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Title:
バルデナフィルを含有する制御放出製剤
Document Type and Number:
Japanese Patent JP2007537175
Kind Code:
A
Abstract:
Controlled release dosage form comprising vardenafil gives an average release rate between 80% in 2 hours and 80% in 24 hours. ACTIVITY : Vasotropic; Hypotensive; Antianginal; Antiarrhythmic; Cerebroprotective; Antiinflammatory; Antiasthmatic; Cardiant; Uropathic; Cytostatic; Nootropic; Neuroprotective; Antiparkinsonian; Anticonvulsant; Neuroleptic; Antipsoriatic; Analgesic; Nephrotropic; Ophthalmological; Antidiabetic; Hepatotropic; Osteopathic; Antiallergic; Antiarteriosclerotic; Antidepressant; Immunosuppressive; Immunomodulator; Antiulcer; Antilipemic; Antimigraine. MECHANISM OF ACTION : Phosphodiesterase type 5 inhibitor.

Inventors:
Zuzanne Treger
Peter Zerno
Helmut Hanning
Kerstin Pauli
Laurent Heinich
Application Number:
JP2007511975A
Publication Date:
December 20, 2007
Filing Date:
April 29, 2005
Export Citation:
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Assignee:
Bayer HealthCare AG
International Classes:
A61K31/53; A61K9/20; A61K9/24; A61K9/28; A61K31/522; A61K47/12; A61K47/30; A61K47/32; A61K47/34; A61K47/36; A61K47/38; A61P15/10
Domestic Patent References:
JP2002528408A2002-09-03
Foreign References:
WO2002060422A22002-08-08
Other References:
JPN5007007720; ROSEN RC.: 'PDE-5 Inhibition and Sexual Response: Pharmacological Mechanisms and Clinical Outcomes' ANNUAL REVIEW OF SEX RESEARCH Vol.13, 2002, p36-88, SOCIETY FOR THE SCIENTIFIC STUDY OF SEX
Attorney, Agent or Firm:
Mitsuo Tanaka
Takuji Yamada
Mitsutaka Iwasaki
Aoyama Aoi
Yasuo Shibata



 
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