Login| Sign Up| Help| Contact|

Patent Searching and Data


Matches 301 - 350 out of 1,379

Document Document Title
WO1990012577A3  
WO/1992/004047A1
Methods for diagnosing pre-hypertension, hypertension, congestive cardiomyopathy, renal failure, salt-sensitivity and adenomas and endocrine cell hyperplasias are disclosed. Also disclosed are methods for monitoring hypertension therapy,...  
WO/1992/004365A1
The invention relates to the novel compound mometasone furoate monohydrate, process for its preparation and pharmaceutical compositions containing said compound.  
WO/1992/003465A1
Disclosed are 20-methyl-5,7-pregnadiene-3$g(b),21-diol derivatives of general formula (I), in which R¿1? is a hydrogen atom or a lower-alkyl group and R¿2? is a lower-alkyl group, or R¿1? and R¿2? together represent a tetramethylene ...  
WO/1992/000316A1
A novel bile alcohol of general formula (I), having an efficacious physiological activity and being specified in the configurations of particularly the 20-, 24- and 25-positions; formula (I) wherein one of the groups R1 and R2 represents...  
WO1991017176A3  
WO/1991/017176A2
The present invention discloses compounds useful for the screening or monitoring of hypertensive individuals, for correction of interference in the measurement of digoxin levels in patients, and as pressor agents, potassium sparing diure...  
WO/1991/014689A1
A process for synthesizing polyoxa heterocycle compounds and in particular the antimalarial agent known as quinghaosu or artemisinin and its analogs is disclosed. A family of new antimalerial analogs of quinghaosu is also disclosed.  
WO/1991/011452A1
For a production of glycosides, especially of steroidal glycosides, molecular iodine is used as a reaction catalyst, wherein an alcohol and/or phenol, especially a hydroxy-steroid, is glycosylated, such that the glycosylation is performe...  
WO/1991/010743A1
The invention is directed to the control of cellular autophagy, cellular agglutination and the immobilization of motile cells. Such control is useful in, for example, the treatment of cancer, contraception, termination of pregnancy, remo...  
WO/1991/002739A1
Methods of stereoselectively preparing a substituted 1,2-anhydrosugar wherein a substituted glycal is converted into a 1,2-anhydrosugar that is utilized to glycosylate a hydroxyl group containing glycal, are disclosed. Methods of prepari...  
WO/1991/000733A1
A method of treatment of androgen-related diseases such as prostate cancer in susceptible male animals, including humans, comprises administering novel antiandrogens and/or novel sex steroid biosynthesis inhibitors as part of a combinati...  
WO/1991/000732A1
Methods for treating sex steroid-dependent diseases by inhibiting sex steroid activity include administration of novel compounds which include an androgenic nucleus substituted at a ring carbon with at least one substituent specified her...  
WO/1990/012577A2
A method of inhibiting hair growth in mammals which comprises the topical administration of a composition comprising an anti-angiogenic effective amount of an angiostatic compound of formula (I). The formula (I) compound is present in an...  
WO1990009394A3  
WO/1990/009394A2
The process of the present invention is a process for the preparation of an 11-oxygenated steroid of formula (II) which comprises (1) contacting a 9alpha-halo steroid of formula (I) with a metal selected from the group consisting of tin ...  
WO/1990/009164A1
A composition for topical application in order to induce and promote hair growth and to reduce hair loss contains, in a physiologically acceptable alcohol-based solvent medium, at least 7-alpha-(acetylthio) 4', 5'-dihydrospiro[androst 4-...  
WO/1990/008315A1
Ginsenosides Rb1 and Rg1 enhance the availability of acetylcholine in the cortical and hippocampal regions of the brain and alleviate the symptoms of Alzheimer-type senile demential. The Rb1 or Rg1 may be administered together with a met...  
WO/1990/003184A1
The invention claims an iscom matrix which is not a lipid vesicle comprising at least one lipid and at least one saponim but no intentional antigenic determinants and optionally also adjuvants for use as an immunomodulating agent, medici...  
WO/1990/003385A1
New 11beta-phenyl-14betaH-steroids of general formula (I), where Z is an oxygen atom or the hydroxyimino-grouping N ~ OH, and M and N are either jointly a second compound or L is a hydrogen atom and M is an alpha-permanent hydroxy group ...  
WO/1990/000174A1
The invention concerns 13-Alkyl-11beta-phenylgonanes of general formula (I), wherein Z, R1, R2, R3 and R4 have the meaning given, a process for their preparation, pharmaceutical preparations containing these compounds, and their use for ...  
WO/1989/003839A1
The invention relates to the field of chemistry and more particularly to the field of therapeutic chemistry. Its specific subject matter concerns compounds of general formula (I), in which R is a hydrogen atom, a lower alkyl, methoxymeth...  
WO/1988/009336A1
Substantially pure saponins are disclosed. The saponins of the present invention are useful as immune adjuvants. Disclosed as well are immune response-provoking compositions comprising an antigen in admixture with the substantially pure ...  
WO/1988/007545A1
Pregnane derivatives represented by general formula (I) (wherein A1 represents a hydrogen atom or a hydroxy group, A2 represents a substituent such as a hydroxy group when A1 represents a hydrogen atom, or A2 represents a hydrogen atom w...  
WO/1988/007050A1
Process for the production of (+)-bicyclo-[3.3.0]octane-3-on-2-carboxylic acid steroid esters having the formula (I), in which X represents oxygen or the -O-(CH2)n-O- or the -O-CH2-C(CH3)2-CH2-O- residue; n represents 2 or 3; R2 represen...  
WO/1988/002252A1
A unique set of compositions of matter characterized by including defined active agents covalently bonded to carbonium ion base groups, as well as the method of creating the compositions. The covalently bonded compositions include base g...  
WO/1987/006706A1
Qualitative and quantitive electrochemiluminescent assays for analytes of interest present in multicomponent liquids. These methods comprise contacting a sample with a reagent labeled with an electrochemiluminescent chemical moiety and c...  
WO/1987/005028A1
Compounds of formula (I), wherein one X is COOR, CH2COOR, CH(COOR)2, CONHR, CH2CONHR, or CN; remaining X's are H, F, CH3, OH, COOR, CH2COOR, CH(COOR)2, CONHR, CH2CONHR, or CN; Y is (i1), (i2), (i3), (i4), or (i5); R is H, alkyl of 1-5 ca...  
WO/1987/002672A1
Novel tetrahydro steroids which are useful in inhibiting angiogenesis and have the following structure: A compound of formula (I), wherein R15 is = O or -OH; wherein R23 with R10 forms a cyclic phosphate of formula (II) or wherein R23 is...  
WO/1986/002078A1
New 24-homo-vitamin D compounds, methods for preparing the same and novel intermediate compounds. The compounds are characterized by vitamin D-like activity of the order of 1alpha,25-dihydroxyvitamin D3, the recognized circulating hormon...  
WO/1986/001208A1
Stereoisometrically pure DELTA2 compound of formula (I) wherein R1 is hydrogen or -(C=O)-R2, wherein R2 is an organic substituent selected from the group consisting of alkyls, alkenyls, alkynyls, cycloalkyls, cycloalkylalkylenes, haloalk...  
WO/1985/000818A1
New derivative of vitamin D, 23,23-difluoro-25-hydroxycholecalciferol, a method for preparing said compound and various new intermediates utilized in such process. The compound is characterized by vitamin D-like activity as evidenced by ...  
WO/1985/000819A1
New derivative of vitamin D, 23,23-difluoro-1,25-dihydroxycholecalciferol. The compound is characterized by vitamin D-like activityas evidenced by its ability to increase intestinal calcium transport. It is further characterized by its r...  
WO/1984/004041A1
A colon-specific drug delivery system based on the use of a synthetic drug glycoside prodrug composition which, when ingested by a mammal, undergoes reaction with glycosidases produced by colonic microflora to release a free drug capable...  
WO/1984/001155A1
Hydroxylated derivatives of vitamin D2., processes for preparing such compounds, intermediates utilized in such processes and certain isotopically labelled vitamin D2 compounds. The vitamin D2 derivatives would find application in the tr...  
WO/1983/003604A1
Process for preparing substitued polycyclo-alkylidene polycyclo-alkanes, such as substituted adamantylidene adamantanes, and the corresponding epidioxy compounds, in which polycyclo-alkylidene polycyclo-alkanes are halogenated with an N-...  
WO/1983/003099A1
The invention relates to products having the general formula I, wherein R1 is thienyl or phenyl optionally substituted, furyl, cycloalkyl, naphtyl, phenyl-phenyl, alkyl or alkenyl; R2 is methyl or ethyl; R3 is H, OH, alkyl, alkenyl, opti...  
WO/1982/003396A1
Novel cundurango glycoside compounds represented by the following general formula: (FORMULA) process for their preparation from an extract of Marsdenia cundurango Reichenbach fil., use of the compound or composition containing it as an a...  
WO/1982/000465A1
Methods for preparing the various isomeric forms of 25-hydroxyvitamin D3-26, 23-lactone utilizing cyanohydrin formation with readily prepared steroid materials followed by actinic radiation of the products and recovery of the desired 25-...  
WO/1981/002577A1
Novel cundurango glycosides represented by the following general formula (1), a process for preparing them from an extract of Marsdenia cundurango Reichenbach fil. of potato family, and the use of a compound or composition containing the...  
WO/1981/002298A1
New derivative of vitamin D, 25-hydroxy-26,26,26,27,27,27-hexafluoro cholecalciferol and process for preparing the same. The compound is characterized by vitamin D-like activity in their ability to increase intestinal calcium transport, ...  
WO/1980/002502A1
New vitamin D derivatives as well as new intermediate compounds derived during the processes for preparing such new derivatives. The new derivatives have been identified as 1(Alpha)-hydroxy-25-keto-27-nor-vitamin D3 and its acylates. 1(A...  
JP2019529550A
The Panax diol type Ginsenoside derivative which has the structure shown in formula I or formula II is provided. Those use in manufacture of the medicine for preventing and treating atheroma Disease is also provided. The above-mentioned ...  
JP2019520416A
Neuroactive steroid or its salt which can be received pharmacologically is indicated in this specification. It is assumed that such a compound acts as a GABA regulation factor in a specific embodiment. The directions for use and the trea...  
JPWO2018016483A1
A Mogrol glycoside and the new manufacturing method of Mogrol were called for. The present invention provides a Mogrol glycoside including the process of cutting at least one glucosidic linkage of a Mogrol glycoside, and/or the manufactu...  
JP2019516720A
The present invention is a compound of general formula (I) : [Formula 1](Inside of a formula: R)1R2R3R4R5R6And Y is as being defined as this specification, and is related for being. The compound is an intermediate in composition of usefu...  
JP2019068741A
To provide algae that produce sterol, and a method for producing sterol using the same.Algae such as AJ7867 strain (FERM P-22304) and a strain derived therefrom, having a sterol production ability, are cultured. From bodies of the result...  
JP2019510051A
Formula (I) :They are [in / the compound boiled and twisted, its salt which can be received pharmacologically, and its pharmacological constituent are provided, and /; type (I) ] A and R.1And R5It is as defining in Is and this specificat...  
JP2019500374A
Generally the present invention relates to a constituent and a method for dealing with cancer and col over Tizons disease . A medicine constituent containing a replaced steroid derivative compound and the above-mentioned compound is prov...  
JP2018519328A
Formula (I)It is alike, the compound of a statement, its salt which can be received pharmacologically, and its pharmacological constituent are provided, and they are inside of; type, and R.1R2And R5It is as defining in Is and this specif...  

Matches 301 - 350 out of 1,379