Title:
ピリドキシンに由来するHIVインテグラーゼ阻害剤
Document Type and Number:
Japanese Patent JP2011521979
Kind Code:
A
Abstract:
The present invention relates to pyridoxine (vitamin B6) derived compounds of formula (I), pharmaceutically acceptable salts, or solvates thereof, wherein R1, R2, R4, A, L B1 and B2 are as defined in the specification, and pharmaceutical compositions comprising the compounds. Compounds of formula (I) inhibit Human Immunodeficiency Virus (HIV)-integrase enzyme and are useful for preventing and treating HIV infection and AIDS.
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Inventors:
Stranix Brent
Beaulieu Francis
Bouchard Jean-Emanuel
Mirogai
Chigan One
Ruel Les Jeans
Beaulieu Francis
Bouchard Jean-Emanuel
Mirogai
Chigan One
Ruel Les Jeans
Application Number:
JP2011511948A
Publication Date:
July 28, 2011
Filing Date:
June 04, 2009
Export Citation:
Assignee:
Ambria by Offermine Inc.
International Classes:
C07D213/81; A61K31/436; A61K31/44; A61K31/443; A61P31/18; A61P43/00; C07D213/82; C07D405/12; C07D491/056
Foreign References:
| WO2005103003A2 | 2005-11-03 | |||
| WO2004039803A2 | 2004-05-13 | |||
| EP1867636A1 | 2007-12-19 |
Attorney, Agent or Firm:
Hatsushi Shimizu
Masao Haruna
Hirotaka Yamaguchi
Toshi Gobe
Ryuichi Inoue
Toshimitsu Sato
Koichi Niimi
Tomohiko Kobayashi
Shinichi Watanabe
Masato Ozeki
Yoshihiro Igarashi
Kazuya Kawamoto
Masao Haruna
Hirotaka Yamaguchi
Toshi Gobe
Ryuichi Inoue
Toshimitsu Sato
Koichi Niimi
Tomohiko Kobayashi
Shinichi Watanabe
Masato Ozeki
Yoshihiro Igarashi
Kazuya Kawamoto