Title:
デングウイルス感染症の治療及び予防のためのチエノピリジン誘導体
Document Type and Number:
Japanese Patent JP2016501883
Kind Code:
A
Abstract:
特定のチエノピリジン誘導体化合物を治療有効量で投与することによる、ウイルス感染症を治療するための方法及び医薬組成物が開示される。該化合物及びその医薬組成物の使用方法も開示される。特に、フラビウイルス（すなわち、限定されないが、デングウイルス、西ナイル熱ウイルス、黄熱病ウイルス、日本脳炎ウイルス、及びダニ媒介脳炎ウイルスを含む）により引き起こされるようなウイルス感染症の治療が開示される。【選択図】なし
Inventors:
Dai, don chan
Bergson, James, Earl.
Chabana Gimat, Chantyakumar, Earl
Bird, Chelsea, M.
Harvey, Dennis, Yee.
Bergson, James, Earl.
Chabana Gimat, Chantyakumar, Earl
Bird, Chelsea, M.
Harvey, Dennis, Yee.
Application Number:
JP2015545858A
Publication Date:
January 21, 2016
Filing Date:
December 06, 2013
Export Citation:
Assignee:
Shiga Technologies, Inc.
International Classes:
C07D495/04; A61K31/4365; A61K31/4375; A61K31/444; A61K31/4545; A61K31/496; A61K31/497; A61K31/5377; A61K31/55; A61K38/21; A61K45/00; A61P31/14; A61P43/00; C07D495/14; C07D495/22
Domestic Patent References:
| JP2009537551A | 2009-10-29 | |||
| JP2008525434A | 2008-07-17 | |||
| JP2006298909A | 2006-11-02 | |||
| JP2001502683A | 2001-02-27 | |||
| JP2007526271A | 2007-09-13 |
Foreign References:
| WO2010099166A1 | 2010-09-02 | |||
| WO2011006158A2 | 2011-01-13 |
Other References:
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WAGNER, G. ET AL.: "Synthesis of 3-alkyl-2-aminopyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4-ones from 3-ethoxycarbonylamin", PHARMAZIE, vol. 48(2), JPN6017030131, 1993, pages 95 - 99, ISSN: 0003751844
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DATABASE REGISTRY [ONLINE] RETRIEVED FROM STN, vol. 掲載日：2009年8月30日以前, JPN7017002609, pages 2017 - 7, ISSN: 0003751846
DABAEVA, V. V. ET AL.: "Synthesis of new condensed derivatives of pyrano[4,3-b]thieno[3,2-e]pyridine and pyrido[3',2':4,5]th", CHEMISTRY OF HETEROCYCLIC COMPOUNDS, vol. 47(5), JPN6017030125, 2011, pages 639 - 643, ISSN: 0003751837
DATABASE REGISTRY [ONLINE] RETRIEVED FROM STN, vol. 掲載日：2011年12月4日以前, JPN7017002608, pages 2017 - 7, ISSN: 0003751838
MADKOUR, HASSAN MOHAMED FAWZY ET AL.: "Synthetic utility of enaminoester moiety in heterocyclic synthesis", EUROPEAN JOURNAL OF CHEMISTRY, vol. 1(4), JPN6017030127, 2010, pages 352 - 359, ISSN: 0003751839
Attorney, Agent or Firm:
Hiroshi Kobayashi
Kyoei Sugiyama
Norio Omori
Yasuhito Suzuki
Kyoei Sugiyama
Norio Omori
Yasuhito Suzuki