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Matches 701 - 750 out of 6,579

Document Document Title
JP2016047827A
To provide: cefquinome acid addition salt particles that have physical stability; and suspensions of cefquinome acid addition salt that are more stable, preferably cefquinome sulfate particles.An acid, preferably sulfuric acid, is added ...  
JP2012529443A5  
JP5864547B2  
JP5859436B2  
JP5852559B2  
JP5852562B2  
JP2015535849A
The present invention is obtained to the functional group in a compound, or the hetero atom of a heterocyclic system by producing and cheating out of the covalent bond of the ornamentation agent of the structure specified by formula 1, T...  
JP2015535210A
The present invention relates to a manufacturing method of an intermediate for manufacturing 2* Alkyl cephem compound useful as an antibacterial medicine. The present invention oxidizes a compound shown by formula (I), or its salt, and p...  
JP2015534995A
The compound of formula (I) of the present invention has an extensive antibacterial spectrum, and is related with 2* substitution cephem compound in which powerful antibacterial activity is especially shown to beta* lactamase production ...  
JP2015531378A
Sample 、 of the constituent containing beta lactam compound and crystalline タゾバクタム arginine, related methods, and these constituents is provided by this indication.  
JP2015155435A
[Subject] Offer of broadband-spectrum beta* lactamase inhibition medicine in which powerful antibacterial activity is shown. [Means for Solution] A compound denoted by formula (I) designed so that a compound might produce a reactant port...  
JP2014513700A5  
JP5733856B2  
JPWO2013051597A1
式(I)[式中、Aは、式(i)〜(iii )のいずれかであり、Bは式(v)または( vi)であり、Eは、置換もしくは非置換の カチオン性窒素原子を有する複素環式基...  
JPWO2013051597A
A is either of formula (i) * (iii) s among a formula (I) [type. B is formula (v) or (vi) and E is a heterocyclic machine which has substitution or an unsubstituted cationic nitrogen atom. Salt permitted on the compound shown by], or its ...  
JPWO2013002215A
The present invention has an extensive antibacterial spectrum and provides a new molecular entity in which strong antibacterial activity is especially shown to beta* lactamase production gram negative bacteria. Specifically, the present ...  
JPWO2013002215A1
本発明は、広範な抗菌スペクトルを有し、特 にβ−ラクタマーゼ産生グラム陰性菌に対し い抗菌活性を示す新規化合物を提供する。 体的には、本発明は、式(I)(式中...  
JP2014528965A
The present invention is a cephalosporin antibacterial-properties compound of formula (I) :Or it is related with the treating method of the infection caused especially with Gram-negative bacteria of the corresponding pharmacologically pe...  
JPWO2012147773A
The present invention has an extensive antibacterial spectrum and provides a new molecular entity in which strong antibacterial activity is especially shown to beta* lactamase production gram negative bacteria. Specifically, the present ...  
JP2012513957A5  
JP2014513700A
The present invention relates to the method and compound for adjusting discharge of the nitric oxide near a biofilm formation microorganism, adjusting the programmed cell death in a microorganism generally, and this promoting distributio...  
JP2014513116A
The present invention is formula (I).The preparing method of those use for the disposal of the infection in の new cephalosporin derivatives, those similar objects, and a mammal, the medicine constituents containing those new molecular ...  
JP5498393B2  
JP2014510750A
The present invention relates to the new cephalosporin derivative expressed with chemical formula 1 of a specification. In chemical formula 1, they are X, Y, L, and R.1R2は -- it is the same as what is defined during detailed explanatio...  
JP2014065732A
To provide a cephem compound having wide antibacterial spectrum against various bacteria including gram-negative bacterium and/or gram-positive bacterium, and to provide a pharmaceutical composition containing the same.There are provided...  
JP5451743B2  
JPWO2011136268A
A cephem compound shown in the following formulas having an extensive antibacterial spectrum, and in which showing strong antibacterial activity to beta* lactamase production gram negative bacteria especially and a medicine constituent c...  
JPWO2011125966A
Formula:(X are *N=, *CH=, etc. among a formula and W is *CH.)2* etc. -- it is -- U is *S* etc. -- R1And R2It is low-grade アルキル etc. which may achieve がそれぞれ independence and may have a hydrogen atom, halogen, and a subst...  
JPWO2011125967A
Formula:(X are *N=, *CH=, etc. among a formula and W is *CH.)2* etc. -- it is -- U is *S* etc. -- R1And R2It is low-grade アルキル etc. which may achieve がそれぞれ independence and may have a hydrogen atom, halogen, and a subst...  
JP5230934B2  
JP2013526502A
The present invention relates to the method of having been improved which oxidizes a 3* hydroxy * methyl * cephem derivative to a corresponding 3* ホルミル * cephem derivative. Especially this oxidation method is 10*I*3 type hyperval...  
JPWO2011093294A
At a simple process, a cephalosporin derivative with high content of Z object which carries out the object, or its alkali metal salt is industrially provided by an advantageous method. Iodine adsorption performance measured in solution o...  
JP5161269B2  
JP2013047267A
To provide new antibiotics that are highly effective against antibiotic-resistant strains.This invention provides a novel cross-linked glycopeptide-cephalosporin compound useful as an antibiotic and a pharmaceutically-acceptable salt the...  
JP2012533596A
The method for manufacture of the particles of the セフキノム acid addition salt by settling the セフキノム acid addition salt which adds acid, preferably sulfuric acid in solid in solution, preferably sulfate from セフキノ...  
JP2012529443A
The high permeability constituent (HPC) or prodrug (HPP) of an antibacterial medicine and an antibacterial medicine related compound is provided. Since it is convertible into a parent medicine or drug metabolite after passing a biologica...  
JP2012528102A
the present invention -- an organic compound -- especially (6R, 7R) *7* [(Z) *2* (5* amino * [1, 2, 4] thiadiazole *3* イル) * [[2* hydroxy imino * acetylamino] *8* oxo *3*] (E) * (R) -- *1'* (5* methyl *2* oxo * [1, 3] * ジオキ sol...  
JP2012528103A
the present invention -- an organic compound -- especially (6R, 7R) *7* [(Z) *2* (5* amino * [1, 2, 4] thiadiazole *3* イル) * [[2* hydroxy imino * acetylamino] *8* oxo *3*] (E) * (R) -- *1'* (5* methyl *2* oxo * [1, 3] * ジオキ sol...  
JP5047418B2  
JP5027042B2  
JP4990462B2
A process which comprises(i) acylating a compound of formula IIwith a compound of formula IVto obtain a compound of formula Iand(ii) deformylating said compound of formula I to obtain a compound of formula III  
JP2012513957A
[Subject] [Means for Solution] It has a clear merit, like solubility of セフジニル 酸式複塩 is high and living thing availability is high, can make to an oral solid tablet and an injectable solution, and demonstrates better the ...  
JP4953501B2  
JP2012511027A
The present invention provides a constituent of a new high permeability constituent (HPC) or a medicine constituent of a parent compound which can pass a biological barrier at high penetration efficiency. After HPC passes along one or mo...  
JPWO2010050468A
Formula having an extensive antibacterial spectrum and in which showing strong antibacterial activity to beta* lactamase production gram negative bacteria especially:(As for B, such as low-grade Al Killen, in A and G, such as S, D, such ...  
JP4856795B2  
JP4749533B2  
JP2011520866A
The present invention relates to an improved process for the preparation of Cefozopran of formula (I), its hydrochloride, its hydrate and its solvate. The present invention more particularly provides a process for preparing Cefozopran hy...  
JP4705199B2  
JP2011516595A
A solid DMSO solvate of a compound of formula (I) is described, which is a useful intermediate for preparing the broad spectrum antibiotics Ceftobiprole and Ceftobiprole Medocaril.  

Matches 701 - 750 out of 6,579