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Document Title |
JP4035852B2 |
An industrially excellent alternative process for producing cyclodepsipeptide derivatives, as represented in formula (1), having an excellent vermicidal activity as an animal and human anthelmintic, wherein R1 represents hydrogen or a hy...
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JP4033920B2 |
Endoparasitic activity of cyclic depsipeptides (I) comprising amino acid and hydroxycarboxylic acid units and having 6-30 ring atoms is increased by praziquantel (II) and epsiprantel (III). An endoparasitic agent contg. (I) together with...
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JP4029047B2 |
Production of polyisocyanates by catalytic conversion of aliphatic diisocyanates comprises using a catalyst consisting of a salt in which the anion comprises 5-97.1 wt.% of 1,2,3- and/or 1,2,4-triazolate structures.
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JP2007538106A |
The invention provides N-cyclic sulfonamido compounds for use in treating or preventing cognitive disorders, such as Alzheimer's Disease. Compounds of particular interest are defined by Formula I, wherein R4, R5, R6, R7, and R8, are as d...
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JP2007314580A |
To enhance the endoparasiticidal activity of cyclic depsipeptides. The present invention relates to the use of praziquantel and epsiprantel for enhancing the endoparasiticidal activity of cyclic depsipeptides in endoparasiticidal composi...
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JP4016097B2 |
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JP2007534696A |
The invention is directed to compositions and methods useful for treating Central Nervous System (CNS) disorders. Furthermore, the invention provides compositions and methods of treating sleep disorders. More specifically, the invention ...
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JP4015192B2 |
Disclosed are "acid-amide" calixarenes of formula (I) wherein: L is [-CH2-] or [-O-CH2-O-] and may be the same or different between each aryl group; R5 is H, halogen, or C1-C10 aliphatic hydrocarbyl group, C6-C20 aryl group, C6-C20 hydro...
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JP2007533718A |
Compounds having therapeutic utility are of general formula (1) wherein R, is H, C 1-C6 alkyl optionally substituted with F or C3-C6 cycloalkyl or C2-C4 alkenyl; A is O, CH2 or S(O)n where n is 0-2; one of W, X, Y and Z is N, CH or CR3 a...
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JP2007297303A |
To provide an organic luminous element prevented from the depletion of luminous intensity. An organic luminous compound is provided, which has a specific structure having a site with the function of a dopant and the function of a host in...
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JP4001381B1 |
Novel derivatives of PF1022 substance, which are cyclodepsipeptides represented by the general formula (I) shown below or their salts are useful as anthelmintic agent for prevention or treatment of parasitic infections.
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JP3995300B2 |
Isocyanate trimers (or mixtures) (I) based on aliphatic,cycloaliphatic, aromatic or araliphatic mono- or poly-isocyanates (II) with a NCO content of less than 70%, optionally with other substituents in the organic groups, such as carbony...
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JP2007528420A |
Muscarinic Acetylcholine receptor antagonists and methods of using them are provided.
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JP3985050B2 |
A novel industrial process for producing an anthelmintic depsipeptide derivative represented by structural formula (I), which is excellent in the yield etc.
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JP2007238510A |
To provide an optically active compound highly sensitive and responsible in high speed. The optically active compound is expressed by general formula (I), wherein X1, X2, X3and X4express each independently -NH2, -N(CH3)2, -H, -CpF2p+1, -...
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JP3968933B2 |
To provide high luminance and shelf life electroluminescent element and highly luminescent color filter based on that electroluminescent element by using inorganic and/or rare-earth complex based phosphor. An electroluminescent element c...
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JP3954127B2 |
PURPOSE: To obtain a new cyclic amide derivative exhibiting excellent weeding activity to injurious weed generating in paddy field or upland field in soil treatment or stem and leaf-treatment and exhibiting high safety to crop and useful...
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JP2007519639A |
The invention relates to compounds of formula wherein Het, A1, A2, A3, A4, D, W, T, Q, Y, X1, X2, R1, R2, R3, R4, k and m are as defined hereinabove, and, where applicable, to possible E/Z isomers, mixtures of E/Z isomers and/or tautomer...
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JP2007182456A |
To provide a herbicide having a selective action for killing only weeds without damaging crops, even when simultaneously applied to both the crops and the weeds.A cyclic amide derivative represented by the general formula [I] [-A-B- is -...
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JP3932559B2 |
The invention refers to a pharmaceutical composition suitable for the protection of the mitochondrial genom and/or mitochondrium from damages or for the treatment of diseases connected with such damages, said composition comprising 0.1 t...
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JP3926662B2 |
To provide a new polymer responding to the chirality of a wide range of optically active substances in improved sensitivity and provide a monomer for the polymer. The invention relates to a polyaryl acetylene derivative and its monomer h...
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JP2007513166A |
Certain noel N-(heteroarylalkyl)alkanediamine derivatives have provided unexpected insecticidal and acaricidal activity. These compounds are represented by formula I: wherein Ar, a, r, R, Ra, Rb, Rc, Rd, b, c, Re, Rf, Rg, Rh, R5, d, e, U...
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JP3909870B2 |
PURPOSE: To provide the novel compounds useful as immunosuppressants, anti- inflammatory agents, antifungal agents, antiproliferative agents and antitumor agents. CONSTITUTION: By protecting an alcoholic site of paramycin with a protecti...
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JP3907207B2 |
Provided is a compound of the formula: I This compound is an intermediate to and is used for preparing the arthropodicidal oxidiazine Compound II described in the specification.
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JP3887769B2 |
This invention relates to the use of a group of aryl ureas in treating cytokine mediated diseases and proteolytic enzyme mediated diseases, and pharmaceutical compositions for use in such therapy.
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JP3887784B2 |
PCT No. PCT/EP94/02533 Sec. 371 Date Feb. 5, 1996 Sec. 102(e) Date Feb. 5, 1996 PCT Filed Jul. 29, 1994 PCT Pub. No. WO95/04728 PCT Pub. Date Feb. 16, 1995The application relates to new azadioxacycloalkenes of the formula (I) (I) in whic...
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JP3882411B2 |
To provide a method for readily and environmentally-friendly producing 3,3-alkyleneoxaziridine in high yield. A cycloalkanone is reacted with ammonia and hydrogen peroxide, and the product is reacted with a carboxylic acid and/or a carbo...
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JP3882195B2 |
A method for making a compound of Formula I which is racemic or enantiomerically enriched at chiral center* comprising hydrogenating a compound of Formula V in the presence of a compound of Formula VII wherein: R 1 is F, Cl, or C 1 -C 3 ...
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JP2007501769A |
The present invention relates to the use of sulphonamide salts as catalysts for oligomerizing isocyanates and also to a process for NCO oligomerization using the catalysts of the invention.
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JP3855538B2 |
To provide a processing solution for a silver halide photographic sensitive material having rapid desilvering performance, not causing the stain of an edge part and excellent in liquid preservation stability and environmental suitability...
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JP2006527763A |
The present invention concerns the use of a sphingoid-polyalkylamine conjugate as a capturing agent of biologically active molecules, such as antigens. In a particular embodiment, the spinogid-polyalkylamines are used for the preparation...
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JP2006308474A |
To provide a means which simply and highly sensitively measures heavy metal ions including trivalent heavy metal ions, without using any flame.A mass analyzing reagent for measuring the heavy metal ions is provided, which is composed of ...
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JPWO2005023788A1 |
Microbes belonging to Beauveria sp. And capable of producing FKI-1366 substance A and / or FKI-1366 substance B and / or FKI-1366 substance C (Beauveria sp. FKI-1366, FERM BP- 08459) was cultured in a medium, FKI-1366 substance A and / o...
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JP3837461B2 |
To obtain the subject new compound having crown ether structure, high in ion transfer ability, capable of solid phase polymerization, and useful as a raw material for functional materials such as electroconductive materials, electrode ma...
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JP2006523691A |
Disclosed herein is an antioxidant that is an alkylated iminodibenzyl of the general formula: wherein: R1, R2, R3, and R4 are independently selected from the group consisting of hydrogen, alkyl moieties, and alkenyl moieties; and R5, R6,...
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JP2006523232A |
Compounds useful for treating cellular proliferative diseases and disorders by inhibiting the activity of KSP are disclosed.
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JP2006232691A |
To provide a method for synthesizing the oligomer by using a lactic acid modified with amino acid (for example, glycyl-lactic acid or the like).The oligodepside compound is a compound represented by any of formula (1), formula (2) and fo...
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JP3790424B2 |
A compound having formula (I) or a pharmaceutically acceptable salt or prodrug thereof, is an immunomodulatory agent and is useful in the treatment of restenosis and immune and autoimmune diseases. Also disclosed are cancer-, fungal grow...
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JP2006514939A |
Methods of making substituted phenylalkynes of formula (I).
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JP3749253B2 |
PCT No. PCT/GB95/00019 Sec. 371 Date Jun. 20, 1996 Sec. 102(e) Date Jun. 20, 1996 PCT Filed Jan. 6, 1995 PCT Pub. No. WO95/18808 PCT Pub. Date Jul. 13, 1995Linked polyamine cyclic compounds of general formula V-R-A-R'-W where V and W are...
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JP2006501291A |
Serratamolide, also named cycloÄ(3R)-3-hydroxydecanoyl-L-seryl-(3R)-3-hydroxydecanoyl
-L-serylÜ, is a cyclic depsipeptide isolated from cultures of bacteria of the species Serratia marcescens. Serratamolide decreases the viability of, ...
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JP2005538926A |
An ammonium selective ionophore for use in ion selective electrodes.
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JP2005533030A |
The invention provides a method for preventing or reducing the effects of oxidative stress on a substrate. The method includes the step of treating the substrate with a compound of formula (I), or a pharmaceutically acceptable salt there...
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JP2005272452A |
To provide a new agricultural chemical, particularly an insecticide or acaricide.This invention relates to a substituted benzanilide compound represented by general formula (1) [wherein G is a ring such as G-7, G-13, G-71 or the like; W1...
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JP2005247716A |
To provide an ABC(ATP-binding cassette) transporter inhibitor overcoming the multidrug resistance(MDR) to anticancer drugs due to the amplification and expression of MDR1 gene as the most important problem in cancer chemotherapy or the d...
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JP3693366B2 |
PURPOSE: To provide a new compound useful as a endoparasiticide for human beings and animals, etc. CONSTITUTION: A compound of the formula I [R1, R2, R11 and R12 are each 1-8C alkyl, 1-8C halogenoalkyl, 3-6C cycloalkyl, aralkyl or aryl; ...
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JP2005523925A |
It has now been found that certain novel heterocyclic derivitives have provided unexpected insecticidal activity. These compounds are represented by formula (I): R Preferred are those compounds of formula (I) where R2 and R3 taken togeth...
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JP2005162760A |
To provide a fungicide for protecting plants.The new azadioxacycloalkene is represented by formula (I) (wherein A is an alkanediyl; Ar is an arylene or the like; E is 1-alkene-1 or the like having a R1 group; R1 is hydrogen, a halogen or...
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JP2005132727A |
To provide a new dioxazine derivative useful as an insecticidal and acaricidal active ingredient.The dioxazine derivative is represented by general formula (1) [wherein, R1 denotes a hydrogen atom, an alkyl group or an alkoxyalkyl group;...
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JP3652986B2 |
The present invention relates to novel herbicidally active 3-hydroxy-4-aryl-5-oxopyrazoline derivatives, to processes for their preparation, to compositions which comprise these compounds and may additionally comprise safeners, and to th...
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