Title:
血漿中のグルコースレベル、コレステロールレベル及びトリグリセリドレベルを低下させるための5-[4-(4-(2-アミノ-2-メトキシカルボニルエチル)フェノキシ)ベンジリデン]チアゾリジン-2,4-ジオン誘導体及び関連化合物
Document Type and Number:
Japanese Patent JP2008530242
Kind Code:
A
Abstract:
Novel diphenyl ether derivatives are provided that exhibit activity useful for reducing glucose, cholesterol, and/or triglyceride levels in plasma, and for treatment of obesity, inflammation, immunological diseases, autoimmune diseases, diabetes and disorders associated with insulin resistance.
Inventors:
Nag Bishwajit
Nag Abhigit
Day Devendranate
Agarwal Shiv Kumar
Neogi Parta
Ruddy Gadam Homme
Buddyger sanga mesh
Singa Jendra
Pandy Slender Kumar
Chitra Santana Gopalan
Nag Abhigit
Day Devendranate
Agarwal Shiv Kumar
Neogi Parta
Ruddy Gadam Homme
Buddyger sanga mesh
Singa Jendra
Pandy Slender Kumar
Chitra Santana Gopalan
Application Number:
JP2007556366A
Publication Date:
August 07, 2008
Filing Date:
February 17, 2006
Export Citation:
Assignee:
Vexel Pharmaceuticals, Inc.
International Classes:
C07D277/20; A61K31/4164; A61K31/421; A61K31/426; A61P3/04; A61P3/06; A61P3/10; A61P25/00; A61P29/00; A61P37/02; A61P37/06; A61P43/00; C07D277/34; C07D277/36
Domestic Patent References:
JPH0228168A | 1990-01-30 | |||
JP2004504299A | 2004-02-12 | |||
JP2003508391A | 2003-03-04 | |||
JPH0228168A | 1990-01-30 |
Foreign References:
WO2004066964A2 | 2004-08-12 | |||
WO2003043998A1 | 2003-05-30 |
Attorney, Agent or Firm:
Sadao Kumakura
Nobuo Ogawa
Atsushi Hakoda
Kenji Asai
Koji Hirayama
Nobuo Ogawa
Atsushi Hakoda
Kenji Asai
Koji Hirayama