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Title:
ヒスタミンH4受容体のベンゾイミダゾール−2−イルピリミジンモジュレータ
Document Type and Number:
Japanese Patent JP2016510752
Kind Code:
A
Abstract:
ベンゾイミダゾール−2−イルピリミジン、その精製方法、並びにアレルギー、喘息、自己免疫性疾患、及びそう痒症を含む、H4受容体活性によって介在された疾病状態、疾患、及び医学的状態の処置のための医薬組成物及び方法。

Inventors:
Hicky, Magari, Bee.
Horns, stephan
Rochner, Suzanne
Conza, mateo
Application Number:
JP2015561646A
Publication Date:
April 11, 2016
Filing Date:
March 06, 2014
Export Citation:
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Assignee:
Janssen Pharmaceuticals N.B.
International Classes:
C07D401/14; A61K31/506; A61P1/00; A61P1/04; A61P1/16; A61P3/06; A61P3/10; A61P5/14; A61P5/16; A61P5/38; A61P7/00; A61P7/02; A61P9/00; A61P9/10; A61P11/00; A61P11/02; A61P11/06; A61P17/00; A61P17/04; A61P17/06; A61P19/00; A61P19/02; A61P21/00; A61P21/04; A61P25/00; A61P27/02; A61P29/00; A61P31/10; A61P31/22; A61P33/00; A61P33/14; A61P35/00; A61P37/02; A61P37/08; A61P43/00
Domestic Patent References:
JP2011526911A2011-10-20
JP2012528849A2012-11-15
JP2010504913A2010-02-18
JP2009532366A2009-09-10
JP2006528161A2006-12-14
JP2005511595A2005-04-28
JP2003531173A2003-10-21
Foreign References:
US6242460B12001-06-05
WO2012069442A12012-05-31
US20110184016A12011-07-28
Other References:
CAIRA M R, TOPICS IN CURRENT CHEMISTRY, vol. V198, JPN5006012237, 1998, DE, pages 163 - 208, ISSN: 0003867433
平山令明, 有機化合物結晶作製ハンドブック, JPN6014022315, 2008, pages 10 - 11, ISSN: 0003867434
Attorney, Agent or Firm:
Hiroshi Kobayashi
Norio Omori
Junko Kobayashi
Takayuki Imazato
Yasuhito Suzuki