メラノコルチン-4受容体作働薬としてのアシル化ピペリジン誘導体

Japanese Patent JP2009510069

A

Certain novel 4 alkyl substituted N acylated piperidine derivatives are ligands of the human melanocortin receptor(s) and, in particular, are selective ligands of the human melanocortin-4 receptor (MC-4R). They are therefore useful for the treatment, control, or prevention of diseases and disorders responsive to the modulation of MC-4R, such as obesity, diabetes, nicotine addiction, alcoholism, sexual dysfunction, including erectile dysfunction and female sexual dysfunction.

JPS6344561	N-(SUBSTITUTED CYCLIC ALKYLENEIMINE)-ALPHA-(3, 5-DIALKYL-4-HYDROXYPHENYL)-ALPHA', ALPHA"-DIALKYLACETAMIDE, ITS PRODUCTION AND STABILIZED COMPOSITION CONTAINING THE SAME
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JP2010507643	A novel phenylsulfamoylbenzamide derivative as a bradykinin antagonist

Bakushi, Rahman, Kay
Hong, Kinmei
Nagand, Ravi, Pea

JP2008533478A

March 12, 2009

September 26, 2006

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MERCK & COMPANY INCOPORATED

C07D211/26; A61K31/445; A61K31/4525; A61K31/453; A61K31/454; A61K31/4545; A61K31/4709; A61K31/496; A61K31/5377; A61P1/04; A61P1/16; A61P3/00; A61P3/04; A61P3/06; A61P3/10; A61P9/04; A61P9/06; A61P9/10; A61P9/12; A61P11/00; A61P11/06; A61P13/12; A61P15/06; A61P15/08; A61P15/10; A61P17/10; A61P17/16; A61P19/02; A61P19/06; A61P25/00; A61P25/20; A61P25/22; A61P25/24; A61P25/28; A61P25/30; A61P25/32; A61P25/34; A61P29/00; A61P31/18; A61P35/00; A61P35/02; A61P43/00; C07D211/38; C07D401/12; C07D405/12; C07D413/12; C07D417/12; C07D491/08

Kenichi Osawa
Kenji Ando

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