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WO/2004/078703A1 |
The invention provides novel acid generators which are unproblematic in combustibility and accumulation inside the human body and can generate acids having high acidities and high boiling points and exhibiting properly short diffusion le...
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WO/2004/074242A2 |
Compounds of the formula (I) or (II) wherein R1 is C1-C10haloalkylsulfonyl, halobenzenesulfonyl, C2-C10haloalkanoyl, halobenzoyl; R2 is halogen or C1-C10haloalkyl; Arl is phenyl, biphenylyl, fluorenyl, naphthyl, anthracyl, phenanthryl, o...
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WO/2004/069823A1 |
The invention relates to the inhibition of histone deacetylase. The invention provides compounds and methods for inhibiting histone deacetylase enzymatic activity. The invention also provides compositions and methods for treating cell pr...
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WO/2004/066929A2 |
Novel thyroid receptor ligands are provided having the general Formula (I) wherein X, R1, R2, R3, R4, R5, R6, R7, R8, R9, R10 and R11, are as defined herein. In addition, a method is provided for preventing, inhibiting or treating diseas...
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WO/2004/067503A1 |
The invention relates to a composition containing formamidine sulfinic acid. Said composition contains up to 1 wt. % gelatine that acts as an agent for improving the flowability and eliminates dust problems. Preferred compositions contai...
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WO/2004/062598A2 |
The invention encompasses compounds of Formula (I), which are antis inflammatory and anti-thrombotic agents. The invention also encompasses certain pharmaceutical compositions and methods for treatment of cyclooxygenases (COX-1 and COX-2...
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WO/2004/062601A2 |
Antibacterial compounds of formula (I) are provided: As well as stereoisomers, pharmaceutically acceptable salts, esters, and prodrugs thereof; pharmaceutical compositions comprising such compounds; methods of treating bacterial infectio...
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WO/2004/058699A2 |
The present invention discloses a new class of triarylsulfonium salt photoacid generators (PAGs), which are thermally stable and can be activated by long wavelength UV or visible light. The sulfonium PAGs of the present invention are add...
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WO/2004/052849A1 |
A benzoic acid compound represented by the formula [I]: [I] (wherein Q represents a group selected from the following groups: Q1 Q2 Q3 Q4 Q5 Q6 R1 and R4 to R15 each represents hydrogen, alkyl, etc.; R2 and R3 each represents alkyl or a ...
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WO/2004/031287A1 |
Compounds of the formula (I) wherein R1 is C1-C18alkyl, C5-C12-cycloalkyl, phenyl, benzyl, or allyl; n is 1 or 2; if n is 1, R2 is C4-C18alkyl, C5-C12cycloalkyl, aryl or heteroaryl, benzyl, allyl, (CH2),mCOOR3, or is (CH2)mCN; if n is ...
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WO/2004/011422A1 |
The subject invention provides convenient, regiospecific and highly stereoselective addition of SF5Cl in high yield to a variety of alkenes and alkynes.
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WO/2003/106410A1 |
Fluorinated cycloalkyl-derivatised benzoylguanidines of formula (I) are suitable for use as anti-arrhythmic medicaments comprising cardioprotective components for the prophylaxis and treatment of infarcts and also for the treatment of an...
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WO/2003/097591A1 |
The invention relates to pentafluorosulfanyl-benzoylguanidines of formula (I) and (II), wherein R1 to R4 have the meaning mentioned in the claims. Said pentafluorosulfanyl-benzoylguanidines are suitable as antiarrhythmic medicaments with...
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WO/2003/093228A1 |
A phthalamide derivative represented by the general formula (I): (I) wherein R1 represents hydrogen, C1-6 alkyl, C1-6 alkyl substituted by C1-6 alkylthio, etc.; R2 and R3 may be the same or different and each represents hydrogen, C1-6 al...
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WO/2003/090297A1 |
An organic salt having an alkali metal bound to a disubstituted amide of alkane iminosulfinic acid has the following general formula: where Ar is an aromatic group, M is an alkali metal such as Li, K, or Na, and cxhy is an alkane. The or...
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WO/2003/087075A1 |
Enantiomerically enriched trans-2,3-epoxyamides of the formula (I) in which R1 is a 1-18C aliphatic hydrocarbyl optionally substituted by one or more substituent groups selected from halo, nitro, phenyl and -ORW, where RW is H, 1-6C alky...
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WO/2003/084997A1 |
Aspects of the present invention include probes, methods, systems that have stand alone utility and may comprise features of a drug discovery system or method. The present invention also includes pharmaceutical compositions. In more deta...
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WO/2003/084982A2 |
The present invention relates to improved covalent coupling of two or more entities such as biomolecules, polymer compositions, organic/inorganic molecules/materials, and the like, including their combinations, through one or more novel ...
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WO/2003/067332A2 |
Chemically amplified photoresist compositions comprising, (a) a compound which cures upon the action of an acid or a compound whose solubility is increased upon the action of an acid&semi and (b) a compound of the formula (Ia), (Ib), (II...
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WO/2003/059824A1 |
This invention relates to a process for improving the purity of an aqueous onium hydroxide solution. In particular, the invention relates to a process for improving the purity of aqueous onium hydroxide solutions containing undesirable a...
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WO/2003/057169A2 |
The present invention pertains, at least in part, to novel substituted 4-dedimethylamino tetracycline compounds. These tetracycline compounds can be used to treat numerous tetracycline compound-responsive states, such as bacterial infect...
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WO2002039965B1 |
The invention relates to a reducing composition for the permanent deformation of the hair comprising an N-substituted formamidinesulphinic acid derivative as reducing agent and to a process for the permanent deformation of the hair emplo...
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WO/2003/055849A1 |
The invention relates to a method for the production of solutions a quaternary cation and an anion from a deprotonated hydroxy aromatic in an organic solvent by a reactive extraction of a quaternary salt in the presence of an aqueous hyd...
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WO/2003/040090A1 |
A hybrid onium salt having an iodonium salt and a sulfonium salt in the molecule. It is useful as, e.g., a cationic photopolymerization initiator or an acid generator for chemical−amplification−type resists. It is represented by the ...
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WO/2003/024448A2 |
The invention relates to the inhibition of histone deacetylase. The invention provides compounds e.g. (1) and methods for inhibiting deacetylase enzymatic activity. The invention also provides compositions and methods for treating cell p...
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WO/2003/014072A1 |
The present invention provides compounds and libraries of compounds having formula (I), wherein L and n are defined as in the claims and A is -S(CH¿2?)¿p?R?A1¿ or -S(O)¿2?R?A2¿ with p, R?A1¿ and R?A2¿ as defined in the claims. The...
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WO/2003/003120A1 |
Thiophene-containing photo acid generators having either of the following general formulas: wherein at least one of R?1¿, R?2¿ or R?3¿ is thiophene or thiophene that is substituted with alkyl, alkoxy or cycloalkyl, and the remaining R...
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WO2002082185B1 |
A photoacid compound having general structure: R-O(CF2)nSO3X wherein n is an integer between about 1 to 4; R is selected from the group consisting of: substituted or unsubstituted C1-C12 linear or branched alkyl or alkenyl, substituted o...
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WO/2002/092559A1 |
The invention relates to sulfonium salts useful as acid generator for resists or cationic photopolymerization initiator and provides sulfonium salts represented by the general formula [1]: [1] (wherein R1 is monofluorophenyl which may ha...
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WO/2002/083633A1 |
Suplatast tosilate crystals showing characteristic peaks at diffraction angles (2$g(u) ± 0.1°) of 5.6°, 9.0°, 11.0°, 15.3°, 16.5°, 17.2°, 17.9°, 19.2° and 21.5° in powder X-ray diffractometry; and a process for producing the s...
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WO/2002/083608A2 |
This invention encompasses novel methods of preparing sulfinamides and sulfoxides, particularly stereomerically pure sulfinamides and sulfoxides. The invention further encompasses novel compounds from which sulfinamides and sulfoxides ca...
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WO/2002/083698A1 |
The present invention provides a process for preparing a metal carbene complex of formula (I): wherein M is a transition metal atom selected from the group consisting of ruthenium, rhodium, iron , cobalt, osmium and iridium; L denotes ne...
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WO/2002/081439A1 |
A triarylsulfonium salt which is useful as an acid generator for resists or a cationic photopolymerization initiator; a novel process for producing a trialkylsulfonium salt; and a sulfonium salt. A compound represented by the general for...
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WO/2002/079691A1 |
The present invention provides compounds and compositions, which include: at least one chromophore having strong simultaneous two-photon or multi-photon absorptivity; at least one acid- or radical-generator in close proximity to the chro...
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WO/2002/079271A2 |
The invention relates to a composition comprising: a) an acid monomer or oligomer of acrylic acid or of an acid derivative of acrylic acid or mixtures thereof; or a mixture of an ethylenically unsaturated monomer or oligomer and an acid ...
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WO/2002/074736A1 |
The present invention relates to a novel diaminedithiol derivative or a pharmaceutically acceptable salt thereof; radiorhenium or radiotechneticum complex thereof; a composition for treating liver cancer comprising the radiorhenium compl...
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WO/2002/072640A1 |
A polymerizable composition comprising (A) a polymerization initiator represented by the general formula (1) and (B) a radical-polymerizable compound: (1) wherein R?5¿, R?6¿, R?7¿, R?8¿, and R?9¿ are each independently hydrogen, alk...
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WO/2002/072540A2 |
The present invention pertains to methods for preparing a compound of Formula (I), wherein A is O or N-L; each L is independently H or an acyl group; K is, together with the two contiguous linking carbon atoms, a phenyl ring, a 5- or 6-m...
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WO/2002/064553A1 |
A process for preparation of halogenoalcohol derivatives represented by the general formula (1) and novel useful intermediates are provided. Halogenoalcohols of the general formula (1), i.e., (2S,3R)-N-Cbz-3-amino-1-halogeno-4-phenylsulf...
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WO/2002/064583A2 |
The invention relates to bis(alkylthio)carbenium salts of formula (I) wherein R?1¿, R?2¿, R?3¿ and Y?-¿ have the cited designations, and a method for the production of the same. The inventive compounds are advantageously suitable as ...
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WO/2002/060388A2 |
A class of acyl sulfamides comprises compounds that are potent ligands for PPAR gamma and generally have antagonist or partial agonist activity. The compounds may be useful in the treatment, control or prevention of obesity, non-insulin ...
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WO/2002/059080A2 |
The present invention relates to novel, non-peptidic small organic compounds having an affinity for cyclophilin (CyP)-type immunophilin proteins, and to pharmaceutical compositions comprising one or more of the said compounds. The invent...
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WO/2002/056874A2 |
Novel nitric-oxide releasing lipid molecules are provided which comprise a lipid molecule selected from (a) phosphoglycerides, (b) lipids having a sphingosine base as a backbone, (c) monoacylglyerols, (d) diacylglycerols, (e) glycosylacy...
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WO/2002/048101A1 |
A process for directly producing the target sulfonium salt not via a metathesis step without using a large excess of an acid. The process comprises reacting an aryl compound (A) in which at least one of the carbon atoms of the aryl group...
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WO/2002/048100A2 |
Novel and known thiosulphonic esters of formula (I), where R1 and R2 have the meaning given in the description, are particularly suitable as pesticides for the protection of commercial materials.
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WO/2002/048081A1 |
The invention relates to liquid crystalline compounds of formula (I) wherein R?1¿, R?2¿, A?1¿, A?2¿, A?3¿, A?4¿, Z?1¿, Z?2¿, a, b and c have the designations cited in claim 1. The invention also relates to liquid crystalline medi...
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WO/2002/046507A2 |
A chemically amplified photoresist composition comprising, (a) a compound which cures upon the action of an acid or a compound whose solubility is increased upon the action of an acid; and (b) as photosensitive acid donor, at least one c...
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WO/2002/042263A1 |
The invention provides polyflurinated aromatic or heterocyclic compounds comprising at least three ring substitutents, at least one of which comprises a sulphurpentafluoride group and at least one of which comprises a labile group; metho...
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WO/2002/042845A2 |
This invention relates to new photoacid generator compounds and photoresist compositions that comprise such compounds. In particular, the invention relates to photoacid generator compounds that generate an $g(a),$g(a)-difluoroalkyl sulfo...
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WO/2002/028917A2 |
A resin and its use as a methylating agent. One embodiment is a resin comprising a solid support and cationic methylated sulfonium, sulfoxonium, selenonium or phosphonium salts immobilized on the solid support. Another embodiment is the ...
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