Login| Sign Up| Help| Contact|

Patent Searching and Data


Title:
環式アミンアザヘテロ環式カルボキサミド
Document Type and Number:
Japanese Patent JP6616390
Kind Code:
B2
Abstract:
The invention provides novel cyclic amine azaheterocyclic carboxamide according to Formula (I), Formula (II) and Formula (III) their manufacture and use for the treatment of hyperproliferative diseases, such as cancer.

Inventors:
Bayyard Earl Hack
Shaolin Chen
Constantine Nigue
Reynard Jones
You Fan Xiao
Igor Mocharkin
Application Number:
JP2017242915A
Publication Date:
December 04, 2019
Filing Date:
December 19, 2017
Export Citation:
Click for automatic bibliography generation   Help
Assignee:
Merck Patent Gesellschaft mit beschraenkter Haftung
International Classes:
C07D401/12; A61K31/4709; A61P1/18; A61P3/10; A61P13/08; A61P13/12; A61P17/00; A61P17/06; A61P25/00; A61P25/04; A61P27/02; A61P29/00; A61P35/00; A61P43/00
Domestic Patent References:
JP5642714B2
JP6014034B2
JP5894157B2
Foreign References:
EP0339768A1
WO2008049047A2
WO2004014861A1
WO2001083456A1
WO1999009024A1
WO1997003069A1
Other References:
Journal of Medicinal Chemistry,1995年,38(14),2748-2762
Journal of Molecular Graphics and Modelling,2008年,27(3),233-243
Attorney, Agent or Firm:
Atsushi Aoki
Shinji Mitsuhashi
Yoichi Watanabe
Masaru Nakajima
Ryotaro Takei
Takahide Sasaki