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Matches 1 - 50 out of 30,654

Document Document Title
WO/2018/222647A1
This disclosure relates, in part, to compounds of Formula (1) (including all stereoisomers), N-oxides of such compounds, and salts of such compounds and N-oxides: wherein wherein L, Y1, R1, J, Q1, R7, Y2, R9 and Q2 are as defined in the ...  
WO/2018/221888A1
Provided in the present invention are: a novel compound comprising a condensed ring structure containing two different heteroatoms in the molecule; and an organic light emitting element comprising same.  
WO/2018/216913A1
The present invention provides a novel compound and an organic light-emitting device using same.  
WO/2018/214959A1
Disclosed is a compound as shown in formula (I), an optical isomer thereof or a pharmaceutically acceptable salt thereof, and the present invention relates to the use of same in the preparation of a drug for treating FXR-related diseases.  
WO/2018/216823A1
Provided are novel compounds represented by the following general formula [1] or pharmaceutically acceptable salts thereof, that inhibit LpxC, as well as pharmaceutical drugs comprising those compounds or pharmaceutically acceptable salt...  
WO/2018/215799A1
The present invention relates to compounds of Formula (I) that function as inhibitors of bacterial metallo-beta-lactamases. The present invention also relates to processes for the preparation of these compounds, to pharmaceutical composi...  
WO/2018/214639A1
Disclosed are a 2-azacyclo-5-trifluoromethyl-8-nitrobenzo(thio)pyran-4-one compound, a preparation method therefor and the use thereof in a drug for treating and/or preventing infectious diseases caused by Mycobacterium tuberculosis. In ...  
WO/2018/215348A1
The present invention relates to a compound of formula 1 and an organic electronic device comprising an organic semiconductor layer, wherein at least one organic semiconductor layer comprises a compound of formula (1), wherein L1 has the...  
WO/2018/215801A1
The present invention relates to compounds of Formula I that function as inhibitors of BCL6 (B-cell lymphoma 6) activity: wherein X1, X2, R1, R2 and R3 are each as defined herein. The present invention also relates to processes for the p...  
WO/2018/210659A1
Heteroaryl compounds as agrochemical fungicides Formula (I) The present invention relates to heteroaryl compounds of formula (I) or a compound in the form of a stereoisomer, an agriculturally acceptable salt, a tautomer, an isotopic form...  
WO/2018/210992A1
The present invention relates to pyrimidine derivatives of formula (I) wherein (R1)n, R3, R4a, R5b, and Ar1 are as described in the description and their use in the treatment of cancer by modulating an immune response comprising a reacti...  
WO/2018/211278A1
The invention provides compounds of formula (I), stereoisomers and pharmaceutically acceptable salts thereof: (I) wherein A1 to A4, R1 and RP are as defined herein. Such compounds are suitable for use in the treatment or prevention of di...  
WO/2018/210987A1
The present invention relates to benzofurane and benzothiophene derivatives of formula (I) Formula (I) wherein (R1)n, R2, R3, R4a, R4b, R5a, R5b and Ar1 are as described in the description and their use in the treatment of cancer by modu...  
WO/2018/210661A1
The present invention relates to heteroaryl compounds of formula (I) or a compound in the form of a stereoisomer, an agriculturally acceptable salt, a tautomer, an isotopic form, a N-oxide, a S- oxide, a prodrug or mixture thereof. The p...  
WO/2018/213150A1
The application relates to phenyl- or naphthylsulfonamide derivatives of the structural formula (I). The compounds are described as inhibitors of USP30 (ubiquitin specific peptidase 30) useful for the treatment of conditions involving mi...  
WO/2018/210297A1
Disclosed are an intermediate of Eribulin and a preparation method therefor. In particular, disclosed are compounds as represented by formula II, formula III and formula V and a preparation method therefor. Ar is C1-10 alkyl substituted,...  
WO/2018/210988A1
The present invention relates to pyrimidine derivatives of formula (I) wherein (R1)n, R3, R4a, R4b, R5a, R5b and Ar1 are as described in the description and their use in the treatment of cancer by modulating an immune response comprising...  
WO/2018/210660A1
The present invention relates to heteroaryl compounds of formula (I) or a compound in the form of a stereoisomer, an agriculturally acceptable salt, a tautomer, an isotopic form, a N-oxide, a S-oxide, a prodrug or mixture thereof. The pr...  
WO/2018/210994A1
The present invention relates to phenyl derivatives of formula (I) Formula (I) wherein (R1)n, R3, R4 a, R4b, R5b and Ar1 are as described in the description and their use in the treatment of cancer by modulating an immune response compri...  
WO/2018/210658A1
The present invention relates to heteroaryl compounds of formula (I) or a compound in the form of a stereoisomer, an agriculturally acceptable salt, a tautomer, an isotopic form, a N-oxide, a S-oxide, a prodrug or mixture thereof. The pr...  
WO/2018/211277A1
The invention provides compounds of formula (I), stereoisomers, tautomers, pharmaceutically acceptable salts and prodrugs thereof: (I) wherein A1 to A6 and R1 to R4 are as defined herein. Such compounds are suitable for use in the treatm...  
WO/2018/209012A1
Disclosed are compounds of Formula (I) or a salt or prodrug thereof, wherein: X is CR4 or N; Y is CR5 or N; provided that only one of X and Y is N; (R1) is: or; wherein R1, R1a, R1b, R1c, R2, and R3 are define herein. Also disclosed are ...  
WO/2018/208064A2
The present invention provides a novel compound and an organic light emitting element using the same.  
WO/2018/207882A1
Provided are compounds that can have an inhibitory action on BET family proteins and are expected to be useful as agents for the prevention or treatment of, for example, autoimmune diseases and/or inflammatory diseases (for example, rheu...  
WO/2018/202524A1
The invention relates to compounds of formula (I), wherein Z, Y, A1, A2, A3, A4, X, R7, R8 and R9 have the above-mentioned meanings, and to methods and intermediate products for the production and use thereof for controlling animal pests...  
WO/2018/198975A1
Provided is a light-emitting element having excellent luminance life. Disclosed is a light-emitting element comprising a positive electrode, a negative electrode, a first organic layer provided between the positive electrode and the nega...  
WO/2018/198973A1
Provided is a composition that is useful for producing a light-emitting element having excellent external quantum efficiency. Disclosed is a composition comprising at least two types of compounds represented by formula (C-1), and a phosp...  
WO/2018/201126A1
The present disclosure is directed to compounds of formula (I) that modulate, e.g., address underlying defects in cellular processing of cystic fibrosis transmembrane conductance regulator (CFTR) activity. The compounds may be used for t...  
WO/2018/198971A1
Provided is a composition useful for manufacturing a light-emitting element having excellent light-emitting efficiency. A composition containing a phosphorescent compound represented by formula (1) and a compound represented by formula (...  
WO/2018/199797A1
The invention relates to the chemistry of organic compounds, pharmacology and medicine, and concerns the prevention and/or treatment of hyperproliferative diseases associated with the malignant transformation of cells expressing the enzy...  
WO/2018/198974A1
Provided is a light-emitting element having excellent luminance life. This light-emitting element comprises: a positive electrode; a negative electrode; and a first organic layer and a second organic layer provided between the positive e...  
WO/2018/199283A1
A composition containing a compound represented by formula (H-1) and a phosphorescent compound, wherein the amount of a compound that is contained as an impurity in said composition, and that has a molecular weight that is greater by 16 ...  
WO/2018/197714A1
The invention provides compounds of the formula (3): or a pharmaceutically acceptable salt or tautomer thereof. The compounds are useful in the treatment of cancers.  
WO/2018/192227A1
The invention relates to an organic compound with a triazine and benzimidazole core and an application thereof in an OLED device. The compound of the invention has a relatively high glass transition temperature and molecular thermal stab...  
WO/2018/194181A1
The present invention aims to provide a compound that may be useful for the prophylaxis or treatment of constipation and the like. The present invention provides a compound represented by the following formula (I) : wherein each symbol i...  
WO/2018/190352A1
A novel compound is provided which controls plant disease. This pyridone compound is novel and can control plant disease.  
WO/2018/189484A1
The present invention relates to a novel bithiophenic matrix for specific detection of alkaloids by MALDI-TOF mass spectrometry.  
WO/2018/189199A1
A 1,3,5-trisubstituted pyridinium salt of general formula I (I) wherein Xn- is a counterion in which n is an integer from 1 to 4; wherein R2 and R3 are each independently a substituent group comprising Ar, wherein Ar is an aryl or hetero...  
WO/2018/189340A1
The present invention relates to novel benzohydroxamic compounds of formula (I) and (II) and pharmaceutically acceptable salts, isomers and prodrugs thereof, exhibiting a high selective inhibitory activity against histone deacetylase 6 (...  
WO/2018/188795A1
The present invention relates to sulfonamide-, sulfinamide- or sulfonimidamide containing compounds which bind to the liver X receptor (LXRa and/or LXRß) and act preferably as inverse agonists of LXR.  
WO/2018/185185A1
Compounds of formula (I) as defined herein, to processes for preparing them, to pesticidal, in particular insecticidal, acaricidal, molluscicidal and nematicidal compositions comprising them and to methods of using them to combat and con...  
WO/2018/185191A1
Compounds of formula (I) as defined herein, to processes for preparing them, to pesticidal, in particular insecticidal, acaricidal, molluscicidal and nematicidal compositions comprising them and to methods of using them to combat and con...  
WO/2018/185187A1
Compounds of formula (I) as defined herein, to processes for preparing them, to pesticidal, in particular insecticidal, acaricidal, molluscicidal and nematicidal compositions comprising them and to methods of using them to combat and con...  
WO/2018/186440A1
The purpose of the present invention is to provide a novel 1- phenylpiperidine derivative and an agricultural/horticultural drug agent including the compound as an effective component, in particular a novel 1-phenylpiperidine derivative ...  
WO/2018/181345A1
Provided is a compound which has an Nrf2-activating activity and is expected to be useful as a prophylactic or therapeutic agent for diseases associated with oxidative stress, particularly hepatitis (e.g., non-alcoholic steatohepatitis (...  
WO/2018/177995A1
The invention relates, inter alia, to compounds of general formula (I). The invention also relates to methods for synthesizing the compounds of formula (I). The compounds according to the invention are in particular suitable for controll...  
WO/2018/183964A1
Isoquinoline compounds and their use as inhibitors of HPK1 (hematopoietic kinase 1) are described. The compounds are useful in treating HPK1 -dependent disorders and enhancing an immune response. Also described are methods of inhibiting ...  
WO/2018/177993A1
The invention relates, inter alia, to compounds of general formula (I). The invention also relates to methods for synthesizing the compounds of formula (I). The compounds according to the invention are in particular suitable for controll...  
WO/2018/172463A1
Processes for preparation of Brexpiprazole, intermediates used during preparation, and polymorphs of Brexpiprazole are provided.  
WO/2018/172852A1
The present invention includes novel substituted bicyclic compounds, and compositions comprising the same, that can be used to treat or prevent hepatitis B virus (HBV) infections in a patient. In certain embodiments, the compounds and co...  

Matches 1 - 50 out of 30,654