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Title:
向上したインドリノン系プロテインキナーゼ阻害剤
Document Type and Number:
Japanese Patent JP2008542294
Kind Code:
A
Abstract:
Alpha-hydroxy-omega-(2-oxo-indolylidenemethyl-pyrrole-3′-carbonyl)amino alkanoic acid and amide derivatives have enhanced and unexpected drug properties as inhibitors of protein kinases and are useful in treating disorders related to abnormal protein kinase activities such as cancer.

Inventors:
Liang, Consin
Fen, yanbo
Voykovsky, Tomas
Application Number:
JP2008513740A
Publication Date:
November 27, 2008
Filing Date:
May 26, 2006
Export Citation:
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Assignee:
The Script Research Institute
International Classes:
C07D403/06; A61K31/404; A61K31/5377; A61P29/00; A61P35/00; A61P43/00; C07D403/14
Attorney, Agent or Firm:
Shoichi Okuyama
Arihara Koichi
Matsushima Tetsuo
Hidefumi Kawamura
Naomi Yoshida
Ayako Nakamura
Masayuki Okamoto
Fukagawa Eri
Satoshi Morimoto