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Matches 251 - 300 out of 915

Document Document Title
JP2011507925A
The invention relates to 17-(1′-propenyl)-17-3′-oxidoestra-4-en-3-one derivatives with the general chemical formula I, where the residues Z, R4, R6a, R6b, R7, R15, R16a, R16b and R18 have the meanings stated in Claim 1, and their sol...  
JP4629030B2  
JP4589869B2  
JP2010531337A
The present invention leaves 17* ketosteroid denoted by formula (III), and is R.3R5R6R7R10R13R15R16R40R41And R42A basis is related with the manufacturing method of the 17alpha* (3* hydroxypropyl) *17beta* hydroxy steroid denoted by formu...  
JP4545929B2  
JP4545868B2  
JP2010530404A
The new neuro-steroid derivative which the present invention acts on a nervous system and has the anti-apoptosis characteristic, the nerve protection characteristic, and the neurogenic characteristic, It is [the method of producing it, a...  
JP4536373B2  
JP2010527380A
The present invention relates to antiandrogenic compounds which may be administered for the treatment of androgen excess in the skin and by way of consequence, the treatment of acne, baldness or hirsuitism in subject or patient. These co...  
JP2010520178A
The mineralcorticoid receptor antagonist comprises spironolactone, eplerenone and drospirenone. Glucocorticoid, progesterone receptor antagonist and estrogen receptor antagonist are also included. The estrogen is ethinylestradiol. - ACTI...  
JP4476480B2  
JP2010120972A
To solve a problem that the necessity of an anti-progestin compound exhibiting higher specificity is left.An cyclic amine-substituted compound such as N-piperidinyl, especially useful when the 4-position of a 11-aryl portion is substitut...  
JP4450435B2  
JP2010031034A
To provide a method of treatment, sapogenin, related compounds and their derivatives.There is disclosed a method of treatment of non-cognitive neurodegeneration, non-cognitive neuromuscular degeneration, motor-sensory neurodegeneration, ...  
JP4414231B2  
JP2009539934A
A novel process for preparing a compound of formula (I) which comprises converting a compound of formula (II) to a compound of formula (I) via a compound of formula (III), or a salt thereof, without isolating any intermediates.  
JP2009539964A
Anti-pro ゲストーゲン with the strong present inventionAnd it is related with the new industrial process for composition without the solvent sum of 17of formula (I) which is anti-glucocorticoid agent alpha* acetoxy *11beta* [4* (N ...  
JP4368945B2  
JP2009537470A
The present invention relates to the use of ドロスピレノン for manufacture of the medicine for preventing advance of the high blood pressure (>=140/90mmHg) in the subject in a hypertensive advance tendency. A subject who needs pre...  
JP4331478B2  
JP2009167188A
To provide a new compound having a specific strong progesterone-like property and devoid of residual androgenic activity.The compound is expressed by formula (I), wherein R1, R2, R3, R4, R5 and R6 are each a hydrogen atom or a specific s...  
JP2009527490A
[Formula 1]The present invention is turned to using the pharmaceutical constituent and them which made new 17* phosphorus steroid derivative and them contain under the obstacle and the sick medical treatment which progesterone or a gluco...  
JP4263478B2  
JPWO2007063930A1
式:【化1】で表される化合物を紫外線照射 により開環し、次いで異性化することを特徴 とする、[{(5Z,7E)−(1S,3R, 0S)−1,3−ジヒドロキシ−9,1...  
JP4260886B2  
JP2009513626A
The medicine constituent and food constituent which contain the extract of the useful department (Dioscoreaceae) plant of yam and the extract in prevention or medical treatment of peripheral neuropathy are provided. The prevention or med...  
JP4215603B2  
JP2009501753A
This invention relates to processes for the production of 3-oxo-pregnane-21,17-carbolactones of formula II as well as 3-oxo-pregn-4-ene-21,17-carbolactones of formula III by the metal-free oxidation of 17-(3-hydroxypropyl)-3,17-dihydroxy...  
JP2004511435A5  
JP4146897B2  
JP4145350B2  
JP2008526709A
The present invention is a general formula. It is related with new 18-methyl 19-ノル- 17-pre グン- 4-エン- 21 of (I), and 17-カルボ lactone. : Inside of a formula, Z is an oxygen atom, two hydrogen atoms, =NOR, or =NNHSOR basis,...  
JP2008522962A
It is synthetic steroid which has progesterone activity, anti-electrolyte corticoid activity, and antiandrogenic activity, and indicates about the manufacture methods of ドロスピレノン useful to the manufacture of a medicine compo...  
JP2008521876A
The present invention relates to the important intermediate for the production method of 17*ヒドロキシ*6beta (formula (I)), 7beta;15beta, and 16beta* screw methylene *17alpha* プレグネ *4* エン *3* ON *21* carboxylic acid gamm...  
JPWO2006062129A1
本発明は、式(I)で示される(5α,7α −3−スピロ−2’−(1’,3’−ジオ ソラン)−24−オキソコレスト−22− ン−7−イル ベンゾアート(不飽和ケ...  
JP4097697B2  
JP2003531148A5  
JP2008100996A
To synthesize epoxymexrenone and an epoxymexrenone-based compound.Multiple novel reaction schemes, novel process steps and novel intermediates are provided for the synthesis of epoxymexrenone compounds of the formula I, wherein: -A-A- re...  
JP2007528389A5  
JP2003531119A5  
JP2008512439A
The method for changing the steroid substrate which has 4 and 7* carbonyl bridge into the structure containing a 7alpha* Alcokey deer ルボニル substituent is preferably indicated by by making a substrate and the source of an alkoxy g...  
JP4039683B2  
JP2007016043A5  
JP4012293B2  
JP2007530557A
The method related with an epoxidation reaction is indicated. Especially the method concerned includes the conversion to the structure by the reaction of the substrate under existence of a peroxide active agent, and a pel オキシド co...  
JP2007528388A
The present invention relates with a molecular dispersion form to steroid medicine, for example, the medicine composite containing ドロスピレノン. A composite is offered as a solid, a semisolid, or a liquid form, and these are app...  
JP2007528389A
The present invention relates to the medicine composite which has the solubility which the oleophilic medicine to the inside of a water medium has improved. The medicine composite containing the powder of oleophilic compounds, such as an...  
JP3984315B2  
JP3983796B2  
JP3977462B2  

Matches 251 - 300 out of 915