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Title:
置換キサンチン誘導体
Document Type and Number:
Japanese Patent JP2011513309
Kind Code:
A
Abstract:
A pharmaceutical composition comprising: a. an effective amount of a compound of Formula B: or a pharmaceutically acceptable salt thereof; b. a second therapeutic agent selected from insulin or insulin analogues, glucagon-like-peptide-1 (GLP-1) receptor agonists, sulfonylurea agents, biguanide agents, alpha-glucosidase inhibitors, PPAR agonists, meglitinide agents, dipeptidyl-peptidase (DPP) IV inhibitors, phosphodiesterase inhibitors, amylin agonists, CoEnzyme A inhibitors, and antiobesity agents; and c. a pharmaceutically acceptable car.

Inventors:
Toon Roger Dee.
Ryu Julie F.
Herbson Scott El.
Application Number:
JP2010548747A
Publication Date:
April 28, 2011
Filing Date:
February 27, 2009
Export Citation:
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Assignee:
Concert Pharmaceuticals Incorporated
International Classes:
C07D473/06; A61K31/522; A61P1/16; A61P3/10; A61P9/00; A61P13/12; A61P27/02
Domestic Patent References:
JPH0525048A1993-02-02
Foreign References:
WO1994022449A11994-10-13
WO1996005854A21996-02-29
Other References:
JPN6013053654; 最新創薬化学 上巻 , 1998, p.379
JPN5011007702; KUSHNER DJ: 'PHARMACOLOGICAL USES AND PERSPECTIVES OF HEAVY WATER AND DEUTERATED COMPOUNDS' CANADIAN JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY V77 N2, 19990201, P79-88
Attorney, Agent or Firm:
Hatsushi Shimizu
Masao Haruna
Hirotaka Yamaguchi
Toshi Gobe
Ryuichi Inoue
Toshimitsu Sato
Koichi Niimi
Tomohiko Kobayashi
Shinichi Watanabe
Masato Ozeki
Yoshihiro Igarashi
Kazuya Kawamoto