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Title:
アルファヒドロキシアミド
Document Type and Number:
Japanese Patent JP2015535832
Kind Code:
A
Abstract:
本発明は、式Iで表される化合物および関連化合物を含むアルファヒドロキシアミド、ならびに、炎症性の障害および疾患の予防および処置におけるそれらの使用に関し、式中T1、T2、WおよびRwは請求項1に与えられた意味を有する。

Inventors:
Muzel, Matilde
Swinen, Dominique
Sini Sammy, Jayapurashnarayanan
Application Number:
JP2015533473A
Publication Date:
December 17, 2015
Filing Date:
September 10, 2013
Export Citation:
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Assignee:
Merck Patent Gesellschaft mit beschraenkter Haftung
International Classes:
C07C235/06; A61K31/16; A61K31/17; A61K31/18; A61K31/195; A61K31/223; A61K31/235; A61K31/24; A61K31/277; A61K31/341; A61K31/381; A61K31/4409; A61K31/445; A61K31/4453; A61K31/4468; A61K31/453; A61K31/454; A61K31/495; A61K31/5375; A61K45/00; A61P1/04; A61P3/10; A61P7/00; A61P7/04; A61P9/00; A61P9/10; A61P11/00; A61P13/12; A61P15/00; A61P17/00; A61P17/06; A61P19/02; A61P19/08; A61P19/10; A61P25/00; A61P25/28; A61P27/02; A61P29/00; A61P31/04; A61P35/00; A61P35/02; A61P37/02; A61P37/06; A61P37/08; A61P43/00; C07C235/10; C07C237/12; C07C237/22; C07C237/42; C07C255/54; C07C311/04; C07C317/22; C07C317/32; C07D211/26; C07D211/58; C07D211/96; C07D213/68; C07D265/32; C07D295/08; C07D295/12; C07D295/18; C07D295/22; C07D307/14; C07D333/20; C07D401/12; C07D405/12
Domestic Patent References:
JPS60248193A1985-12-07
JPS60248193A1985-12-07
Foreign References:
WO2011152720A12011-12-08
US2692895A1954-10-26
WO2011152720A12011-12-08
US2692895A1954-10-26
Other References:
LUTZ, R. E.ET AL., JOURNAL OF ORGANIC CHEMISTRY, vol. Vol. 12, JPN6017023695, 1947, pages pp. 96-107
BULLER, A. R. ET AL., JOURNAL OF MOLECULAR BIOLOGY, vol. Vol. 422, JPN6017023696, 2012, pages pp. 508-518
LUTZ, R. E.ET AL., JOURNAL OF ORGANIC CHEMISTRY, vol. Vol. 12, JPN6017023695, 1947, pages pp. 96-107
BULLER, A. R. ET AL., JOURNAL OF MOLECULAR BIOLOGY, vol. Vol. 422, JPN6017023696, 2012, pages pp. 508-518
Attorney, Agent or Firm:
Kiyoji Kuzuwa