非ペプチドGnRH剤、医薬組成物、およびそれらの使用方法

Japanese Patent JP2005538064

A

Non-peptide GnRH agents capable of inhibiting the effect of gonadotropin-releasing hormone are described. Such compounds and their pharmaceutically acceptable salts, prodrugs, and active metabolites are suitable for treating mammalian reproductive disorders and steroid hormone-dependent tumors as well as for regulating fertility, where suppression of gonadotropin release is indicated. Methods for synthesizing the compounds and intermediates useful in their preparation are also described.

JP2002511387	INDUSTRIAL APPLICABILITY [title] Substituent semicarbazide and its use
WO/2005/030702	BIPHENYLOXY-ACIDS
JPH075530	[Title of the Invention] Carboxyalkylcarbonyl Amino Acid Endopeptidase Inhibitor

Mark Brian Anderson
Lance Christopher Christie
Quen Quen Sai Do
Jun Feng
Yufeng Hong
High Taori
Ved Prakash Pasak
Ranjan Jagas Rajapakse
Eric Tuck On Sun
Aileen Valenzuela Thompkins

JP2004513278A

December 15, 2005

June 04, 2003

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Pfizer Inc.

C07D307/68; A61K31/341; A61K31/435; A61K31/4353; A61K31/437; A61K31/443; A61K31/4709; A61K31/495; A61K31/501; A61K31/506; A61K31/519; A61K31/53; A61P5/02; A61P5/04; A61P13/08; A61P15/00; A61P15/08; A61P15/16; A61P25/20; A61P31/00; A61P31/18; A61P35/00; A61P37/02; A61P43/00; C07D307/46; C07D405/12; C07D405/14; C07D471/04; C07D495/04; C07D519/00; (IPC1-7): C07D307/68; A61K31/341; A61K31/437; A61K31/443; A61K31/4709; A61K31/501; A61K31/506; A61K31/519; A61K31/53; A61P5/02; A61P5/04; A61P13/08; A61P15/00; A61P15/08; A61P15/16; A61P25/20; A61P31/00; A61P31/18; A61P35/00; A61P37/02; A61P43/00; C07D405/12; C07D405/14; C07D471/04; C07D495/04; C07D519/00

WO2000020358A2	2000-04-13
WO2000069810A1	2000-11-23

Yoshinobu Murofushi

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