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Matches 1 - 50 out of 816

Document Document Title
WO/2018/074926A1
The present invention relates to new bi-functional and polyfunctional bis- dioxolanes and bis-dioxanes. The present inventors have established that the bis- dioxolanes and bis-dioxanes of the invention are highly advantageous as building...  
WO/2018/055496A1
The present invention relates to a process for the preparation of crystalline Form G1 of Ertugliflozin (1). (I) The invention also relates to crystalline Form G l obtained by the process of the present invention, the said Form Gl being s...  
WO/2017/190568A1
Disclosed are an amine solvate of a sodium-glucose linked transporter (SGLT) inhibitor, and a preparation method and application thereof. The SGLT inhibitor is (1S,2S,3S,4R,5S)-5-(3-((2,3-dihydrobenzo[b][1,4]dioxin-6-yl) methyl)-4-ethylb...  
WO/2017/178513A1
The present invention relates to a method for preparing monomers via depolymerisation from lignocellulose-containing biomass.  
WO/2017/134606A1
The present invention relates to a crystalline Form B of {(1 R,2S,3S,4R,5S)-5-[4-chloro-3-(4-ethoxybenzylphenyl]- 2,3,4-trihydroxy- 6,8-dioxabicyclo [3.2. 1]oct-1-yl}methyl acetate of Formula (II) and a process for its preparation. The p...  
WO/2017/088839A1
This present invention relates to a complex of a glucopyranosyl derivative and L-pyroglutamic acid as a sodium dependent glucose cotransporter (SGLT) inhibitor, and preparation processes thereof, and a pharmaceutical composition containi...  
WO/2017/085144A1
The invention relates to new compounds of formulae: Wherein: R 1 and R 2 can be independently H; a C 1 to C 6 alkyl including methyl, ethyl, propyl, butyl; aryl including phenyl, para-methoxyphenyl; or R 1, R 2 together with the carbon C...  
WO/2017/047816A1
The present invention provides a method for producing guanidine crosslinked artificial nucleic acid (abbreviated hereinafter as GuNA), and an intermediate compound for the production thereof. Specifically, the present invention provides ...  
WO/2017/034004A1
[Problem] To provide a novel gelling agent containing a sugar derivative. [Solution] A gelling agent comprising a compound represented by the formula (1) or (2). (in the formulae: R1 represents a C9-20 straight or branched alkyl, a C13-2...  
WO/2016/173425A1
This present invention relates to a glucopyranosyl derivative as sodium dependent glucose cotransporters (SGLTs) inhibitor, preparation processes thereof, and pharmaceutical uses thereof, pharmaceutical compositions containing the compou...  
WO/2016/050134A1
Provided are an L-proline compound of a sodium-glucose cotransporter 2 inhibitor, and a monohydrate and a crystal of the L-proline compound. Specifically, provided are 1,6-dehydrated-1-C{4-chloro-3-[(3-fluoro-4-ethoxyphenyl)meth yl]pheny...  
WO/2016/000599A1
Disclosed are a C-benzo five-membered heteroaromatic ring aryl glucoside derivative represented by general formula (I), a preparation method for the derivative or an intermediate thereof, and a use of the derivative, wherein R, R1, R2, R...  
WO/2015/137838A1
A compound of formula I : or a salt thereof, wherein: R1 is -OC(H) (X) (CH2)nC(=O)OH; R2 is -OH, -N3, or -N (H) C (=O) CH3; or R1 and R2 together with the carbon atoms to which they are attached form R3 is -H, -CH3, -CH2C(=O)OH, or -CH2O...  
WO/2015/109049A1
Provided herein are glycomimetic E-selectin antagonist compounds of formula (I)) and pharmaceutical compositions comprising at least one of the same. The compounds of the present disclosure include trisaccharide domain mimics comprising ...  
WO/2015/043473A1
Provided herein are glucopyranosyl derivatives used as sodium dependent glucose cotransporters (SGLTs) inhibitors and pharmaceutical uses thereof, particularly 6,8-dioxabicyclo [3.2.1] octane derivatives represented by Formula (I), or ph...  
WO/2015/032272A1
The present invention relates to a C-aryl glucoside derivative, a preparation method for same, and medical applications thereof. Specifically, the present invention relates to compounds as represented by formula I, and, tautomers, enanti...  
WO/2015/027963A1
The present invention relates to an aromatic ring derivative, and pharmaceutical composition and use thereof, in particular to aromatic ring derivatives or hydrates as represented by general formula (II), solvates, stereoisomers thereof,...  
WO/2014/132468A1
Provided is a sugar chain compound as mentioned in item (a) or (b), which contains a 1,2-cis-type sugar residue: (a) a polysaccharide or oligosaccharide formed by repeatedly binding a sugar unit represented by formula (I) or (I'); and (b...  
WO/2014/125967A1
The present invention addresses the problem of providing a highly-versatile method for easily producing α-O-pyranosides with a high degree of selectivity without establishing severe reaction conditions, and a pyranose donor used in said...  
WO/2014/122621A3
The invention relates to the compounds of formula I and formula II or its pharmaceutical acceptable salts, as well as polymorphs, solvates, enantiomers, stereoisomers and hydrates thereof. The pharmaceutical compositions comprising an ef...  
WO/2014/094544A1
Provided are a phenyl C-glucoside derivative containing a deoxyglucose structure as represented by formula I, preparation method thereof, pharmaceutical composition containing same, and uses thereof in the preparation of drugs for treati...  
WO/2014/067003A1
The invention provides compounds with enhanced permeability for selectively inhibiting glycosidases, prodrugs of the compounds, and pharmaceutical compositions including the compounds or prodrugs of the compounds. The invention also prov...  
WO/2014/037832A3
The invention relates to the compounds of formula I or its pharmaceutical acceptable salts, as well as polymorphs, solvates, enatitiomers, stereoisomers and hydrates thereof. The pharmaceutical compositions comprising an effective amount...  
WO/2014/013181A1
The invention relates to a thiophene derivative of the following general formula (I) or an enantiomer, diastereoisomer, hydrate, solvate, tautomer, racemic mixture or pharmaceutically acceptable salt thereof, and the use of same as a med...  
WO/2013/178064A1
Disclosed are a substituted pyranol derivative with sodium dependent glucose transporters (SGLTs) inhibitor compound 4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl, a preparation method thereof, and a pharmaceutical application thereof; and p...  
WO/2013/172239A1
The present invention is an acid diffusion control agent consisting of at least one compound selected from among the group consisting of a compound represented by formula (1) and a compound represented by formula (2). In formula (1), R2 ...  
WO/2013/152359A1
Provided herein, inter alia, are compositions and methods of synthesis and detection of tetrazines and diazonorcaradienes.  
WO/2013/133419A1
[Problem] To provide a novel gelling agent that includes a sugar derivative. [Solution] A gelling agent comprising a compound represented by formula (1) or (2) (wherein R1 and R3 each independently represent a C1-20 straight-chain or bra...  
WO/2013/123896A1
Provided is a method for preparing 3-O-benzyl-1,2-O-isopropylidene-α-L-furan idose, which comprises: (1) protecting hydroxyl of 3-O-benzyl-1,2-O-isopropylidene-α-D-glucofuranose (III) by benzoyl and methylsulfonyl to obtain 6-O-benzoyl...  
WO/2013/097042A1
Disclosed is a compound of formula 1, as shown below, where R1, R2, R3, R4, R5, R6 and R7 are as described herein. Also, disclosed is a process for the preparation of compounds of formula 1, and intermediates used therein. The compound o...  
WO/2013/046180A1
A method that can be used to make a precursor of L-fiicose from D-glucose, that comprises the steps of: a) making a compound of formula (1) from D-glucose, formula (1) wherein R1 is acyloxy, and Q is a group (a), (b), (c) or (d), Formula...  
WO/2013/004626A1
The present invention is concerned with a process for preparing acetals and ketals which comprises (i) reacting an aldehyde or ketone with an alcohol in the presence of a solid acid at a temperature of below -40 °C, and (ii) removing wa...  
WO/2013/000086A1
The invention provides compounds for selectively inhibiting glycosidases, prodrugs of the compounds, and pharmaceutical compositions including the compounds or prodrugs of the compounds. The invention also provides methods of treating di...  
WO/2013/000084A1
The invention provides compounds with enhanced permeability for selectively inhibiting glycosidases, prodrugs of the compounds, and pharmaceutical compositions including the compounds or prodrugs of the compounds. The invention also prov...  
WO/2012/129651A1
The invention provides compounds of formula (I) with substituents as specified in claim 1 for selectively inhibiting glycosidases, prodrugs of the compounds, and pharmaceuticals compositions including the compounds or prodrugs of the com...  
WO/2012/126091A1
The invention provides compounds for selectively inhibiting glycosidases, prodrugs of the compounds, and pharmaceutical compositions including the compounds or prodrugs of the compounds. The invention also provides methods of treating di...  
WO/2012/083435A1
The invention provides compounds with enhanced permeability for selectively inhibiting glycosidases, prodrugs of the compounds, and pharmaceutical compositions including the compounds or prodrugs of the compounds. The invention also prov...  
WO/2012/061927A1
The invention provides compounds for selectively inhibiting glycosidases, prodrugs of the compounds, and pharmaceutical compositions including the compounds or prodrugs of the compounds. The invention also provides methods of treating di...  
WO/2012/008228A1
Disclosed is a method for oxidizing alcohols, wherein it is possible to efficiently oxidize primary alcohols and secondary alcohols and to achieve high reaction efficiency even when air is used as the bulk oxidant. Specifically disclosed...  
WO/2011/098460A1
The invention relates to a method for generating three-dimensional self-supporting and/or substrate-supported molded bodies or structures on surfaces by solidifying a liquid to paste-like organic or organically modified material in selec...  
WO/2011/096934A1
A process for the preparation of topiramate in an one pot reaction comprises the following steps: A) reacting 2,3:4, 5 -bis -O- { 1-methylethylidene) -β-D-f ructopyranose with sulfurylchloride in xylene in the presence of an organic or ...  
WO/2011/021398A1
Provided are pyranose derivatives and furanose derivatives, depicted in formulas (I) through (V), of glucose, mannose, psicose, sorbose, tagatose, allose, altrose, gulose, idose, or talose. (In the formulas, M1 represents a specific poly...  
WO/2010/150789A1
Disclosed is a novel production method for efficiently and easily synthesizing an NC-type nucleoside at a high yield without requiring a step for converting an unnecessary protecting group. Specifically disclosed are a step for inverting...  
WO2010110382A1
Disclosed is a novel compound contained in blue rose. This novel compound, which is contained in blue rose, has a chemical structure represented by general formula (I) [wherein R1 is a group as set forth in claim 1; and R2 represents -OH...  
WO/2010/103857A1
Disclosed are a novel method for the synthesis of a glycopeptide by which glycopeptides of various types can be deprotected and excised from a resin, each under weakly acidic to weakly basic conditions, without causing the problems of th...  
WO/2009/102022A1
Provided is a 3,6-O-bridged pyranose inversion compound useful as a β-O-glycosylating agent for use in selectively and easily producing β-O-pyranoside. The 3,6-O-bridged pyranose inversion compound is represented by general formula (1)...  
WO/2009/014970A1
Methods of synthesizing sodium glucose co-transporter 2 inhibitors, as well as compounds useful therein, are disclosed. Particular inhibitors are compounds of formula (I).  
WO/2008/152386A1
The invention relates to a process for preparing furanose derivatives, to furanose intermediates used in said process and to the use of said derivatives in the manufacture of atorvastatin.  
WO/2008/148549A3
The invention relates to a process for the catalytic conversion of a carbohydrate, an alcohol, an aldehyde or a polyhydroxy compound in the presence of a catalyst containing gold in a solvent.  
WO/2008/148549A2
The invention relates to a process for the catalytic conversion of a carbohydrate, an alcohol, an aldehyde or a polyhydroxy compound in the presence of a catalyst containing gold in a solvent.  

Matches 1 - 50 out of 816