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Title:
血漿中のグルコースレベル、コレステロールレベル及びトリグリセリドレベルを低下させるための5-[4-(4-(2-アミノ-2-メトキシカルボニルエチル)フェノキシ)ベンジリデン]チアゾリジン-2,4-ジオン誘導体及び関連化合物
Document Type and Number:
Japanese Patent JP2008530242
Kind Code:
A
Abstract:
Novel diphenyl ether derivatives are provided that exhibit activity useful for reducing glucose, cholesterol, and/or triglyceride levels in plasma, and for treatment of obesity, inflammation, immunological diseases, autoimmune diseases, diabetes and disorders associated with insulin resistance.

Inventors:
Nag Bishwajit
Nag Abhigit
Day Devendranate
Agarwal Shiv Kumar
Neogi Parta
Ruddy Gadam Homme
Buddyger sanga mesh
Singa Jendra
Pandy Slender Kumar
Chitra Santana Gopalan
Application Number:
JP2007556366A
Publication Date:
August 07, 2008
Filing Date:
February 17, 2006
Export Citation:
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Assignee:
Vexel Pharmaceuticals, Inc.
International Classes:
C07D277/20; A61K31/4164; A61K31/421; A61K31/426; A61P3/04; A61P3/06; A61P3/10; A61P25/00; A61P29/00; A61P37/02; A61P37/06; A61P43/00; C07D277/34; C07D277/36
Domestic Patent References:
JPH0228168A1990-01-30
JP2004504299A2004-02-12
JP2003508391A2003-03-04
JPH0228168A1990-01-30
Foreign References:
WO2004066964A22004-08-12
WO2003043998A12003-05-30
Attorney, Agent or Firm:
Sadao Kumakura
Nobuo Ogawa
Atsushi Hakoda
Kenji Asai
Koji Hirayama