トロンビンレセプターアンタゴニストとしての条件付きヒンバシンアナログ

Japanese Patent JP2008500360

A

A compound represented by the structural formula and pharmaceutically acceptable salts and solvents thereof is disclosed, wherein: the single-dashed line between the ring carbons to which R¹⁰ and R³⁴ are attached represents either a single bond or a double bond; the double-dashed line between X and the carbon to which Y is attached represents either a single bond or an absent bond; X is -O- or -NR⁶- when the double-dashed line represents a single bond; X is H, -OH or -NHR²⁰ when the double-dashed line represents an absent bond; and other parameters are as defined herein. Also disclosed are pharmaceutical compositions and combinations containing said compounds and their uses as thrombin receptor antagonists and binders to cannabinoid receptors.

JPS5675407	HERBICIDE
JP2006513165	Mucin synthesis inhibitor
WO/2004/067529	INDOLE-DERIVATIVE MODULATORS OF STEROID HORMONE NUCLEAR RECEPTORS

Shellier, Maria Pan Buoy.
Chacala Manil, Samuel
Xia, Yang
Clasby, Martin Sea.
Greenlee, William Jay.
One, Yukowan
Bertri, Enricopy.
Wu, Wen Shwe
Graziano, Michael Pea.
Koso glow, teddy
Chintara, Madu

JP2007515301A

January 10, 2008

May 25, 2005

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Schering Corporation

C07D405/06; A61K31/443; A61K31/4433; A61P1/00; A61P1/16; A61P3/10; A61P7/00; A61P7/02; A61P9/00; A61P9/04; A61P9/06; A61P9/08; A61P9/10; A61P9/12; A61P11/00; A61P11/06; A61P11/08; A61P11/16; A61P13/12; A61P15/10; A61P17/00; A61P17/02; A61P17/06; A61P19/02; A61P19/08; A61P25/00; A61P25/06; A61P25/14; A61P25/16; A61P25/28; A61P27/02; A61P27/06; A61P29/00; A61P35/00; A61P43/00; C07D405/08; C07D493/04

JP2004503551A	2004-02-05
JP2003128670A	2003-05-08
JP2004503551A	2004-02-05
JP2003128670A	2003-05-08

Hidesaku Yamamoto
Takaaki Yasumura
Natsuki Morishita

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