4-フェノキシ-ニコチンアミド又は4-フェノキシ-ピリミジン-5-カルボキサミド化合物

Japanese Patent JP2013517313

A

This invention relates to novel phenyl amide or pyridyl amide derivatives of the formula wherein A1, A2, B1, B2 and R1 to R11 are as defined in the description and in the claims, as well as pharmaceutically acceptable salts thereof. These compounds are GPBAR1 agonists and can be used as medicaments for the treatment of diseases such as type II diabetes.

Bisants, Katerina
Henrietta, Damelow
Ericson, Sean David
Kim, Kyung Jin
Martin, Rainer A
Opst Zander, Ulrike
Pietranico-Cole, Sherry Lynn
Richter, Hans
Ulmer, Christoph

JP2012549325A

May 16, 2013

January 18, 2011

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F. HOFFMANN-LA ROCHE AKTIENGESELLSCHAFT

C07D213/80; A61K31/44; A61K31/4709; A61K31/498; A61K31/506; A61P1/04; A61P1/14; A61P1/16; A61P3/00; A61P3/04; A61P3/06; A61P3/10; A61P9/00; A61P9/10; A61P9/12; A61P11/00; A61P11/06; A61P13/12; A61P17/06; A61P19/02; A61P25/00; A61P25/18; A61P25/24; A61P25/28; A61P27/02; A61P29/00; A61P37/08; C07D215/08; C07D215/40; C07D401/06; C07D401/14; C07D417/14

JP2004238361A	2004-08-26
JP2006528659A	2006-12-21
JP2012506887A	2012-03-22
JP2009543823A	2009-12-10
JP2006521344A	2006-09-21
JP2001522834A	2001-11-20
JPH07509695A	1995-10-26

WO2005009443A1	2005-02-03
WO1997024404A1	1997-07-10
WO2008125627A1	2008-10-23

Patent business corporation Tsukuni
Hajime Tsukuni
Yasuo Yanagibashi
Satoko Ito
Keiko Ozawa
Toshio Miyake
Yasuhiro Oguni
Yoko Tanaka
Atsushi Shiomi
Fusayuki Saito

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