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Matches 701 - 750 out of 29,343

Document Document Title
WO/2013/061724A1
Provided are a novel radical inhibitor, a composition containing the same, and a radical generation inhibition method using the same. This radical inhibitor comprises a salen complex compound of a divalent metal.  
WO/2013/060860A1
The present invention relates to compounds having the general formula (I) as described herein; methods of preparing said compounds; and their use in treating Type 1 and/or Type 2 Diabetes Mellitus. The compounds were assayed for binding ...  
WO/2013/061962A1
The present invention provides a compound represented by formula (I) or a salt thereof. (In the formula, the symbols are as defined in the description.)  
WO/2013/061224A1
The present invention provides a novel process and novel intermediates useful in the synthesis of pharmaceutically active compounds, especially renin inhibitors, such as Aliskiren, or a salt thereof, preferably Aliskiren hemifumarate.  
WO/2013/061004A1
The present invention relates to novel disubstituted 3,4-diamino-3-cyclobutene-1,2-dione compounds corresponding to the following general formula (I): , to the pharmaceutical compositions containing these compounds and also to the use of...  
WO/2013/059215A1
Disclosed herein are substituted biaryl alkyl amide compounds, methods of synthesizing substituted biaryl alkyl amide compounds and methods of treating diseases and/or conditions with substituted biaryl alkyl amide compounds.  
WO/2013/058631A2
The present invention relates to a diterpene furanoids compound which inhibits an activity of protein tyrosine phosphatase 1B (PTP1B) and to the use thereof. More particularly, the present invention relates to diterpene furanoids which a...  
WO/2013/059582A2
The disclosure relates to small molecules and methods, compositions, and kits comprising these small molecules. In still another embodiment, the disclosure relates to small molecules that inhibit HDAC activity. In yet another embodiment,...  
WO/2013/059582A3
The disclosure relates to small molecules and methods, compositions, and kits comprising these small molecules. In still another embodiment, the disclosure relates to small molecules that inhibit HDAC activity. In yet another embodiment,...  
WO/2013/058631A3
The present invention relates to a diterpene furanoids compound which inhibits an activity of protein tyrosine phosphatase 1B (PTP1B) and to the use thereof. More particularly, the present invention relates to diterpene furanoids which a...  
WO/2013/053046A1
The present application, relates to iron bisphenolate complexes and methods of use and synthesis thereof. The iron complexes are prepared from tridentate or tetradentate ligands of Formula I: wherein R1 and R2 are as defined herein. Also...  
WO/2013/053816A1
The present invention relates to a process for producing 5-hydroxymethylfurfural (HMF) from fructose in a single-phase aqueous solution comprising an organic solvent.  
WO/2013/053287A1
(-)-(S)-3-(3'-hydroxy)-butylphthalide (a compound shown by Formula I) and an ester formed of the same and an acid are proved by experiments to be applicable to treatment and prevention of cerebral ischemic diseases and have a sleep-impro...  
WO/2013/055577A1
The present invention provides novel selective androgen receptor modulators and their salts and pharmaceutical compositions thereof.  
WO/2013/050301A1
The present invention relates to processes for the enantio-selective preparation of spyrrolidine derivatives useful in the manufacture of pesticidally active compounds, as well as to intermedates in the processes. The processes include t...  
WO/2013/047904A1
The present invention provides a novel compound having a control efficacy on harmful arthropods. A compound represented by Formula (I): wherein Y represents a 3-7-membered saturated heterocyclic group containing one or more atoms or grou...  
WO/2013/047984A1
The present invention relates to a method for producing a furan-based compound using an ion exchange resin in the presence of an organic solvent. In the method for producing a furan-based compound according to the present invention, a fu...  
WO/2013/049711A1
Provided are methods of producing 2,5-furandicarboxylic acid (FDCA) from renewable sources such as seaweed, alginate, oligoalginate, pectin, oligopectin, polygalacturonate, galacturonate, and/or oligogalacturonate. The sugars in the rene...  
WO/2013/047055A1
Provided is a heat shock protein expression inducer based on a heat shock protein (HSP) expression-inducing action. The present invention is a heat shock protein (HSP) expression inducer comprising eupalinolide A and/or B, the heat shock...  
WO/2013/044371A1
A compound according to Formula IA and IB, reversibly convertible under photochromic and electrochromic conditions between a ring-open isomer A and a ring-closed isomer B is provided. For substitutent groups, Z is N, O or S; each R1 is i...  
WO/2013/047044A1
The present invention is a composition for forming a film for liquid-immersion exposure, said composition containing the following: a polymer component (A) containing a polymer (a1) that has a constitutional unit (I) represented by diagr...  
WO/2013/043131A1
Disclosed herein is a process for preparing 5-hydroxymethylfurfural comprising the step of contacting a carbohydrate and a Brønsted acid in an alcoholic solvent comprising an alcohol selected from the group consisting of secondary alcoh...  
WO/2013/042138A3
A process for the preparation of 4-[4-[4-[4-[[(3R,5R)-5-(2,4-difluorophenyl) tetrahydro-5-(lH-l,2,4-triazol-l-ylmefhyl) -3-furanyl]mefhoxy] phenyl] -1 -piperazinyl] phenyl]-2-[(lS,2S)-l-efhyl-2-hydroxypropyl]-2,4-dihydro-3H-l ,2,4-triazo...  
WO/2013/042124A8
Compound of formula X wherein P1 is a fused-ring system comprising one 6-membered and two 5- membered rings; v indicates an S or R configuration; or individual isomers or pharmaceutically acceptable salts thereof, or mixtures thereof, in...  
WO/2013/042775A1
An aromatic amine derivative represented by general formula (1-1). In general formula (1-1), R2-R5 and R7-R10 are each independently a hydrogen atom or a substituent group. In general formula (1-1), R1 and R6 are represented by general f...  
WO/2013/041895A1
The invention relates to novel compounds of general formula (I), and their preparation, pharmaceutical preparations containing compounds of general formula (I), and the use of these compounds in therapeutic procedures. The invention also...  
WO/2013/042124A1
Compound of formula X wherein P1 is a fused-ring system comprising one 6-membered and two 5- membered rings; v indicates an S or R configuration; or individual isomers or pharmaceutically acceptable salts thereof, or mixtures thereof, in...  
WO/2013/041807A1
The present invention relates to compounds having the following formula (I-I): in which A represents a cycle chosen from the group comprising the aryl, heteroaryl, C5-8 cycloalkenyl, and heterocycloalkenyl groups, said cycle (A) being op...  
WO/2013/042769A1
This aromatic amine derivative is represented by general formula (1). In general formula (1), R2, R3, R4, R5, R7, R8, R9, and R10 each independently are a hydrogen atom or a substituent group. In general formula (1): R1 and R6 are repres...  
WO/2013/039184A1
An aromatic amine derivative represented by general formula (1). In general formula (1), R1 to R10 each independently are a hydrogen atom or a substituent group. In general formula (1), any one of R1 to R10 is represented by general form...  
WO/2013/039221A1
An aromatic amine derivative represented by general formula (1). In general formula (1), R1 to R10 each independently are a hydrogen atom or substituent group. In general formula (1), R1 is represented by general formula (2), and any one...  
WO/2013/040068A2
The presently disclosed subject matter provides methods of preparing synthetic prostacyclin analogues, including Beraprost, either as racemic mixtures or as single stereoisomers. Also provided are novel synthetic intermediates for use in...  
WO/2013/038430A1
Disclosed herein is 10-α/β-D-Arabinofuranosylundecenes of general Formula (II) or pharmaceutically acceptable salts thereof as anti-mycobacterial agents in vitro; (II) wherein R, R1 and R" are as defined herein in the specification. Th...  
WO/2013/038650A1
A compound represented by formula (1). (In the formula, A1 represents O, S, Si(Ar1)(Ar2), P(=O)(Ar3)(Ar4), a substituted or unsubstituted arylene group having 6 to 30 ring-forming carbon atoms, or a substituted or unsubstituted heteroary...  
WO/2013/038931A1
This method of cheaply and easily producing a 2-oxo-2H-cyclohepta[b]furan analogue useful as a pharmaceutical intermediate with high purity and high yields. In this method, a 2-oxo-2H-cyclohepta[b]furan analogue represented by general fo...  
WO/2013/040540A3
A composition comprising between 95 and 100% biobased succinic acid, MAS or DAS wherein at least 75 % of the carbons are biobased.  
WO/2013/040068A3
The presently disclosed subject matter provides methods of preparing synthetic prostacyclin analogues, including Beraprost, either as racemic mixtures or as single stereoisomers. Also provided are novel synthetic intermediates for use in...  
WO/2013/034048A1
The present invention relates to compounds of formula (I) that are useful as hepatitis C virus (HCV) NS5B polymerase inhibitors, the synthesis of such compounds, and the use of such compounds for inhibiting HCV NS5B polymerase activity, ...  
WO/2013/033899A1
The present invention relates to compounds of formula (I) that are useful as hepatitis C virus (HCV) NS5B polymerase inhibitors, the synthesis of such compounds, and the use of such compounds for inhibiting HCV NS5B polymerase activity, ...  
WO/2013/033971A1
The present invention relates to compounds of formula (I) that are useful as hepatitis C virus (HCV) NS5B polymerase inhibitors, the synthesis of such compounds, and the use of such compounds for inhibiting HCV NS5B polymerase activity, ...  
WO/2013/033081A2
A process is provided for carrying out an oxidation on a feed including levulinic acid and/or a levulinic acid oxidation precursor to succinic acid, one or more furanic oxidation precursors of 2,5-furandicarboxylic acid and a catalytical...  
WO/2013/033058A1
A process is provided for carrying out an oxidation on a sprayable feed including a furanic substrate to be oxidized and a catalytically effective combination of cobalt, manganese, and bromide components for catalyzing the oxidation of t...  
WO/2013/029555A1
Provided are lavendustin A derivatives, a preparation method and use thereof. The compounds are shown by the structure of formula (I), wherein R is alkyl, ether group, carbonyl, p-tolyl, five-membered heterocyclic group, five-membered su...  
WO/2013/029479A1
Disclosed in the present invention is a mycophenolic acid derivative shown by the following general formula (V) and the pharmaceutically acceptable salts thereof, wherein L1 is -O-R2, -QCOOR2 or -QCONR2R3, Q is C1~C10. Alkylidene or C1~C...  
WO/2013/033081A3
A process is provided for carrying out an oxidation on a feed including levulinic acid and/or a levulinic acid oxidation precursor to succinic acid, one or more furanic oxidation precursors of 2,5-furandicarboxylic acid and a catalytical...  
WO/2013/030131A1
The invention relates to a method for producing furfural by reacting pentose in water and in the presence of carboxylic acid and a heterogeneous acid catalyst, said method being carried out in an aqueous solution of carboxylic acid as th...  
WO/2013/030193A1
The present invention relates to γ,δ-unsaturated a-amino acids of general formula (I). The present invention also provides a versatile process for the stereospecific synthesis of said compounds of formula (I), involving a Wittig reacti...  
WO/2013/026724A1
The present invention relates to compounds of formula (IA) wherein QA is QA1 or QA2 P is P1, heterocyclyl or heterocyclyl substituted by one to five Z; and wherein A1, A2, A3, A4, G1, Z, R1, R2, R3 and R4 are as defined in claim 1; or a ...  
WO/2013/026737A3
The invention relates to a method for producing γ-hydroxycarboxylic esters and γ-lactones, which are suitable as aromatic substances, by electrochemical reductive cross-coupling of α,β-unsaturated esters with carbonyl compounds in an...  
WO/2013/026392A1
A 3-(α-methoxyl) methylene benzofuran-2(3H)-ketone synthesis method comprises the synthesis of O-hydroxy phenylacetic acid, the synthesis of lactone and the synthesis of an end product, with focus on lactone synthesis improvement, such ...  

Matches 701 - 750 out of 29,343