Title:
17α-ALKYL-17β-OXY-ESTRATRIENES, INTERMEDIATE PRODUCTS FOR THEIR PRODUCTION AND USE OF THE 17α-ALKYL-17β-OXY-ESTRATRIENES FOR PRODUCING PHARMACEUTICAL AGENT AND PHARMACEUTICAL PREPARATION
Document Type and Number:
Japanese Patent JP2006306896
Kind Code:
A
Abstract:
To provide a novel compound having an antiestrogenic action.
The novel compound is 17α-alkyl-17β-oxy-estra-1,3,5(10)-triene which is represented by formula I and has an antiestrogenic action. The 17α-alkyl-17β-oxy-estratriene is used for preparing a pharmaceutical agent. A pharmaceutical preparation contains at least one 17α-alkyl-17β-oxy-estratriene and at least one pharmaceutically acceptable vehicle.
Inventors:
BOHLMANN ROLF
HEINRICH NIKOLAUS
JAUTELAT ROLF
KROLL JORG
PETROV ORLIN
REICHEL ANDREAS
HOFFMANN JENS
LICHTNER ROSEMARIE
HEINRICH NIKOLAUS
JAUTELAT ROLF
KROLL JORG
PETROV ORLIN
REICHEL ANDREAS
HOFFMANN JENS
LICHTNER ROSEMARIE
Application Number:
JP2006222528A
Publication Date:
November 09, 2006
Filing Date:
August 17, 2006
Export Citation:
Assignee:
SCHERING AG
International Classes:
A61K31/567; C07J41/00; A61K31/5685; A61K31/569; A61K31/58; A61P5/32; A61P13/08; A61P15/00; A61P15/08; A61P15/12; A61P15/16; A61P15/18; A61P17/14; A61P35/00; C07J1/00; C07J43/00
Domestic Patent References:
JPS6097995A | 1985-05-31 | |||
JP2001503024A | 2001-03-06 | |||
JP2000510861A | 2000-08-22 | |||
JP2001527088A | 2001-12-25 |
Attorney, Agent or Firm:
Atsushi Aoki
Takashi Ishida
Fukumoto product
Tetsuji Koga
Kazuhiro Nakamura
Takashi Ishida
Fukumoto product
Tetsuji Koga
Kazuhiro Nakamura
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