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Title:
5−HT(2B)受容体でアンタゴニスト活性を有する高選択性5−HT(2C)受容体アゴニスト
Document Type and Number:
Japanese Patent JP5810099
Kind Code:
B2
Abstract:
Highly selective 5-HT(2C) receptor agonists receptors are disclosed. The 5-HT(2C) receptor agonists are used in the treatments of disease and conditions wherein modulation of 5-HT(2C) receptors provides a benefit, such as obesity and psychiatric disorders.

Inventors:
Kozykovsky, Alan
Ross, Brian
Sven Nebring, Andrea
Chen, Go
Cho, Song Jin
Application Number:
JP2012552072A
Publication Date:
November 11, 2015
Filing Date:
February 03, 2011
Export Citation:
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Assignee:
THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS
International Classes:
C07C217/74; A61K31/13; A61K45/00; A61P1/04; A61P3/00; A61P3/04; A61P3/06; A61P3/10; A61P7/12; A61P9/00; A61P9/12; A61P15/10; A61P21/00; A61P25/00; A61P25/04; A61P25/06; A61P25/08; A61P25/14; A61P25/16; A61P25/18; A61P25/22; A61P25/24; A61P25/28; A61P25/32; A61P25/36; A61P43/00
Foreign References:
WO2007025144A1
WO2005007614A1
Other References:
Sun Jin Cho et al.,Journal of Medicinal Chemistry,2009年,Vol.52,p.1885-1902
Ulf Appelberg et al.,Bioorganic & Medicinal Chemistry Letters,1996年,Vol.6, No.4,p.415-420
Attorney, Agent or Firm:
Patent business corporation Yuko patent office



 
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