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Matches 351 - 400 out of 852

Document Document Title
JPWO2008111526A1
The manufacturing process of the glycoside which uses the manufacturing method in which an oxazoline derivative is simpler than unprotected sugar, and its output is provided. The sugar oxazoline derivative is compounded at one step of pr...  
JPWO2008096880A1
本発明は、未だ確立されていない効率的な糖 脂質合成法を開発することを課題とする。本 発明により、糖脂質を生成するための方法が 提供される。この方法は、以下:(a)...  
JP2010070541A
To provide a TG synthesis inhibitor effective for prevention or amelioration of hyperlipidemia and obesity.The TG synthesis inhibitor comprises as an effective ingredient thereof ellagitannin, having a partial structure represented by fo...  
JP2010070462A
To provide an industrially more advantageous method for producing 2,2'-anhydroarabinosylthymine which is a suitable intermediate for producing a nucleic acid derivative such as L-thymidine.A 2,2'-anhydro-5,6-dihydrouridine-5-alkoxymethyl...  
JP2010065038A
To provide conjugates of fatty alcohols and pharmaceutical agents useful in treating cancer, viral deseases, psychiatric disorders.Compositions (1) are expressed by chemical formula (1). In the formula, R is an 8-26C fat group of a fatty...  
JP4435305B2  
JP2010501598A
The invention provides compounds of formula (I) for selectively inhibiting glycosidases, prodrugs of the compounds, and pharmaceutical compositions including the compounds or prodrugs of the compounds. The invention also provides methods...  
JP4393863B2  
JP4347488B2  
JPWO2009102022A
The present invention makes it a subject to provide a useful as beta*O * glycosylation agent for manufacturing beta*O * pyranoside alternatively and simple 3, and 6*O* bridge construction reversal pyranose compound. A 3 of the present in...  
JP4294317B2  
JP2009515899A
The present invention is based, in part, on our discovery that certain types of therapeutic agents can be used in combination to treat a variety of neuropsychiatric and related disorders, including addiction (e.g., to a substance or to a...  
JP4251410B2  
JP2008545650A
[化 1] The present invention relates to the production method of a スルホニル imine derivative [especially, thing of the thing] of formula (XII) and the スルファミド derivative [, especially formula (I)]. This method under ex...  
JP4182218B2  
JP2002201372A5  
JP4162491B2  
JPWO2008111526A
A manufacturing process of a glycoside which uses a manufacturing method in which an oxazoline derivative is simpler than unprotected sugar, and its output is provided. The sugar oxazoline derivative is compounded at one step of processe...  
JP4153057B2  
JPWO2008096880A
The present invention makes it a subject to develop the efficient glycolipid synthesis method which is not yet established. The method for generating a glycolipid is provided by the present invention. This method makes the sugar and lipi...  
JP2008531604A
The present invention contains the pharmacological composite containing the prodrug of the compound for checking glycosidase alternatively, the prodrug of the compound and its compound, or a compound. The present invention includes the m...  
JP4097294B2  
JP2007530700A
The new compound useful to control, disposal, and prevention and method of fungus activity. [Selection figure] Nothing  
JP3992510B2  
JP2007527520A
The method of building the sample library of a complex or a new composite on a support medium is indicated. This method includes the method of giving a concentration gradient on the surface of a support medium, and making one or the ingr...  
JP2007230930A
To provide a glycosyl donor compound enabling stereoselective 1,2-cis glycosylation reaction. The compound is expressed by formula (1) (X1 and X2 are each independently hydrogen atom or hydroxyl-protecting group; Y is a 7-20C aralkyl gro...  
JP2007197362A
To obtain a sialic acid derivative as a saccharide donor, which forms a glycosyl bond having a high yield and high α selectivity in a glycosylation reaction of a saccharide receptor using a sialic acid as a saccharide donor. The sialic ...  
JP3942414B2
To provide a new efficient synthesis method for industrially producing an L-type nucleic acid derivative as a medicine. A method by which the L-type nucleic acid derivative can industrially be produced from L-arabinose, one of few indust...  
JP2002537326A5  
JP2002536328A5  
JP2004505004A5  
JP2006232861A
To provide a novel efficient synthetic method for industrially producing an L-nucleic acid derivative as a medicine.Provided is the method industrially producing the L-nucleic acid derivative in a short process by using L-arabinose which...  
JP2006519860A
the present invention -- general formula (I) -- the フルクト pyranose スルファ mate derivative denoted by [化 1 [the inside of a formula, X, R, R, R, R, and R are as describing on these specifications] ] is turned to the method ...  
JP2006518759A
When the エンケファ phosphorus peptide glycosylated by two sugar is carried out in a blood brain barrier, and is conveyed and it is introduced into a blood flow, producing the analgesic effect superior to morphine is taught. Two sug...  
JP2006518394A
The present invention offers the method for preparing LPS アンタゴニストリポ two sugar B1287 and its stereoisomeric form, and this compound, It is useful to the preventive disposal and the positive disposal of inner toxin 血症...  
JPWO2004104163A1
単糖体であり、又は二糖体以上のオリゴ糖な いし糖鎖の還元末端である6炭糖以上の糖構 造体における4位と6位の水酸基にわたって シリルアセタール構造の保護基を環状に...  
JP2006169157A
To provide a capping reagent quickly reactive with a hydroxy group in a capping reaction, and more stable in a deprotective reaction for a temporary protective group, and to provide a capping method using the reagent.The capping reagent ...  
JP3789951B2
PURPOSE: To obtain a new compound capable of producing hydantocidin in high yield without forming stereoisomers. CONSTITUTION: This sugar derivative is a compound of formula I [R1 and R2 each is H or together form a (substituted) alkylid...  
JP2006514071A
The present invention relates to the pharmaceutical composite which contains the manufacture methods of the new pharmaceutically permissible salt of a useful anticonvulsant derivative, and this salt, and this salt in the medical treatmen...  
JP2006508949A
the present invention -- general formula (I) -- the フルクト pyranose スルファ mate derivative denoted by [化 1 [the inside of a formula, R, R, R, R, R, and X are as defining by this specification] ] is turned to the method of m...  
JP2006052182A
To provide a method for producing a fluorinated purine nucleoside derivative, by which the 3-position (preferably the α-position) is economically and efficiently fluorinated and which is suitable for industrial production.This method fo...  
JP2006502103A
The present invention relates to the new palatinose condensate obtained by condensing disaccharide palatinose in 溶融物 of palatinose, water, and organic acid.  
JP3725233B2
To obtain a trehalose derivative excellent in surface-active ability and safety to skin and useful as a surfactant, etc., capable of using for cosmetics, medicines, foods, etc., by reacting trehalose with an acetal compound in the presen...  
JP2005536493A
The present invention relates to the production method of the アルキルアミノグルコサミニドホス compound which contains like various new intermediate fields and Takumi Nakama, and a disaccharide compound. Glycosyl halide i...  
JP2005289964A
To provide an efficient production method of a 2-deoxy-L-ribose compound and its protection compound.This production method comprises reacting an aldehyde compound represented by formula (1) (wherein R1 and R2 are each independently or i...  
JP3706875B2
To provide tea leaves with reduced caffeine content, capable of being taken by a large amount for a long time as an antiallergic beverage or food. A method for producing tea leaves is provided by immersing any of raw leaves of "Benifuuki...  
JP2005530808A
The present invention relates to the new pharmaceutically useful compound of tramadol hydrochloride and a トピラ mate which is an addition of 1: 1 stoichiometrically, and its manufacture and use.  
JP2005526813A
Are a compound of formula (I), and n is 0 or 1, and here; R6 and R7, Are hydrogen, or become together, form carbonyl oxygen, and; R1, Hydrogen; *N (Z) Y and *C (Z) When it is chosen from the group which consists of Y and R1 is *N (Z) Y h...  
JP2005526852A
[化 1] The present invention aims at the pharmaceutical composite containing the manufacturing process of the new compound of formula (I) which is as X, R, R, R, R, R, and R having written in the specification, and this derivative, and ...  
JP3662954B2
PURPOSE: To obtain the subject compound, useful for a raw material, etc., for liquid crystals, medicines, agrochemicals, etc., by optically resolving a recemic 1-benzyloxy-6,6,6-trifluoro-4-hexyn-3-ol, then carrying out the reduction of ...  

Matches 351 - 400 out of 852