Title:
ＴＲＰＶ１阻害活性を有する化合物とその使用
Document Type and Number:
Japanese Patent JP5876423
Kind Code:
B2
Abstract:
The invention relates to compounds of Formula I and pharmaceutically acceptable derivatives thereof, compositions comprising an effective amount of a compound of Formula I or a pharmaceutically acceptable derivative thereof, and methods for treating or preventing a condition such as pain, UI, an ulcer, IBD and IBS, comprising administering to an animal in need thereof an effective amount of a compound of Formula I or a pharmaceutically acceptable derivative thereof.
Inventors:
Noriyuki Kurose
Application Number:
JP2012556732A
Publication Date:
March 02, 2016
Filing Date:
June 22, 2011
Export Citation:
Assignee:
Shionogi Pharmaceutical Co., Ltd.
International Classes:
C07D401/14; A61K31/444; A61K31/4545; A61K31/496; A61K31/55; A61P1/04; A61P13/02; A61P29/00; C07D401/04; C07D417/12; C07D417/14; C07D487/08
Domestic Patent References:
| JP2006528642A | ||||
| JP2006528643A | ||||
| JP2009516729A |
Foreign References:
| WO2008132600A1 | ||||
| WO2003089410A1 |
Other References:
Martin J. Gunthorpe et al.,Characterization of SB-705498, a Potent and Selective Vanilloid Receptor-1 (VR1/TRPV1) Antagonist That Inhibits the Capsaicin-, Acid-, and Heat-Mediated Activation of the Receptor,The Journal of Pharmacology and Experimental Therapeutics,2007年,321(3),p. 1183-1192
Attorney, Agent or Firm:
Kyousei Tamura
Samejima Mutsumi
Masahiro Nitta
Kure Hidenori
Samejima Mutsumi
Masahiro Nitta
Kure Hidenori
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