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Patent Searching and Data


Title:
化合物
Document Type and Number:
Japanese Patent JP2017521456
Kind Code:
A
Abstract:
本発明は、Lp−PLA2活性を阻害する新規化合物、それらの製造方法、それらを含む組成物、および、Lp−PLA2の活性に関連する疾患、例えばアルツハイマー病の治療におけるそれらの使用に関する。

Inventors:
Zehon, Wan
Chang, Xiao Ming
One, Jean
Matthew, Robert, Sender
Eric, Stephen, Manas
Rafael, Antony, Libero
Joseph, E. Pero
Christopher, Ernst, Knyp
Baipur Kumar, Cantibai, Patel
Application Number:
JP2017503553A
Publication Date:
August 03, 2017
Filing Date:
July 21, 2015
Export Citation:
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Assignee:
GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED
International Classes:
C07D471/14; A61K31/519; A61K31/527; A61K31/5365; A61K31/5383; A61K31/542; A61P9/10; A61P25/28; C07D471/20; C07D487/04; C07D487/14; C07D491/20; C07D498/14; C07D513/14
Domestic Patent References:
JP2017520613A2017-07-27
JP2013537203A2013-09-30
Foreign References:
WO2013013503A12013-01-31
WO2013014185A12013-01-31
Attorney, Agent or Firm:
Hiroyuki Nagai
Yukitaka Nakamura
Yasukazu Sato
Satoru Asakura
Hiroyuki Fujii
Hiroshi Sorimachi