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Title:
【発明の名称】強力なバニロイド受容体アゴニストおよび鎮痛剤としてのレジニフェラトキシンファーマコフォアを含むバニロイド同類体、その組成物およびその用途
Document Type and Number:
Japanese Patent JP2002537373
Kind Code:
A
Abstract:
The present invention is related to new vanilloid analogues containing resiniferatoxin pharmacophores, pharmaceutical compositions comprising such analogues, and their uses as vanilloid receptor agonists and potent analgesics. The present invention provides a pharmaceutical composition for treating acute, chronic, inflammatory or neuropathic pains or for treating bladder hypersensitivity.

Inventors:
Lee, Zee Woo
Oh, Ootaek
Park, Yoon-ho
Sue, Youn-Gel
Park, Hyeun-Gaeun
Kim, hee-do
Application Number:
JP2000600971A
Publication Date:
November 05, 2002
Filing Date:
February 21, 2000
Export Citation:
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Assignee:
Pacific Corporation
Digital Biotech Company Limited
International Classes:
C07C235/34; C07C335/12; (IPC1-7): C07C335/12; A61K31/222; A61P13/02; A61P13/10; A61P25/04; A61P29/00; A61P43/00; C07C235/34
Attorney, Agent or Firm:
Takehiko Suzue (4 outside)