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Matches 201 - 250 out of 599

Document Document Title
WO/1994/029301A1
The present invention relates to a process for producing predominantly pure cis nucleoside analogues using a novel bicyclic intermediate of formula (III), wherein X is S, or O; Y is S, CH2, O or CH(R); wherein R is azido or halogen; and ...  
WO/1994/027594A2
There is disclosed stable copper(I) complexes and methods relating thereto. The stable copper(I) complexes comprise a copper(I) ion complexed by a multi-dentate ligand which favors the +1 oxidation state for copper. Methods of this inven...  
WO/1994/012478A1
This invention relates to compounds of formula (I) which are effective for inhibiting platelet aggregation, pharmaceutical compositions for effecting such activity, and a method for inhibiting platelet aggregation.  
WO/1994/009793A1
The invention is a method for the treatment of humans infected with HBV that includes administering an HBV treatment amount of an enatiomerically pure beta-D-dioxolanyl purine nucleoside of formula (I), wherein R is OH, Cl, NH2 or H, and...  
WO/1994/004154A1
A method and composition for the treatment of humans infected with HIV that includes the administration of an HIV treatment amount of an enantiomerically pure beta-D-dioxolanyl purine nucleoside of formula (I), wherein R is OH, Cl, NH2, ...  
WO/1993/009122A1
Tetrahydrobenzothienopyridines of formula (I), processes for their preparation and their use in the treatment and/or prophylaxis of CNS disorders (I).  
WO/1993/007128A1
This invention relates to substituted cyclic carbonyls and derivatives thereof useful as retroviral protease inhibitors, to pharmaceutical compositions comprising such compounds, and to methods of using these compounds for treating viral...  
WO1993002710A3  
WO/1993/002710A2
The present invention provides the use of a persistent aryloxy or arylthio free radicals, other than perhalo radicals, for the manufacture of a contrast medium for use in magnetic resonance imaging. Also provided are magnetic resonance i...  
WO/1993/002711A1
The present invention provides the use of a persistent $g(p)-system free radical for the manufacture of a contrast medium for use in magnetic resonance imaging, wherein the electron delocalising $g(p)-system of said radical comprises at ...  
WO/1993/002084A1
A process for the production of ambergris-type labdane spiroketals of general formulae (I) and (II), where R represents oxygen or sulphur, useful in the perfumery industry, the said process being characterized by the intramolecular cycli...  
WO/1992/010496A1
An asymmetric process for the preparation of enantiomerically pure $g(b)-L-(-)-1,3-oxathiolane-nucleosides that includes the initial preparation of the key chiral intermediates (2R,5R) and (2R,5S)-5-(O-protected)-2-(protected-oxymethyl)-...  
WO/1992/010479A1
Bicyclic and polycyclic amidic derivatives of glumatic, aspartic and 2-amino adipic acids having activities antagonistic to gastrin, of general formula (I) in which r is between 1 and 3 and R¿1? is selected from mono- and disubstituted ...  
WO/1992/010497A1
An asymmetric process for the preparation of enantiomerically pure beta-D-(-)-dioxolane-nucleosides. The enantiomerically pure dioxolane nucleosides are active HIV agents, that are significantly more effective than the prior prepared rac...  
WO/1992/005146A1
This invention is directed to a stereoselective process and useful intermediates for the preparation of substantially optically pure acid sensitive compounds including certain dibenzofuran-carboxamides and dibenzofurancarboxamide acids.  
WO/1991/013872A1
A therapeutically useful compound of formula (I) or pharmaceutically acceptable salts thereof where A and B are oxygen, sulfur or CH2, X is an amine moiety as defined herein and R1 and R2 are as defined herein having 5HT1A neuronal activ...  
WO/1991/012024A1
The invention relates to the use of carbon stable free radicals as image enhancements agents in Overhauser MRI.  
WO/1991/004256A1
Process for alkylatine protected spectinomycin enone derivatives in the gamma position in order to produce intermediates useful in the synthesis of 6'alkylspectinomycins. The intermediate have formula (III) which comprises reacting a com...  
WO/1991/002741A1
The invention provides a novel class of versatile intermediates, i.e. 1,4 cyclic sulfates of sugar alcohols having protected hydroxy groups, such as 1,4 cyclic sulfates of D-mannitol having protected 2-, 3-, 5- and 6-hydroxy groups and D...  
WO/1988/005047A1
Novel carbamoyloxylabdanes, intermediates and processes for the preparation thereof, and methods for reducing intraocular pressure and treating cardiac failure utilizing compounds and compositions thereof.  
JP2020164541A
[Subject] a polycyclic compound, its synthesizing method, and the medicine constituent containing the compound -- and -- especially -- offer of the directions for a mental disease and schizophrenia. [Means for Solution] A compound illust...  
JP2020152714A
[Subject] Offer of a compound which can manufacture a resist pattern by good line edge roughness (LER), and a resist composition containing this. [Means for Solution] For example, the following compound (reaction product). For example, a...  
JP6661070B2  
JP2019531302A
The present invention relates to the many forms, solvent Japanese food , Enantiomer , stereoisomeric form, and hydrate which can permit the compound concerned and the compound concerned pharmacologically. A therapeutic method of the medi...  
JP2019182866A
To provide a photochromic compound capable of developing excellent photochromic characteristics and of suppressing white turbidness of the cured body in various cured bodies.A photochromic compound characterized by having an oligomer cha...  
JP6539760B2  
JP2019514863A
17-chloro 5, 13, and 14, 22-tetramethyl 28- Oxa - 2, 9-dithia 5, 6, 12, and 13, and 22- Penta aza-heptacyclo [27.7. 1.14, 7.011, 15.016, 21.020, 24.030, 35] Octa -- doria -- contour 1 (37), The compound which is 4 (38), 6, 11, 14, 16, 18...  
JP2019066659A
To provide: a chemically amplified positive photosensitive resin composition capable of suppressing occurrence of "footing", in which a width of a bottom (a side proximal to the surface of a support) becomes narrower than a top (a side p...  
JP2019052093A
To provide a method for obtaining 2-methylspiro(1,3-oxathiolane-5,3')quinuclidine sulfate at a high isomer ratio (cis/trans) from 3-hydroxy-3-mercaptomethylquinuclidine without requiring fractionation of isomers or an isomerization step....  
JP2019508376A
The present invention is general formula (I).The inside of a formula, Y, Y', Z, Z' and X and the structure unit (D) that has coefficient o, p, and q1~D3And A1And A2It is related with Is and the compound defined as indicated by Claim 1, r...  
JP6477339B2  
JP6420143B2  
JP2018168196A
To provide novel compounds useful for manufacturing salacinol, a method for manufacturing the compounds, a method for manufacturing salacinol, methods for protecting and deprotecting a diol group, and a protective agent for a diol group....  
JP2018531213A
The present invention relates to composition and application of cancer, other diseases and histone deacetylase useful for the medical treatment of an obstacle especially inhibitor of HDAC8, and the inhibitor. The present invention relate...  
JP2018131443A
To provide a resist composition that can improve lithography properties, a resist pattern forming method prepared with the resist composition, and a compound useful as the resist composition.The present invention provides a compound repr...  
JP6334876B2  
JP2017505995A5  
JP2018505203A
The new tricyclic compound which can combine the present invention with FXR and can work as a modulator of FXR, Or it is related with use of the compound concerned for the medical treatment of the stereoisomeric form, geometric isomer, a...  
JP6268014B2  
JP2017537933A
The present invention relates to those use as a new antimicrobial compound, the medicine constituent containing them, and antibacterial medicine.  
JP2017214422A
To provide novel compounds useful for manufacturing salacinol, a method for manufacturing the compounds, a method for manufacturing salacinol, methods for protecting and deprotecting a diol group, and a protective agent for a diol group....  
JP6243608B2  
JP6224004B2  
JP2017122100A
To provide compounds to be photoacid generators (PAGs) having greater diffusion control and attendant properties such as resist profile and photoresist compositions including the same.A photoacid generator compound has formula (I): [A-(C...  
JP2017043590A
To provide a compound that gives a polymer that can contribute to excellent open-circuit voltage and/or excellent photoelectric conversion efficiency when used for an organic thin film solar cell.The present invention provides a compound...  
JP2017505995A
The present invention is the compound guided from Acceptor * donor * Acceptor (A*D*A) cage Gothic Offen based on hetero Acencore , and relates to a compound of formula (I) used as an electron hole transportation material in an optical el...  
JP2017505350A
In this specification, a change sugar compound, an imino sugar compound, an aza-sugar compound, and the method of producing them are written. One or more of these change compounds contain Sulfate , Sulfit , a Sulfa mart, and/or Sulfone a...  
JP2017031152A
To provide novel organic electroluminescence devices.The present invention provides spiro condensed organic devices of an aromatic or heteroaromatic ring system having 5 to 40 aromatic ring atoms illustrated by formula (6a).SELECTED DRAW...  
JP2017031098A
To provide a manufacturing method of dialkyl dithienobenzodifuran.There is provided a manufacturing method of dialkyl dithienobenzodifuran represented by the following general formula (1) by continuous processes of at least (A) to (E). (...  
JPWO2014129446A1
A subject of the present invention is providing a streptoavidin mutant which reduced compatibility over natural biotin, and providing a biotin change object which has high compatibility to a streptoavidin mutant of low compatibility to t...  

Matches 201 - 250 out of 599