyl ketone derivative. This process is suitable for industrial production and enables economical and efficie...
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WO/2000/053585A1 |
Compounds of Formula T-E-Y?1¿-Y?2¿-Z, and their $i(N)-oxides and agriculturally suitable salts, are disclosed which are useful as fungicides and acaricides wherein E, together with two contiguous carbon atoms forms certain aromatic rin...
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WO/2000/053574A1 |
Novel manganese complexes of salen ligands and the use thereof as catalysts that enhance the action of peroxy compounds in washing, cleaning and disinfecting processes.
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WO/2000/051979A1 |
The invention provides novel PGF analogs. In particular, the present invention relates to compounds having a structure according to formula (I) wherein R¿1?, X, and Z are defined below. This invention also includes optical isomers, dias...
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WO2000002887B1 |
One aspect of the present invention relates to novel ligands for transition metals. A second aspect of the present invention relates to the use of catalysts comprising these ligands in transition metal-catalyzed carbon-heteroatom and car...
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WO/2000/046209A1 |
The invention concerns N-piperidino-5-(4-bromophenyl)-1-(2,4dichlorophenyl)-4-ethyl
pyrazole-3-carboxamide, the salts and solvents thereof which are powerful antagonists of cannabinoid CB¿1? receptors. The method for preparing them cons...
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WO/2000/046187A2 |
The present invention is directed to agmatine and polyamine analogs and their use as drugs, as well as agricultural or environmentally useful agents. As drugs, the analogs decrease cellular polyamine levels, possibly by inducing antizyme...
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WO/2000/046184A1 |
The invention provides fungicidal compounds of formula (I) and salts thereof wherein: R?1¿ is alkyl, alkenyl, alkynyl, carbocyclyl or heterocyclyl, each of which may be substituted, or hydrogen; R?2¿ and R?3¿, which may be the same or...
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WO/2000/046210A2 |
The invention relates to a process for the preparation of a compound of formula (I): wherein W, R?1¿, R?2¿ and R?3¿ are as defined in the description.
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WO2000006146A9 |
This invention relates to substituted anilide compounds which are modulators, agonists or antagonists, of the CCR5 receptor. In addition, this invention relates to the treatment and prevention of disease states mediated by CCR5.
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WO/2000/044706A1 |
A process which comprises converting a $g(a)-amino acid ester into the corresponding imine to thereby protect the amino group of the ester, reacting the imine with a halomethyllithium to form an N-protected $g(a)-amino halomethyl ketone,...
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WO/2000/044742A1 |
Families of brominated, iodated or brominated and iodated squaraines and squarylium derivatives are disclosed. The derivatives have one of general formulas (IA, IB, IC, IIA, III, IV) where X is R12NR13, for example, where R12 and R13 can...
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WO/2000/041476A2 |
Compounds of formula (I) wherein R¿1? is C¿1?-C¿4?-alkyl or cyclopropyl; R¿2? is C¿1?-C¿6?-alkyl, C¿2?-C¿6?-alkenyl, C¿2?-C¿6?-alkinyl; or C¿1?-C¿6?-alkyl substituted by 1 to 5 fluorine atoms; R¿3? is C¿1?-C¿6?-alkyl, C¿1...
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WO/2000/041998A1 |
Propargylether derivatives of formula (I) including the optical isomers thereof and mixtures of such isomers, wherein R¿1? is hydrogen, alkyl, cycloalkyl or optionally substituted aryl, R¿2? and R¿3? are each independently hydrogen or...
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WO/2000/041999A1 |
Oxime derivatives represented by general formula (1) and having excellent plant disease controlling effects and insecticidal and acaricidal activities: wherein R?1¿ is optionally substituted C¿1?-C¿10? alkyl or the like; one of U and ...
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