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Matches 51 - 100 out of 829

Document Document Title
WO/2010/103857A1
Disclosed are a novel method for the synthesis of a glycopeptide by which glycopeptides of various types can be deprotected and excised from a resin, each under weakly acidic to weakly basic conditions, without causing the problems of th...  
WO/2009/102022A1
Provided is a 3,6-O-bridged pyranose inversion compound useful as a β-O-glycosylating agent for use in selectively and easily producing β-O-pyranoside. The 3,6-O-bridged pyranose inversion compound is represented by general formula (1)...  
WO/2008/148549A3
The invention relates to a process for the catalytic conversion of a carbohydrate, an alcohol, an aldehyde or a polyhydroxy compound in the presence of a catalyst containing gold in a solvent.  
WO/2009/014970A1
Methods of synthesizing sodium glucose co-transporter 2 inhibitors, as well as compounds useful therein, are disclosed. Particular inhibitors are compounds of formula (I).  
WO/2008/152386A1
The invention relates to a process for preparing furanose derivatives, to furanose intermediates used in said process and to the use of said derivatives in the manufacture of atorvastatin.  
WO/2008/148549A2
The invention relates to a process for the catalytic conversion of a carbohydrate, an alcohol, an aldehyde or a polyhydroxy compound in the presence of a catalyst containing gold in a solvent.  
WO/2008/111526A1
Disclosed is a method for producing an oxazoline derivative from a non-protected sugar in a simple manner. Also disclosed is a method for producing a glycoside by utilizing the product of the aforementioned method. A sugar oxazoline deri...  
WO/2008/096880A1
It is intended to develop a method of effectively synthesizing a glycolipid that has never been established so far. Thus, a method for synthesizing a glycolipid is provided. This method comprises the following steps: (a) the step wherein...  
WO/2008/068413A2
The invention relates to a method for preparing acetyl,docosahexaenoyl-glycerophosphocholine (AcedoPC) and to the use thereof for the delivery of DHA and Neuroprotectin D1.  
WO/2007/108009A1
The present invention provides novel process for the preparation of Topiramate Form I which comprising purifying crude Topiramate base by treating the same with mixture of acetone and water to obtain topiramate of at least 99.5% purity.  
WO/2007/099388A1
An improved process for the manufacture of 2,3:4,5-bis-O-(1-methylethylidene)-β-D-fructopyranose sulfamate, viz. Topiramate is reported. It consists of subjecting an intermediate of the formula 2,3:4,5-bis-O-(1-methylethylidene)-β-D-fr...  
WO/2007/093769A1
This invention provides a method for inhibiting oligosaccharide biosynthesis in vivo and in vitro comprising the steps of administering at least one monosaccharide derivative, wherein the hydroxyl group which is the glycosyl acceptor (i....  
WO/2006/111783A1
The present invention relates to monosaccharide derivatives as anti-inflammatory agents. The compounds disorder herein can be useful for inhibition and prevention of inflammation and associated pathologies including inflammatory and auto...  
WO2005081904A3
Compositions useful for inhibiting the growth of bacteria, including bacteria that can cause gastric ulcers, are provided. In addition, transgenic organism that can produce such compositions are provided. Methods of using the composition...  
WO2005092907B1
The present invention relates to monosaccharide derivatives as anti-inflammatory agents. The compounds disorder herein can be useful for inhibition and prevention of inflammation and associated pathologies including inflammatory and auto...  
WO2005092907A3
The present invention relates to monosaccharide derivatives as anti-inflammatory agents. The compounds disorder herein can be useful for inhibition and prevention of inflammation and associated pathologies including inflammatory and auto...  
WO2005100373A3
The present invention relates to monosaccharide derivatives as anti-inflammatory agents. The compounds disclosed herein can be useful for inhibition and prevention of inflammation and associated pathologies, including inflammatory and au...  
WO2005062748A3
Bicyclic carbohydrates for the treatment of infections caused by herpseviridae, and in particular cytomegalovirus. The invention consists of the novel bicyclic carbohydrates the generic structure of which is formula I: wherein R
WO/2005/100373A2
The present invention relates to monosaccharide derivatives as anti-inflammatory agents. The compounds disclosed herein can be useful for inhibition and prevention of inflammation and associated pathologies, including inflammatory and au...  
WO/2005/092907A2
The present invention relates to monosaccharide derivatives as anti-inflammatory agents. The compounds disorder herein can be useful for inhibition and prevention of inflammation and associated pathologies including inflammatory and auto...  
WO/2005/062748A2
Bicyclic carbohydrates for the treatment of infections caused by herpseviridae, and in particular cytomegalovirus. The invention consists of the novel bicyclic carbohydrates the generic structure of which is formula I: wherein R1 is eith...  
WO2005016514A3
Methods are disclosed for providing a library of composite or novel composition samples on a support. The method involves depositing one or more components as concentration gradients on the surface of the support. The concentration gradi...  
WO2004075843A3
It is taught here that enkephalin peptides which are glycosylated with a disaccharide will be transported across the blood brain barrier and deliver analgesic effects superior to morphine when introduced into the bloodstream. Glycosylate...  
WO2004104163A3
A method of alpha-selective glycosylation comprising forming a cyclic protective group having a silyl acetal structure over hydroxyl groups at the 4- and 6-positions in a hexose or higher saccharide structure, which is a monosaccharide o...  
WO/2005/016514A2
Methods are disclosed for providing a library of composite or novel composition samples on a support. The method involves depositing one or more components as concentration gradients on the surface of the support. The concentration gradi...  
WO2004089965A3
A process of preparing topiramate of the Formula (I) which comprises the following reaction steps and topiramate prepared thereby, compositions containing the same, therapeutic uses thereof and methods of treatment employing the same.  
WO2004074303A3  
WO/2004/104163A2
A method of &agr -selective glycosylation comprising forming a cyclic protective group having a silyl acetal structure over hydroxyl groups at the 4- and 6-positions in a hexose or higher saccharide structure, which is a monosaccharide o...  
WO/2004/099229A1
The present invention relates to processes for the synthesis of base addition salts of particular ß-L- gulofuranosides. More specifically, the invention relates to synthetic processes for making base addition salts of 2,3-O-isopropylide...  
WO/2004/089965A2
A process of preparing topiramate of the Formula (I) which comprises the following reaction steps and topiramate prepared thereby, compositions containing the same, therapeutic uses thereof and methods of treatment employing the same.  
WO2004034960A3
The present invention relates to pentose and pentose derivatives that are effective at increasing glucose transport in a non-insulin dependent manner, and to uses thereof for a) treating and/or preventing hyperglycemia; b) treating and/o...  
WO/2004/078769A1
The present invention is directed to a one-step process for the preparation of fructopyranose sulfamate derivatives of general formula (I), wherein X, R1, R3, R4, R5 and R6 are as described in the specification.  
WO/2004/075843A2
It is taught here that enkephalin peptides which are glycosylated with a disaccharide will be transported across the blood brain barrier and deliver analgesic effects superior to morphine when introduced into the bloodstream. Glycosylate...  
WO2004032625A3
This invention relates to devices, kits, and methods for eliminating termite colonies. The kits, devices, and methods employ a termiticidal bait matrix containing a) a termiticide selected such that the termiticide causes death to about ...  
WO/2004/074303A2
The present invention provides methods for preparing LPS antagonist lipodisaccharide B1287 and stereoisomers thereof, which compounds are useful as in the prophylactic and affirmative treatment of endotoxemia including sepsis, septicemia...  
WO2003000200A3
The present invention includes compounds and compositions of beta -halonucleosides, as well as methods to treat HIV, HBV or abnormal cellular proliferation comprising administering said compounds or compositions.  
WO/2004/063210A1
The invention relates to novel pharmaceutically acceptable salts of anticonvulsant derivatives, processes for preparation of and pharmaceutical compositions containing said salts, useful in the treatment of epilepsy.  
WO/2004/050676A1
A method in which a glucide, examples of which include a monosaccharide, an oligosaccharide, a polysaccharide, a composite saccharide comprising any of these saccharides and a protein or lipid bonded thereto, a polyalcohol, an aldehyde, ...  
WO2003097656A3
The present invention is directed to novel compounds of the formula (I) wherein X, R1, R2 , R3, R4, R5 and R6 are as described in the specification, processes for the preparation of and pharmaceutical compositions comprising said derivat...  
WO/2004/041836A1
The present invention is directed to a continuous process for the preparation of fructopyranose sulfamate derivatives of the general formula (I) wherein R1, R3, R4, R5, R6 and X are as herein defined. The present invention is further dir...  
WO/2004/034960A2
The present invention relates to pentose and pentose derivatives that are effective at increasing glucose transport in a non-insulin dependent manner, and to uses thereof for a) treating and/or preventing hyperglycemia; b) treating and/o...  
WO/2004/032625A2
This invention relates to devices, kits, and methods for eliminating termite colonies. The kits, devices, and methods employ a termiticidal bait matrix containing a) a termiticide selected such that the termiticide causes death to about ...  
WO2004005308A3
This invention relates to processes for production of alkylamino glucosaminide phosphate compounds, and of disaccharide compounds, including various novel intermediates and intermediate processes. In one aspect, glycosyl halides are prod...  
WO2003087118A3
The invention relates to a novel method, essentially having four stages, for producing beta-L-2'-deoxy-thymidine with L-arabinose as the starting material. The inventive method is particularly useful for the large-scale production of bet...  
WO2003032905A3
Novel carbohydrate-based compounds with an attached ring system that have antimicrobial or cytostatic activity. The compounds are administered to humans and animals for the treatment or amelioration of bacterial, fungal, viral or protozo...  
WO/2004/005307A1
Enantiomerically enriched (S)-(-)-3-N-methylamino-l-(2-thienyl)-1-propanol or (R)-(+)-3-N-methylamino-l-(2-thienyl)-l-propanol of the formulae, or mirror image are prepared by i) treating an enantiomeric mixture of the amines Ia and Ib w...  
WO/2004/005308A2
This invention relates to processes for production of alkylamino glucosaminide phosphate compounds, and of disaccharide compounds, including various novel intermediates and intermediate processes. In one aspect, glycosyl halides are prod...  
WO2002069704A8
This invention relates to devices, kits, and methods for eliminating termite colonies. The kits, devices, and methods employ a termiticidal bait matrix containinga) a termiticide selected such that the termiticide causes death to about 5...  
WO/2003/105580A1
This invention relates to devices, kits, and methods for eliminating termite colonies. The kits, devices, and methods employ a termiticidal bait matrix containing a) a termiticide selected such that the termiticide causes death to about ...  
WO/2003/106395A1
This invention relates to devices, kits, and methods for eliminating termite colonies. The kits, devices, and methods employ a termiticidal bait matrix containing a) a termiticide selected such that the termiticide causes death to about ...  

Matches 51 - 100 out of 829