Title:
新規な自己反応性アーム及び同物を含むプロドラッグ
Document Type and Number:
Japanese Patent JP2013532132
Kind Code:
A
Abstract:
The present invention relates to a compound of general formula (I): in which: X is OH, NH2, NHOH or RNH, where R may be a linear or branched, saturated or unsaturated, C1-C10 alkyl radical, Y is H, or an electron-withdrawing group, in particular selected from NO2, CF3 or a halogen, R1 and R2 are H or a linear or branched, saturated or unsaturated, C1-C10 alkyl radical, F is a reactive functional group that can be activated by click chemistry.
Inventors:
Papot, Sebastian
Thomas, Michael
Thomas, Michael
Application Number:
JP2013510716A
Publication Date:
August 15, 2013
Filing Date:
May 18, 2011
Export Citation:
Assignee:
Center National de la Recherche Scientific
UNIVERSITE DE POITIERS
UNIVERSITE DE POITIERS
International Classes:
C07C205/22; A61K31/704; A61K45/00; A61K47/48; A61P35/00; A61P35/02; A61P43/00; C07H15/252
Domestic Patent References:
| JP2008069175A | 2008-03-27 | |||
| JP2006523646A | 2006-10-19 | |||
| JPH10508291A | 1998-08-18 | |||
| JPH05117236A | 1993-05-14 |
Foreign References:
| US4379166A | 1983-04-05 |
Other References:
JPN6015021205; Ａｎｇｅｗａｎｄｔｅ Ｃｈｅｍｉｅ， Ｉｎｔｅｒｎａｔｉｏｎａｌ Ｅｄｉｔｉｏｎ ４２（３）, 2003, ｐ．３２７-３３２
Attorney, Agent or Firm:
Mitsuo Matsui