Title:
抗生物質の調製物、該調製物の使用およびその製造方法
Document Type and Number:
Japanese Patent JP4181331
Kind Code:
B2
Abstract:
An amphiphilic organic sulfate, sulfamate, sulfonate, disulfate, disulfonate or trisulfonate is included in an aminoglycoside, lincosamide, 4-quinolone or tetracycline antibiotic preparation to retard the release of the antibiotic from the preparation. An antibiotic preparation comprises a mixture of an amphiphilic component consisting of one or more alkyl, aryl, alkylaryl, cycloalkyl or alkylcycloalkyl sulfates, sulfamates or sulfonates, fatty acid-2-sulfonates, alkyl or cycloalkyl disulfates, alkyl, cycloalkyl, aryl or alkylaryl disulfonates or aryl or alkylaryl trisulfonates and one or more aminoglycoside, lincosamide, 4-quinolone or tetracycline antibiotics.
Inventors:
Sebastian Voigt
Matthias Schnaberlauf
Claus-Dieeter Kien
Matthias Schnaberlauf
Claus-Dieeter Kien
Application Number:
JP2002081307A
Publication Date:
November 12, 2008
Filing Date:
March 22, 2002
Export Citation:
Assignee:
Heraeus Kulzer GmbH
International Classes:
A61K47/20; A61K9/00; A61K9/10; A61K9/14; A61K9/22; A61K9/70; A61K31/00; A61K31/70; A61K31/7036; A61K31/726; A61K45/06; A61K45/08; A61K47/02; A61K47/14; A61K47/16; A61K47/24; A61L27/54; A61L31/16; A61P31/04; A61K9/20
Domestic Patent References:
JP53041418A | ||||
JP63307815A | ||||
JP6298639A | ||||
JP9030988A | ||||
JP10033657A |
Foreign References:
US5035891 | ||||
EP0052916A1 | ||||
US5670142 | ||||
GB1120992B |
Attorney, Agent or Firm:
Toshio Yano
Toshiomi Yamazaki
Takuya Kuno
Einzel Felix-Reinhard
Toshiomi Yamazaki
Takuya Kuno
Einzel Felix-Reinhard