Title:
エナンチオ選択的合成
Document Type and Number:
Japanese Patent JP4461048
Kind Code:
B2
Abstract:
A short practical commercial process for the efficient enantioselective synthesis of the non-steroidal antiestrogen of formula (I) or (XIV) or a pharmaceutically acceptable salt thereof.
Inventors:
Richard W. Draper
Ladabuy. Yale
Yuri Lou
Eugene Jay Beater
Ladabuy. Yale
Yuri Lou
Eugene Jay Beater
Application Number:
JP2005112900A
Publication Date:
May 12, 2010
Filing Date:
April 08, 2005
Export Citation:
Assignee:
Schering Corporation
International Classes:
A61K31/352; C07D311/04; A61P5/32; C07D311/26; C07B57/00; C07B61/00; C07D311/60
Domestic Patent References:
| JP7188008A |
Foreign References:
| WO1996026201A1 | ||||
| WO1999063974A1 | ||||
| US5254568 | ||||
| US5395842 | ||||
| WO1999002512A1 | ||||
| WO1999002513A1 |
Other References:
J. Med. Chem.,1997年 7月 4日,Vol.40,No.14,pp.2117-2122
J.Med.Chem.,1990年,Vol.33,No.12,pp.3222-3229
Bioorg. Med. Chem.,1995年,Vol.3,No.11,pp.1417-1421
Bioorg. Med. Chem.,1997年,Vol.7,No.16,pp.2131-2136
Tetrahedron Letters,1995年,Vol.36,No.49,pp.8913-8916
Eur. J. Med. Chem.,1997年,Vol.32,pp.135-142
J.Med.Chem.,1990年,Vol.33,No.12,pp.3222-3229
Bioorg. Med. Chem.,1995年,Vol.3,No.11,pp.1417-1421
Bioorg. Med. Chem.,1997年,Vol.7,No.16,pp.2131-2136
Tetrahedron Letters,1995年,Vol.36,No.49,pp.8913-8916
Eur. J. Med. Chem.,1997年,Vol.32,pp.135-142
Attorney, Agent or Firm:
Hidesaku Yamamoto
Takaaki Yasumura
Natsuki Morishita
Takaaki Yasumura
Natsuki Morishita