Title:
眼の疾患及び障害を治療する化合物
Document Type and Number:
Japanese Patent JP5773877
Kind Code:
B2
Abstract:
Provided are compounds, pharmaceutical compositions thereof, and methods of treating ophthalmic diseases and disorders, such as age-related macular degeneration and Stargardt's Disease, using said compounds and compositions.
Inventors:
Scott, Ian Elle.
Kukusa, Vladimir A.
Hong, phone
Ryo Kubota
Gauge, jennifer
Kukusa, Vladimir A.
Hong, phone
Ryo Kubota
Gauge, jennifer
Application Number:
JP2011533310A
Publication Date:
September 02, 2015
Filing Date:
October 21, 2009
Export Citation:
Assignee:
Accusera Inc.
International Classes:
C07C211/49; A61K31/137; A61K31/167; A61K31/17; A61K31/18; A61K31/426; A61P9/00; A61P9/10; A61P27/02; A61P43/00; C07C215/08; C07C215/10; C07C215/68; C07C215/70; C07C217/30; C07C217/76; C07C225/22; C07C233/07; C07C233/62; C07C275/40; C07C311/08; C07C311/14; C07C311/21; C07C311/24; C07C335/18; C07D277/28
Domestic Patent References:
| JP8012579A | ||||
| JP2006502118A | ||||
| JP2006505511A | ||||
| JP2006501195A | ||||
| JP2007536280A | ||||
| JP2006508101A | ||||
| JP2004535390A | ||||
| JP2003518057A | ||||
| JP10510248A | ||||
| JP2008500284A |
Foreign References:
| US20030216456 | ||||
| GB1108577A | ||||
| WO2004033419A1 | ||||
| US20030100580 | ||||
| US3341584 |
Other References:
R.J. ALTENBACH, ET AL,Synthesis and structure-activity studies on N-(5-(1H-imidazol-4-yl)-5 ,6,7,8-tetrahydro-1-naphthalenyl)methanesu lfonamide, an imidazole-containing alpha1A-adrenoceptor agonist,JOURNAL OF MEDICINAL CHEMISTRY,2004年,47,3220-3235
Sikazwe, Donald; Bondarev, Mikhail L.; Dukat, Malgorzata; Rangisetty, Jagadeesh B.; Roth, Bryan L.; Glennon, Richard A.,Binding of Sulfonyl-Containing Arylalkylamines at Human 5-HT6 Serotonin Receptors,Journal of Medicinal Chemistry ,2006年,49(17),5217-5225
WASHBURN W. N. ET AL,Arylpropanolamines: Selective .beta.3 agonists arising from strategies to mitigate phase I metabolic transformations,BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS,2007年,17,4290-4296
Sikazwe, Donald; Bondarev, Mikhail L.; Dukat, Malgorzata; Rangisetty, Jagadeesh B.; Roth, Bryan L.; Glennon, Richard A.,Binding of Sulfonyl-Containing Arylalkylamines at Human 5-HT6 Serotonin Receptors,Journal of Medicinal Chemistry ,2006年,49(17),5217-5225
WASHBURN W. N. ET AL,Arylpropanolamines: Selective .beta.3 agonists arising from strategies to mitigate phase I metabolic transformations,BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS,2007年,17,4290-4296
Attorney, Agent or Firm:
Asamura patent office