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Title:
Bisphosphonate prodrug
Document Type and Number:
Japanese Patent JP6029596
Kind Code:
B2
Abstract:
The present invention relates to a prodrug, comprising a pharmaceutically and/or diagnostically active compound, and one or more bisphosphonate groups, to a process for producing such a prodrug, and to a pharmaceutical composition comprising said prodrug, to be used for the treatment of bone-related disorders such as bone cancer.

Inventors:
Kratz Felix
Hochdelfer Katrin
Application Number:
JP2013554818A
Publication Date:
November 24, 2016
Filing Date:
February 24, 2012
Export Citation:
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Assignee:
Kate bates morfolsungs gezelshaft mitt beschlenktel haftung
International Classes:
A61K47/48; A61K31/663; A61K31/704; A61K45/00; A61P19/08; A61P35/00; A61P35/04; A61P43/00
Domestic Patent References:
JP2009505974A
JP8501546A
Foreign References:
WO2009083614A1
Other References:
Bioorganic & Medicinal Chemistry Letters,2008年,Vol.18,p.816-820
Biomacromolecules,2005年,Vol.6,p.2800-2808
Calcified Tissue International,1996年,Vol.59,p.168-173
Pharmaceutical Research,2001年,Vol.18, No.5,p.646-651
Journal of Applied Polymer Science,2006年,Vol.101,p.3192-3201
Attorney, Agent or Firm:
Patent Business Corporation Saegusa International Patent Office