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Title:
ALLOSTERIC CHROMENONE INHIBITORS OF PHOSPHOINOSITIDE 3-KINASE (PI3K) FOR TREATMENT OF DISEASE
Document Type and Number:
Japanese Patent JP2023164409
Kind Code:
A
Abstract:
To provide compounds as allosteric chromenone inhibitors of phosphoinositide 3 kinase (PI3K) useful in treatment of diseases or disorders associated with PI3K modulation.SOLUTION: The disclosure relates to compounds of Formula (I) or pharmaceutically acceptable salts thereof.SELECTED DRAWING: None

Inventors:
SEAN DOUGLAS ARONOW
CARINA IVONNE JETTE
GABRIELLE R KOLAKOWSKI
CHRISTOPHER GLENN MAYNE
WANG HUA-YU
MICHAEL BRIAN WELCH
NATHAN EDWARD WRIGHT
GERIT MARIA POTOTSCHNIG
SUN ZHICHENG
WARREN CHRISTOPHER CHAN
SURENDRA DAWADI
MANOJ KUMAR
KATELYN FRANCES LONG
ALFREDO PICADO
MARCOS ADRIAN SAINZ
TAREK SAMMAKIA
LATOYA DENISE SCAGGS
ERIN DANIELLE ANDERSON
CHEN SHUAI
THOMAS C IRVIN
EDWARD A KESICKI
GANESH MANGALSING MURHADE
WANG XIA
Application Number:
JP2023075096A
Publication Date:
November 10, 2023
Filing Date:
April 28, 2023
Export Citation:
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Assignee:
PETRA PHARMA CORP
International Classes:
C07D311/60; A61K31/352; A61K31/381; A61K31/4245; A61K31/425; A61K31/4433; A61K31/444; A61K31/4545; A61K31/506; A61K31/519; A61K31/5377; A61K31/5383; A61K31/553; A61K31/665; A61P35/00; A61P35/02; A61P35/04; A61P43/00; C07C53/18; C07D405/04; C07D405/12; C07D405/14; C07D409/12; C07D413/04; C07D413/12; C07D417/12; C07D471/04; C07D487/04; C07D491/107; C07D498/04; C07F9/655
Attorney, Agent or Firm:
Norito Yamao
Wu Yingyan
Wataru Sato
Nagatoshi Shinagawa