Title:
ドーパミンD3受容体のモジュレーターとしての3-(1,2,4-トリアゾール-3-イルアルキル)アザビシクロ(3.1.0)ヘキサン誘導体
Document Type and Number:
Japanese Patent JP5150481
Kind Code:
B2
Abstract:
The present invention relates to novel compounds of formula (I) or pharmaceutically acceptable salt thereof: processes for their preparation, intermediates used in these processes, pharmaceutical compositions containing them and their use in therapy, as modulators of dopamine D3 receptors, e.g. to treat drug dependency, as antipsychotic agents, to treat obsessive compulsive spectrum disorders, premature ejaculation or cognition impairment.
Inventors:
Giorgio Bonanomi
Anna Kecchia
Elleta Fazzolari
Dieter Humprecht
Fabrizio Micheli
Luca Tarsi
Sylvia Terreni
Anna Kecchia
Elleta Fazzolari
Dieter Humprecht
Fabrizio Micheli
Luca Tarsi
Sylvia Terreni
Application Number:
JP2008505840A
Publication Date:
February 20, 2013
Filing Date:
April 12, 2006
Export Citation:
Assignee:
GLAXO GROUP LIMITED
International Classes:
C07D401/14; C07D403/06; C07D403/14; C07D405/14; C07D409/14; C07D413/14; C07D417/14; A61K31/4196; A61K31/422; A61K31/427; A61K31/4439; A61K31/497; A61K31/501; A61P15/08; A61P25/16; A61P25/18; A61P25/20; A61P25/22; A61P25/24; A61P25/28; A61P25/30; A61P25/32; A61P25/34; A61P25/36; A61P43/00
Domestic Patent References:
JP2004513946A | ||||
JP9506346A | ||||
JP2002534519A | ||||
JP58013568A |
Foreign References:
WO2005080382A1 | ||||
WO2006133946A1 |
Attorney, Agent or Firm:
Mitsuo Tanaka
Hiroshi Yamazaki
Kenji Tomita
Hiroshi Yamazaki
Kenji Tomita