Title:
【発明の名称】アンドロゲンとしての14β,17α-ヒドロキシメチルアンドロスタン誘導体
Document Type and Number:
Japanese Patent JP2002539135
Kind Code:
A
Abstract:
Androgenic steroids having a (14beta,17alpha-)-17-(hydroxymetheyl) configuration, useful for the preparation of male contraceptives and pharmaceutical formulations for the treatment of androgen insufficiency.
Inventors:
Rosen, Hubert Jan Josef
Reisen, Derke
Juan, Del Row Jaap
Reisen, Derke
Juan, Del Row Jaap
Application Number:
JP2000604054A
Publication Date:
November 19, 2002
Filing Date:
March 02, 2000
Export Citation:
Assignee:
Akzo Novel N B
International Classes:
A61K31/565; A61K31/57; A61P5/26; A61P15/16; C07J3/00; C07J5/00; A61K31/568; C07J15/00; C07J53/00; (IPC1-7): C07J3/00; A61K31/568; A61K31/57; A61P5/26; A61P15/16; C07J5/00
Domestic Patent References:
| JPS63216895A | 1988-09-09 |
Foreign References:
| WO1993015104A1 | 1993-08-05 | |||
| US3086027A | 1963-04-16 |
Other References:
JPN5002004261, Ｍ．ＯＫＡＤＡ, ＣＨＥＭＩＣＡＬ ＡＮＤ ＰＨＡＲＭＡＣＥＵＴＩＣＡＬ ＢＵＬＬＥＴＩＮ, 1968, Ｖ１６ Ｎ１１, Ｐ２２２３−２２２７
JPN6010041663, ＣＲＡＢＢＥ， Ｐ．, "Ｓｔｅｒｏｉｄｓ． ＣＣＣＩＸ． Ｓｙｎｔｈｅｓｉｓ ｏｆ ｎｅｗ ｓｔｅｒｏｉｄｓ ｗｉｔｈ ｕｎｎａｔｕｒａｌ ｃｏｎｆｉｇｕｒａｔｉｏｎ", Ｃａｎａｄｉａｎ Ｊｏｕｒｎａｌ ｏｆ Ｃｈｅｍｉｓｔｒｙ, 1968, ４６（３）, ｐ． ３４９−３６３
JPN6010041664, ＳＨＯＰＰＥＥ， Ｃ． Ｗ．, "Ｓｔｅｒｏｉｄｓ． Ｐａｒｔ ＸＶＩＩ． Ｔｈｅ Ｓｔｒｕｃｔｕｒｅ ｏｆ Ｄｉｇｉｎｉｎ ａｎｄ Ｄｉｇｉｎｉｇｅｎｉｎ", Ｊｏｕｒｎａｌ ｏｆ ｔｈｅ Ｃｈｅｍｉｃａｌ Ｓｏｃｉｅｔｙ, 1962, ｐ． ３６１０−３６２４
JPN5002004262, Ｃ．Ｗ．ＳＨＯＰＰＥＥ, ＨＥＬＶＥＴＩＣＡ ＣＨＩＭＩＣＡ ＡＣＴＡ, 1944, Ｖ２７, Ｐ２４６−２６０, CH
JPN5002004263, Ｄ．Ｈ．ＢＡＲＴＯＮ, ＪＯＵＲＮＡＬ ＯＦ ＴＨＥ ＣＨＥＭＩＣＡＬ ＳＯＣＩＥＴＹ, 19570601, Ｎ６, Ｐ２６９８−２７０６, GB
JPN6010041663, ＣＲＡＢＢＥ， Ｐ．, "Ｓｔｅｒｏｉｄｓ． ＣＣＣＩＸ． Ｓｙｎｔｈｅｓｉｓ ｏｆ ｎｅｗ ｓｔｅｒｏｉｄｓ ｗｉｔｈ ｕｎｎａｔｕｒａｌ ｃｏｎｆｉｇｕｒａｔｉｏｎ", Ｃａｎａｄｉａｎ Ｊｏｕｒｎａｌ ｏｆ Ｃｈｅｍｉｓｔｒｙ, 1968, ４６（３）, ｐ． ３４９−３６３
JPN6010041664, ＳＨＯＰＰＥＥ， Ｃ． Ｗ．, "Ｓｔｅｒｏｉｄｓ． Ｐａｒｔ ＸＶＩＩ． Ｔｈｅ Ｓｔｒｕｃｔｕｒｅ ｏｆ Ｄｉｇｉｎｉｎ ａｎｄ Ｄｉｇｉｎｉｇｅｎｉｎ", Ｊｏｕｒｎａｌ ｏｆ ｔｈｅ Ｃｈｅｍｉｃａｌ Ｓｏｃｉｅｔｙ, 1962, ｐ． ３６１０−３６２４
JPN5002004262, Ｃ．Ｗ．ＳＨＯＰＰＥＥ, ＨＥＬＶＥＴＩＣＡ ＣＨＩＭＩＣＡ ＡＣＴＡ, 1944, Ｖ２７, Ｐ２４６−２６０, CH
JPN5002004263, Ｄ．Ｈ．ＢＡＲＴＯＮ, ＪＯＵＲＮＡＬ ＯＦ ＴＨＥ ＣＨＥＭＩＣＡＬ ＳＯＣＩＥＴＹ, 19570601, Ｎ６, Ｐ２６９８−２７０６, GB
Attorney, Agent or Firm:
Yoshio Kawaguchi (5 outside)