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Title:
GABA類似体の全身濃度が持続するアミノ酸コンジュゲート
Document Type and Number:
Japanese Patent JP2005501013
Kind Code:
A
Abstract:
Compounds that provide for sustained systemic concentrations of GABA analogs following oral administration to animals are disclosed. Pharmaceutical compositions including, and methods using, such compounds are also disclosed.

Inventors:
Gallop, Mark A.
Kandy, Kenneth See
Schuurman, Randall A
Barrett, Ronald W.
Zelange, Noah
Application Number:
JP2003503171A
Publication Date:
January 13, 2005
Filing Date:
June 11, 2002
Export Citation:
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Assignee:
Zenoport, Inc.
International Classes:
C07D295/18; A61K31/197; A61K31/198; A61K31/275; A61K31/381; A61K31/40; A61K31/426; A61K31/4402; A61K31/4406; A61K31/4409; A61K31/4453; A61K31/4458; A61K31/47; A61K47/48; A61P1/00; A61P25/00; A61P25/04; A61P25/08; A61P25/18; A61P25/20; A61P25/22; A61P25/24; A61P25/28; A61P25/32; A61P29/00; A61P43/00; C07C237/12; C07C237/20; C07C237/24; C07C255/58; C07C317/50; C07C323/59; C07C323/60; C07D207/16; C07D211/60; C07D213/53; C07D213/56; C07D215/12; C07D229/02; C07D233/54; C07D277/20; C07D277/30; C07D333/24; C07D333/60; C07K5/02; G01N33/566; A61K38/00; (IPC1-7): C07C237/12; A61K31/197; A61K31/198; A61K31/275; A61K31/381; A61K31/40; A61K31/426; A61K31/4402; A61K31/4406; A61K31/4409; A61K31/4453; A61K31/4458; A61K31/47; A61P1/00; A61P25/00; A61P25/04; A61P25/08; A61P25/18; A61P25/20; A61P25/22; A61P25/24; A61P25/28; A61P25/32; A61P29/00; A61P43/00; C07C237/20; C07C237/24; C07C255/58; C07D211/60; C07D213/53; C07D213/56; C07D215/12; C07D277/20; C07D277/30; C07D295/18; C07D333/24; C07D333/60
Attorney, Agent or Firm:
Shoichi Okuyama
Arihara Koichi
Matsushima Tetsuo