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JP5705215B2 |
The invention relates to a process for preparing urethane-containing acrylic- and (meth)acrylic esters by reacting a urethane-containing alcohol with a reactant acrylic- or (meth)acrylic ester of a saturated alcohol in the presence of at...
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JP2015074642A |
To provide a method of producing tertiary amine or tertiary amine derivative with high selectivity.In the method of producing tertiary amine or tertiary amine derivative, a reaction system including: an organic chemical raw material cont...
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JP5701832B2 |
The present invention provides a method represented by Scheme 1: wherein X represents I, Br, Cl, alkylsulfonate, or arylsulfonate; Z represents optionally substituted aryl, heteroaryl or alkenyl; L represents hydrogen or a negative charg...
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JP5700595B2 |
The present invention provides a separation method of separating (A) and (B), comprising: a step of separating at least either an active hydrogen-containing compound (A) or a compound (B) that reversibly reacts with (A) from a mixture co...
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JP5697998B2 |
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JP5686413B2 |
Disclosed is an adamantanamine derivative which is useful as a significant intermediate of an 11²HSD-1 inhibitor. Disclosed is a compound represented by the formula (II): wherein R 10 is a group represented by the formula: -(CR 13 R 14 ...
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JP5682622B2 |
The present invention relates to a method of producing a carbamate compound, comprising reacting a fluorine-containing carbonic diester compound represented by formula (1) and a non-aromatic diamine compound represented by formula (2) wi...
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JP5671456B2 |
The present invention relates to a ruthenium carbonyl complex that is represented by the following Formula (1): RuXY(CO)(L)
(1) (in the Formula (1), X and Y, which may be the same or di...
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JP5670842B2 |
Methods for synthesis of 1-(acyloxy)-alkyl carbamates, particularly, the synthesis of 1-(acyloxy)-alkyl carbamate prodrugs of primary or secondary amine-containing drugs are described. Also described are methods for synthesis of 1-(acylo...
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JP5667044B2 |
The present invention relates to substituted phenoxybenzamide compounds of general formula (I): in which R1, R2, R3, R4, R5, X, R6 and q are as defined in the claims, to methods of preparing said compounds, to pharmaceutical compositions...
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JP2015025110A |
To provide a novel (meth)acrylate compound that can impart a microbial adhesion preventing function to a radical polymer of the compound, and to provide an easy production method of the above compound with high yield.The (meth)acrylate c...
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JP2015013862A |
To provide a novel process for the preparation of a protected L-alanine derivative, useful as an intermediate in the synthesis of a compound useful as a μ/δ opioid modulator.A process comprises the steps of: producing a compound repres...
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JP5652879B2 |
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JP5650777B2 |
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JP5645911B2 |
The invention is directed to a process for preparing aromatic carbamates which comprises the reaction of an aromatic amine with an organic carbonate in the presence of a catalyst characterized in that Zn4O(OAc)6 is used as catalyst.
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JP5641582B2 |
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JP5634130B2 |
Disclosed is a novel zinc cluster compound represented by general formula (1): Zn 4 O(OCOR) 6 (RCOOH) n , wherein R represents an alkyl group which has 1 to 4 carbon atoms and may be substituted with a halogen atom, and n represents 0.1 ...
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JP5628332B2 |
A process for coproducing di- and/or polyisocyanates and glycols, comprising process stages A, B, C and E for preparing glycols and process stages A, C, D, E, F and G for preparing di- and/or polyisocyanates, which comprises accomplishin...
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JP5619139B2 |
The present invention relates to the production and the use of 1:1 adducts having a low monomer content from hydroxyalkyl(meth)acrylates and diisocyanates.
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JP5615644B2 |
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JP5611227B2 |
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JP2014196312A |
To provide a novel production method, a novel production process and a novel intermediate useful for synthesis of pharmaceutically active compounds, especially renin inhibitors, e.g. aliskiren.A method of producing compounds of formula (...
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JP5608268B2 |
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JP5603487B2 |
This invention is directed to a process for the preparation of high yield alkyl or aryl iodide from its corresponding carboxylic acid using N-iodo amides.
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JP2014171924A |
To provide a catalyst for selective chemical catalytic reduction capable of selectively hydrogenating, by targeting an organic compound or polymer possessing at least one type of functional group selected from the group consisting of car...
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JP2014523903A |
this indication -- composition of aryl fluoride -- for example18It is related with a reagent and a method useful to the manufacture of a radioactive tracer in which the sign was carried out by F. The reagent and method of indicating in t...
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JP5592786B2 |
An object of the present invention is to provide a process that enables isocyanate to be produced stably over a long period of time and at high yield without encountering problems of the prior art during production of isocyanate without ...
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JP5592893B2 |
The present invention is directed to a novel process for the preparation of protected L-alanine derivatives, useful as intermediates in the synthesis of compounds useful as mu/delta opioid modulators.
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JP5586391B2 |
The present invention relates to a method for producing N-protected amino acid. Specifically, the present invention provides a method in which a protecting group is introduced to the amino group of an amino acid in a reaction under alkal...
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JP5582634B2 |
Compounds of formula (I): in which R1, R2, R7, R8, R9, R10 and A have the meanings given in the specification, are DP2 receptor modulators useful in the treatment of immunologic diseases.
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JP5584632B2 |
An aniline derivative of formula: useful in synthesis of insecticides.
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JP2014144947A |
To provide a compound that can inhibit histone deacetylase (HDAC) and is suitable as a therapeutic agent for diseases associated with cell proliferation such as malignant tumors.This invention provides a novel stilbene-like compound such...
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JP5568137B2 |
Disclosed is a method for producing a compound represented by general formula (2) by causing a compound represented by general formula (1) to react with ammonia.
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JP5566149B2 |
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JP2014139151A |
To provide a production method which allows easy acquisition of (E)-1-halo-enamide derivatives with high purity and is applicable to reactions on the gram scale and novel (E)-1-halo-enamide derivatives.A method of producing (E)-1-halo-en...
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JP5563887B2 |
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JP5563483B2 |
Methods of enzymatically resolving acyloxyalkyl thiocarbonates useful in the synthesis of acyloxyalkyl carbamate prodrugs are disclosed.
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JP5560715B2 |
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JP5563886B2 |
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JP5563816B2 |
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JP5554698B2 |
The invention relates to a process for the preparation of N-protected alpha-aminoaldehydes by deacetalization of the acetal functional group of corresponding N-protected alpha-aminoacetals using formic acid.
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JP5552489B2 |
The present invention relates to a method for producing taxane derivatives with anticancer activity. The method of the present invention produces taxane derivatives in a short time under mild conditions by employing phenyl oxazinan dione...
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JP5541594B2 |
Compounds are provided which comprise (a) at least two polymerisable moieties, (b) at least one amino acid residue of an amino acid comprising at least two amine groups of which at least two amine groups have formed a carbamate, a thioca...
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JP5545215B2 |
A method for production of an N-carboxy amino acid anhydride with efficiency is provided. The method for production of an N-carboxy amino acid anhydride includes a step of reaction of an amino acid organic salt compound with a carbonic a...
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JP5529110B2 |
The invention provides metal carbamates of the general formula (I) where R1 and R2 are each an alkyl group.
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JP5529540B2 |
The compounds and the synthesis of [F-18]-labeled L-glutamic acid, [F-18]-labeled L-glutamate, their derivatives as set forth in formula (I) and their uses are described.
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JP5524629B2 |
Cyclohexanedione compounds, and derivatives thereof, which are substituted in 5-position, are suitable for use as herbicides. The cyclohexanedione compounds and derivatives of the invention are compounds of formula (I) wherein the substi...
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JP5516177B2 |
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JP5518056B2 |
Procedure for preparing carbamates comprising reaction between at least: an amine or polyamines, an organic carbonate of formula (OR)(OR')C=O, a catalyst formed at least by a support selected from among at least a metal oxide, a micropor...
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JP5518605B2 |
A method for producing toluenedicarbamate includes a carbamate production process of producing toluenedicarbamate by reaction between toluenediamine, urea, and/or N-unsubstituted carbamic acid ester, and alcohol; and a benzoyleneurea red...
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