Login| Sign Up| Help| Contact|

Patent Searching and Data


Title:
ドーパミンD3受容体のモジュレーターとしての3-(1,2,4-トリアゾール-3-イルアルキル)アザビシクロ(3.1.0)ヘキサン誘導体
Document Type and Number:
Japanese Patent JP5150481
Kind Code:
B2
Abstract:
The present invention relates to novel compounds of formula (I) or pharmaceutically acceptable salt thereof: processes for their preparation, intermediates used in these processes, pharmaceutical compositions containing them and their use in therapy, as modulators of dopamine D3 receptors, e.g. to treat drug dependency, as antipsychotic agents, to treat obsessive compulsive spectrum disorders, premature ejaculation or cognition impairment.

Inventors:
Giorgio Bonanomi
Anna Kecchia
Elleta Fazzolari
Dieter Humprecht
Fabrizio Micheli
Luca Tarsi
Sylvia Terreni
Application Number:
JP2008505840A
Publication Date:
February 20, 2013
Filing Date:
April 12, 2006
Export Citation:
Click for automatic bibliography generation   Help
Assignee:
GLAXO GROUP LIMITED
International Classes:
C07D401/14; C07D403/06; C07D403/14; C07D405/14; C07D409/14; C07D413/14; C07D417/14; A61K31/4196; A61K31/422; A61K31/427; A61K31/4439; A61K31/497; A61K31/501; A61P15/08; A61P25/16; A61P25/18; A61P25/20; A61P25/22; A61P25/24; A61P25/28; A61P25/30; A61P25/32; A61P25/34; A61P25/36; A61P43/00
Domestic Patent References:
JP2004513946A
JP9506346A
JP2002534519A
JP58013568A
Foreign References:
WO2005080382A1
WO2006133946A1
Attorney, Agent or Firm:
Mitsuo Tanaka
Hiroshi Yamazaki
Kenji Tomita



 
Previous Patent: JPS5150480

Next Patent: 排気ガス浄化装置