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Title:
ホスホジエステラーゼ-4阻害剤としての第3アミン誘導体
Document Type and Number:
Japanese Patent JP2011517687
Kind Code:
A
Abstract:
The invention relates to inhibitors of the phosphodiesterase 4 (PDE4) enzyme. More particularly, the invention relates to compounds that are tertiary amines, methods of preparing such compounds, compositions containing them and therapeutic use thereof.

Inventors:
Rizzi, Andrea
Armani, Elisabetta
Pellets, illaria
La Porta, Elena
Application Number:
JP2011504342A
Publication Date:
June 16, 2011
Filing Date:
March 27, 2009
Export Citation:
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Assignee:
Siecie Pharmaceuti Societa Peratini
International Classes:
C07D213/61; A61K31/4409; A61K31/4436; A61P9/10; A61P25/00; A61P25/14; A61P25/16; A61P25/18; A61P25/24; A61P25/28; A61P43/00; C07D405/12; C07D409/12
Domestic Patent References:
JP2007513957A2007-05-31
JP2008543781A2008-12-04
JP2006508987A2006-03-16
JP2006516727A2006-07-06
JP2010500329A2010-01-07
Attorney, Agent or Firm:
Akio Miyazaki
Ishibashi Masayuki
Masaaki Ogata