Title:
【発明の名称】置換キノリン類およびシンノリン類
Document Type and Number:
Japanese Patent JP2675119
Kind Code:
B2
Abstract:
Compounds of the formula (1): wherein: R<1> to R<4> are independently H, halo, (C1-C4) alkyl, branched (C3-C4) alkyl, halo (C1-C4) alkyl, (C1-C4) alkoxy, NO2, or NH2, at least two of R<1> to R<4> being H, or one of R<2> to R<4> is -NR<7>-Y-Ar or O-Y-Ar and the rest of R<1> to R<4> are H; W is N, or CR<5>; R<5> is H, CH3, Cl, O-Y-Ar, or -NR<7>-Y-Ar; R<6> is H, CH3, Cl or Br; A is -O-Alk or -X-Y-Ar; Alk is a C2-C18 saturated or unsaturated hydrocarbon chain, straight chain or branched, optionally substituted with halo, halo (C1-C4) alkoxy, (C3-C8) cycloalkyl, hydroxy, or acetyl; X is O, NR<7>, or CR<8>R<9>, provided that if one of R<2> to R<5> is NR<7>-Y-Ar or O-Y-Ar, then X-Y-Ar is an identical group; R<7> is H, (C1-C4) alkyl, or acetyl; R<8> and R<9> are independently H, (C1-C4) alkyl, (C1-C4) acyl, halo, or OH, or R<8> and R<9> combine to form a saturated or unsaturated carbocyclic ring comprising three to seven carbon atoms; Y is an alkylene chain 2 to 8 carbon atoms long, optionally including an O, S, SO, SO2, or NR<7> group or a saturated or unsaturated carbocyclic ring comprising three to seven carbon atoms, or substituted with (C1-C3) alkyl, (C2-C4) alkenyl, phenyl, (C3-C8) cycloalkyl, hydroxy, halo, or (C1-C4) acyl; and Ar is 1,3-benzodioxolyl fluorenyl, pyridyl, imidazolyl, indolyl, thienyl, optionally substituted with CH3 or Cl, thiazolyl, cyclopentyl, 1-methylcyclopentyl, cyclohexenyl (hexahydrophenyl), cyclohexyl (tetrahydrophenyl), naphthyl, dihydronaphthyl, tetrahydronaphthyl, decahydronaphthyl, or a group of the formula (2): where R<1><0> to R<1><4> are independently H, halo, I, (C1-C10) alkyl, branched (C3-C6) alkyl, halo (C1-C4) alkyl, (C1-C4) alkoxy, halo (C1-C4) alkoxy, phenoxy, substituted phenoxy, phenylthio, substituted phenylthio, phenyl, substituted phenyl, NO2, NH2, acetoxy, OH, CN, or SiR<1><5>R<1><6>R<1><7>, OSir<1><5>, R<1><6>, R<1><7>, where R<1><5>, R<1><6>, and R<1><7> are independently (C1-C4) alkyl or (C3-C4) branched alkyl, provided that unless each of R<1><0> to R<1><4> is F, CH3, or H, then at least two of R<1><0> to R<1><4> are H; or an acid addition salt of a compound of formula (1) or an N-oxide of a compound of formula (1) when W is CR<5> are fungicides, insecticides, and miticides.
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Inventors:
Barry Alan Draycorn
Glen Phil Jordan
Robert George Sur
Glen Phil Jordan
Robert George Sur
Application Number:
JP1940289A
Publication Date:
November 12, 1997
Filing Date:
January 27, 1989
Export Citation:
Assignee:
ELI LILLY AND COMPANY
International Classes:
A01N43/42; A01N43/50; A01N43/56; A01N43/58; A01N43/78; C07D215/04; C07D215/12; C07D215/18; C07D215/22; C07D215/233; C07D215/26; C07D237/28; C07D215/36; C07D215/42; C07D215/60; C07D401/12; C07D405/12; C07D409/12; C07D417/12; (IPC1-7): C07D215/04; A01N43/42; A01N43/50; C07D215/18; C07D215/22; C07D215/42; C07D237/28; C07D401/12; C07D405/12; C07D409/12; C07D417/12
Attorney, Agent or Firm:
Aoyama Ryo (1 person outside)