Title:
化合物
Document Type and Number:
Japanese Patent JP2017521456
Kind Code:
A
Abstract:
本発明は、Lp−PLA2活性を阻害する新規化合物、それらの製造方法、それらを含む組成物、および、Lp−PLA2の活性に関連する疾患、例えばアルツハイマー病の治療におけるそれらの使用に関する。
Inventors:
Zehon, Wan
Chang, Xiao Ming
One, Jean
Matthew, Robert, Sender
Eric, Stephen, Manas
Rafael, Antony, Libero
Joseph, E. Pero
Christopher, Ernst, Knyp
Baipur Kumar, Cantibai, Patel
Chang, Xiao Ming
One, Jean
Matthew, Robert, Sender
Eric, Stephen, Manas
Rafael, Antony, Libero
Joseph, E. Pero
Christopher, Ernst, Knyp
Baipur Kumar, Cantibai, Patel
Application Number:
JP2017503553A
Publication Date:
August 03, 2017
Filing Date:
July 21, 2015
Export Citation:
Assignee:
GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED
International Classes:
C07D471/14; A61K31/519; A61K31/527; A61K31/5365; A61K31/5383; A61K31/542; A61P9/10; A61P25/28; C07D471/20; C07D487/04; C07D487/14; C07D491/20; C07D498/14; C07D513/14
Domestic Patent References:
JP2017520613A | 2017-07-27 | |||
JP2013537203A | 2013-09-30 |
Foreign References:
WO2013013503A1 | 2013-01-31 | |||
WO2013014185A1 | 2013-01-31 |
Attorney, Agent or Firm:
Hiroyuki Nagai
Yukitaka Nakamura
Yasukazu Sato
Satoru Asakura
Hiroyuki Fujii
Hiroshi Sorimachi
Yukitaka Nakamura
Yasukazu Sato
Satoru Asakura
Hiroyuki Fujii
Hiroshi Sorimachi