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Title:
炎症性疾患の治療のためのPDE4インヒビターとしての6-ヘテロアリール-1,2,3,4,4a,10b-ヘキサヒドロフェナントリジン
Document Type and Number:
Japanese Patent JP2008531654
Kind Code:
A
Abstract:
Compounds of a certain formula I in which R1, R2, R3, R31, R4, R5, R51 and Har have the meanings indicated in the description, are novel effective PDE4 inhibitors.

Inventors:
Ulrich Kautz
Beate Schmidt
Dieter Frocker Tsi
Maria Vittoria Chiesa
Armin Hazelmann
Christoph Zitt
Andrea Wolsen
Degenhard Marx
Hans-Peter Cry
Application Number:
JP2007557506A
Publication Date:
August 14, 2008
Filing Date:
March 01, 2006
Export Citation:
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Assignee:
Nycomed GmbH
International Classes:
C07D401/04; A61K31/473; A61K31/501; A61K31/506; A61P11/00; C07D401/14; A61P1/04; A61P3/10; A61P9/00; A61P9/04; A61P11/02; A61P11/04; A61P11/06; A61P13/02; A61P13/12; A61P15/10; A61P17/00; A61P17/02; A61P17/06; A61P17/08; A61P17/14; A61P19/02; A61P19/10; A61P25/00; A61P25/16; A61P25/24; A61P25/28; A61P27/14; A61P29/00; A61P35/02; A61P37/00; A61P37/08; A61P43/00
Attorney, Agent or Firm:
Toshio Yano
Toshiomi Yamazaki
Takuya Kuno
Hiroshi Sugimoto
Kimihiro Hoshi
Hiroyasu Ninomiya
Einzel Felix-Reinhard
Reinhard Einsel