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Matches 301 - 350 out of 850

Document Document Title
JP2014001230A
To provide a compound useful for synthesis of a sodium glucose co-transporter 2 inhibitor.Provided is a compound represented by the following formula. Further, provided are specific compounds obtained from the compound, such as (4-chloro...  
JP5380293B2  
JP2013541596A
The invention is directed to compounds for selectively inhibiting glycosidases, uses of the compounds and pharmaceutical compositions including the compounds, and methods of treating diseases and disorders related to deficiency or overex...  
JP2013213037A
To provide compounds for selectively inhibiting glycosidases, prodrugs of the compounds, uses of the compounds or prodrugs, pharmaceutical compositions including the compounds or prodrugs of the compounds, and methods of treating disease...  
JP5301427B2
Disclosed is a process for producing an oxazoline derivative from a non-protected sugar in a simple manner. Also disclosed is a process for producing a glycoside by utilizing the product of the aforementioned process. A sugar oxazoline d...  
JP2013531654A
This application indicates the preparing method of 5* deoxy *L* arabinose of formula (VI) containing the step which changes the compound of formula (XII) (the inside of a formula and n are 0, 1, or 2) which can be used as an intermediate...  
JP5258798B2  
JP2013136625A
To provide methods for preparing LPS antagonist lipodisaccharide B1287 and stereoisomers thereof, which compounds are useful in the prophylactic and affirmative treatment of endotoxemia including sepsis, septicemia and various forms of s...  
JP2013107885A
To provide a method of conjugating peptides and proteins by means of glycosyltransferase.It is an object of the invention to provide means and methods which allow for a convenient synthesis or semisynthesis of therapeutic proteins, where...  
JP5154954B2  
JP2013505267A
The process and intermediate for composition of the nucleoside of pyrrolo [of formula I] [1, 2*f], and [1, 2, 4] thoriadinyl and imidazo [1, 2*f], and [1, 2, 4] thoriadinyl heterocycle are provided.Formula I  
JP2013503207A
- (1S, 4R) 2-オキサ- 3-azabicyclo [2.2. 1] hept 5-エン which is denoted by the following formulas and which was condensed in enantiomorphism, [Formula 1]The inside of a formula, PG1It is prepared via; hetero ディールス Alder cy...  
JPWO2011021398A1
下記式(I)〜(V)で表されるグルコース 、マンノース、プシコース、ソルボース、タ ガトース、アロース、アルトロース、グロー ス、イドース、タロースのピラノース誘...  
JPWO2011021398A
The pyranose derivative and furanose derivative (inside of a formula, M) of glucose, mannose and プシコース which are denoted by following formula (I) * (V), Sol Bose, タガトース, アロース, an alto sirloin, Glaus, イドー...  
JP5099653B2  
JPWO2010150789A1
不要な保護基の変換工程を必要とせず、効率 が良く簡便に、高収率で、NC型ヌクレオシ ドを合成するための新たな製造方法を提供す る。式(I):で表される化合物を反転...  
JPWO2010150789A
A conversion process of an unnecessary blocking group is not needed, but a new manufacturing method for efficiency to compound NC type nucleoside by quantity 収率 simple well is provided. Formula (I) :It comes out, a compound expressed...  
JP5078108B2  
JP2012528198A
this indication -- anhydro pliers トール and ケタール compound; from oxo carboxylate -- the derivative, a homopolymer, and copolymer; -- and -- and it is related with various constituents guided, a tablet, and manufacture of an ar...  
JPWO2010110382A
Offer of the new molecular entity contained in a blue rose. It is contained in a blue rose and the new molecular entity concerning the present invention is following general formula (I) :{Inside of a formula, R1It is a basis given in the...  
JPWO2010110382A1
青いバラに含まれる新規化合物の提供。本発 明に係る新規化合物は、青いバラに含まれ、 下記一般式(I):{式中、R1は、請求の 範囲1に記載の基であり、かつ、R2は...  
JP4992074B2  
JP2012509268A
[Subject] Offer of the manufacturing method of a deoxyribo furanose compound. [Means for Solution] The present invention relates to a method of manufacturing deoxyribo furanose compounds, such as a compound (2). The above-mentioned deoxy...  
JP4920163B2  
JP4892191B2  
JP4877695B2  
JP2004510700A5  
JP4866515B2  
JP2012502024A
The present invention is [1S* [1alpha, and 2alpha and 3beta (1S).*, 2R*), 5beta]] *3* [7* [2* (-- three -- four -- * -- difluoro one -- phenyl --) -- * -- cyclobutylpropylamino --] -- * -- five -- * (pro ピルチオ) -- * -- three -- H ...  
JP2012006845A
To develop a multistage reaction in a fluorous multiphase system dispensing with concentration operation in the middle of synthesis, usable of a separated fluorous phase for the next reaction as it is, because a multistage synthesis of a...  
JP2011254780A
To provide a method of producing a novel sugar derivative by utilizing C6 sugars such as glucose and C5 sugars such as xylose by using microorganisms.This method of producing chemical compound expressed by the following formula (1) compr...  
JP4825353B2  
JP4825322B1
The use for medical treatment of a disease, a state, and/or an obstacle which are carried with a compound of formula (I) and sodium * glucose transporter inhibitor (especially SGLT2 inhibitor) is written in this specification. A compound...  
JP2011184365A
To provide an organic nanotube in which a π-electron aromatic compound having optical, electronic, and energy characteristics is introduced at high density, and to provide a simple method for producing the same.An ester obtained by dehy...  
JP4773336B2  
JP4726477B2  
JP4725976B2  
JPWO2009102022A1
本発明は、β−O−ピラノシドを選択的に、 かも簡便に製造するためのβ−O−グリコ ル化剤として有用な3,6−O−架橋反転 ラノース化合物を提供することを課題...  
JP2011516478T
In the medical treatment and prevention of the fall of microorganism infection and an immunity system, the disease from which the cell serves as an obligate anaerobiosis, and a cell-growth disease including cancer, the present invention ...  
JP2011516478A
In the medical treatment and prevention of the fall of microorganism infection and an immunity system, the disease from which the cell serves as an obligate anaerobiosis, and a cell-growth disease including cancer, the present invention ...  
JP2011037885A
To provide methods for preparing LPS (linear programming system) antagonist lipodisaccharide B1287 and stereoisomers thereof.The invention provides methods for preparing LPS antagonist lipodisaccharide B1287 useful in the prophylactic an...  
JP4610197B2  
JP2010285446A
To provide processes for producing alkylamino glucosaminide phosphate compounds and disaccharide compounds functioning as immunoeffectors or adjuvants intended for vaccines and the like comprising various novel intermediates and intermed...  
JP4599295B2  
JP4577478B2  
JP2003012683A5  
JP2010189410A
To provide a new aminobenzophenone derivative which has excellent physicochemical properties, especially has improved bioavailability, and is pharmacologically active.The new aminobenzophenone derivative is represented by general formula...  
JP2010528048A
A method for preparing isofagomine, its derivatives, intermediates and salts thereof using novel processes to make isofagomine from D-(-)-arabinose and L-(-)-xylose.  
JP4504018B2  
JPWO2008111526A1
The manufacturing process of the glycoside which uses the manufacturing method in which an oxazoline derivative is simpler than unprotected sugar, and its output is provided. The sugar oxazoline derivative is compounded at one step of pr...  

Matches 301 - 350 out of 850